Synthesis and antibacterial activity of the tricyclic Ketolides TE-802 and its analogs

Journal of Antibiotics

Volumn 54, Issue 8, 2001, Pages 664-678

  Kashimura, M ^a   Asaka, T ^a   Misawa, Y ^a   Matsumoto, K ^a   Morimoto, S ^a  

^a TAISHO PHARMACEUTICAL CO LTD   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

11 AMINO 9 DEOXO 11 DEOXY 9,11 NITRILOETHANO 5 O DESOSAMINYL 6 O METHYLERYTHRONOLIDE A 11,12 CYCLIC CARBAMATE; 11 AMINO 9 DEOXO 11 DEOXY 9,11 NITRILOETHANO 6 O METHYLERYTHROMYCIN A 11,12 CYCLIC CARBAMATE; 11 AMINO 9 DEOXO 3,11 DIDEOXY 9 N,11 N ETHANO 3 OXO 5 O DESOSAMINYL 6 O METHYLERYTHRONOLIDE A 9 AMINE 11,12 CYCLIC CARBAMATE; 11 AMINO 9 DEOXO 3,11 DIDEOXY 9,11 N (2,2 DIMETHYL)NITRILOETHANO 3 OXO 5 O DESOSAMINYL 6 O METHYLERYTHRONOLIDE A 11,12 CYCLIC CARBAMATE; 11 AMINO 9 DEOXO 3,11 DIDEOXY 9,11 N METHYLNITRILOETHANO 3 OXO 5 O DESOSAMINYL 6 O METHYLERYTHRONOLIDE A 11,12 CYCLIC CARBAMATE; 11 AMINO 9 DEOXO 3,11 DIDEOXY 9,11 N NITRILOETHANO 3 OXO 5 O DESOSAMINYL 6 O METHYLERYTHRONOLIDE A 11,12 CYCLIC CARBAMATE; 9,11 DIAZAHEPTENE; AZITHROMYCIN; CARBAMIC ACID DERIVATIVE; CETHROMYCIN; CLARITHROMYCIN; ERYTHROMYCIN; KETOLIDE; KETOLIDE DERIVATIVE; MACROLIDE; ROXITHROMYCIN; TE 802; TELITHROMYCIN; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIBIOTIC SENSITIVITY; ARTICLE; CHEMICAL REACTION; CONTROLLED STUDY; CYCLIZATION; DEHYDRATION; DRUG BIOAVAILABILITY; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; HOSPITAL INFECTION; IN VITRO STUDY; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PRIORITY JOURNAL; RESPIRATORY TRACT INFECTION; STAPHYLOCOCCUS AUREUS; STREPTOCOCCUS PNEUMONIAE;

EID: 0034824275     PISSN: 00218820     EISSN: None     Source Type: Journal    
DOI: 10.7164/antibiotics.54.664     Document Type: Article

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