A new class of cytotoxic DNA minor groove binders: α-halogenoacrylic derivatives of pyrrolecarbamoyl oligomers

Farmaco

Volumn 56, Issue 1-2, 2001, Pages 57-65

  Cozzi, Paolo ^a  

^a UNIVERSITY OF MILAN   (Italy)

Author keywords

Halogenoacrylamides; Distamycin; Glutathione; Minor groove binders; Tallimustine

Indexed keywords

ADOZELESIN; BIZELESIN; BROSTALLICIN; CAMPTOTHECIN; CARZELESIN; CHLORMETHINE DERIVATIVE; CISPLATIN; DISTAMYCIN A; DISTAMYCIN A DERIVATIVE; GLUTATHIONE; MELPHALAN; PNU 151807; PNU 160366; PNU 57911; TALLIMUSTINE; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; BONE MARROW TOXICITY; CANCER CELL; CONFERENCE PAPER; CYTOTOXICITY; DNA ALKYLATION; DRUG DNA INTERACTION; DRUG SYNTHESIS; HEMATOPOIETIC CELL; HUMAN; HUMAN CELL; IN VITRO STUDY; STRUCTURE ACTIVITY RELATION;

ACRYLAMIDES; ALKYLATION; ANTINEOPLASTIC AGENTS; DISTAMYCINS; DNA; GLUTATHIONE; GLUTATHIONE TRANSFERASE; HUMANS; NITROGEN MUSTARD COMPOUNDS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035272741     PISSN: 0014827X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-827X(01)01009-6     Document Type: Conference Paper

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