Synthesis and antibacterial activity of acylides (3-O-acyl-erythromycin derivatives): A novel class of macrolide antibiotics

Journal of Medicinal Chemistry

Volumn 44, Issue 24, 2001, Pages 4027-4030

  Tanikawa, T ^a,b   Asaka, T ^a   Kashimura, M ^a   Misawa, Y ^a   Suzuki, K ^a   Sato, M ^a   Kameot, K ^a   Morimoto, S ^a   Nishida, A ^b  

^a TAISHO PHARMACEUTICAL CO LTD   (Japan)

^b CHIBA UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

3 O ACYL ERYTHROMYCIN DERIVATIVE; ACYLIDE DERIVATIVE; AZITHROMYCIN; CLARITHROMYCIN; ERYTHROMYCIN DERIVATIVE; LINCOSAMIDE; MACROLIDE; MIKAMYCIN B; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIBIOTIC RESISTANCE; ARTICLE; DRUG POTENCY; DRUG SYNTHESIS; GRAM POSITIVE BACTERIUM; MINIMUM INHIBITORY CONCENTRATION; STAPHYLOCOCCUS AUREUS; STREPTOCOCCUS PNEUMONIAE;

ANIMALS; ANTI-BACTERIAL AGENTS; ENTEROCOCCUS FAECALIS; ENTEROCOCCUS FAECIUM; ERYTHROMYCIN; MICE; MICROBIAL SENSITIVITY TESTS; STAPHYLOCOCCAL INFECTIONS; STAPHYLOCOCCUS AUREUS; STREPTOCOCCUS PNEUMONIAE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035935698     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm015566s     Document Type: Article

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