Uptake and efflux of the peptidic delta-opioid receptor agonist [D-penicillamine2,5]-enkephalin at the murine blood-brain barrier by in situ perfusion

Neuroscience Letters

Volumn 301, Issue 3, 2001, Pages 155-158

  Dagenais, Claude ^a   Ducharme, Julie ^b,c   Pollack, Gary M ^a  

^a UNIVERSITY OF NORTH CAROLINA   (United States)

^b ASTRAZENECA   (United Kingdom)

^c UNIVERSITÉ DE MONTRÉAL   (Canada)

Author keywords

Blood brain barrier; Delta opioid receptor agonist; Efflux; Inhibitors; Organic anion transporting polypeptide; P glycoprotein; Uptake

Indexed keywords

DELTA OPIATE RECEPTOR AGONIST; DEXVERAPAMIL; DIGOXIN; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; ESTRADIOL 17 GLUCURONIDE; FEXOFENADINE; GLYCOPROTEIN P; LU 33925; MEMBRANE PROTEIN;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BLOOD BRAIN BARRIER; BRAIN PERFUSION; BRAIN TISSUE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG UPTAKE; EFFUSION; MALE; MEMBRANE PERMEABILITY; MEMBRANE TRANSPORT; MOUSE; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; TISSUE LEVEL;

EID: 0035815578     PISSN: 03043940     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0304-3940(01)01640-8     Document Type: Article

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