Conformationally restricted indolopiperidine derivatives as potent CCR2B receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 11, Issue 16, 2001, Pages 2177-2180

  Witherington, Jason ^a   Bordas, Vincent ^a   Cooper, Dave G ^a   Forbes, Ian T ^a   Gribble, Andrew D ^a   Ife, Robert J ^a   Berkhout, Theo ^a   Gohil, Jayneeta ^a   Groot, Pieter H E ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

CHEMOKINE RECEPTOR CCR2B ANTAGONIST; DOPAMINE RECEPTOR; INDOLOPIPERIDINE DERIVATIVE; PIPERIDINE DERIVATIVE; RECEPTOR BLOCKING AGENT; SEROTONIN RECEPTOR; UNCLASSIFIED DRUG;

ARTICLE; DRUG IDENTIFICATION; DRUG POTENCY; DRUG SCREENING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; REACTION ANALYSIS;

DOPAMINE ANTAGONISTS; INDOLES; MOLECULAR CONFORMATION; PIPERIDINES; RECEPTORS, CHEMOKINE; SEROTONIN ANTAGONISTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035921020     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(01)00397-3     Document Type: Article

References (11)