Comparative activities of the enantiomeric GABA B receptor agonists CGP 44532 and 44533 in central and peripheral tissues

European Journal of Pharmacology

Volumn 412, Issue 1, 2001, Pages 27-37

  Ong, Jennifer ^a   Bexis, Sotiria ^a   Marino, Victor ^a   Parker, David A S ^a   Kerr, David I B ^a   Froestl, Wolfgang ^b  

^a UNIVERSITY OF ADELAIDE   (Australia)

^b NOVARTIS PHARMA AG   (Switzerland)

Author keywords

Baclofen; CGP 44532; CGP 44533; GABA B receptor agonist; Guinea pig; Ileum; Rat neocortex

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID B RECEPTOR; 5,5 DIMETHYL 2 MORPHOLINEACETIC ACID; BACLOFEN; CGP 44532; CGP 44533; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENCY; ELECTROSTIMULATION; ENANTIOMER; GABAERGIC TRANSMISSION; GUINEA PIG; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR UPREGULATION; TISSUE SPECIFICITY;

ANIMALS; BACLOFEN; DOSE-RESPONSE RELATIONSHIP, DRUG; GABA AGONISTS; GUINEA PIGS; ILEUM; MALE; NEOCORTEX; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, GABA-B;

EID: 0035910372     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(00)00945-6     Document Type: Article

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