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Journal of Medicinal Chemistry

Volumn 44, Issue 10, 2001, Pages 1623-1626

Combinatorial lead optimization of a neuropeptide FF antagonist

(5) Prokai, L a,b Prokai Tatrai, K b Zharikova, A a Li, X a Rocca, J R b

a Department of Pharmacotherapy and Translational Research (United States)

b UNIVERSITY OF FLORIDA (United States)

Author keywords

[No Author keywords available]

Indexed keywords

5 (DIMETHYLAMINO) 1 NAPHTHALENESULFONYLDANSYLPROLYLGLUTAMYLARGININAMIDE; 5 (DIMETHYLAMINO) 1 NAPHTHALENESULFONYLGLYCYLSERYLARGININAMIDE; NEUROPEPTIDE FF; RECEPTOR BLOCKING AGENT; TRIPEPTIDE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; DOSE RESPONSE; DRUG BINDING; DRUG PENETRATION; DRUG POTENCY; DRUG POTENTIATION; DRUG SOLUBILITY; DRUG STRUCTURE; NONHUMAN; RADIOASSAY; RADIOIODINATION; RAT; RECEPTOR AFFINITY; WITHDRAWAL SYNDROME;

ANIMALS; BINDING, COMPETITIVE; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; COMBINATORIAL CHEMISTRY TECHNIQUES; DANSYL COMPOUNDS; OLIGOPEPTIDES; RADIOLIGAND ASSAY; RATS; RECEPTORS, NEUROPEPTIDE; SPINAL CORD; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035837074 PISSN: 00222623 EISSN: None Source Type: Journal
DOI: 10.1021/jm000512o Document Type: Article

Times cited : (25)

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