Affinity of serotonin receptor antagonists and agonists to recombinant and native α1-adrenoceptor subtypes

Japanese Journal of Pharmacology

Volumn 86, Issue 2, 2001, Pages 189-195

  Yoshio, R ^a   Taniguchi, T ^a   Itoh, H ^a   Muramatsu, I ^a  

^a UNIVERSITY OF FUKUI   (Japan)

Author keywords

Selectivity; Serotonin receptor agonist; Serotonin receptor antagonist; 1 adrenoceptor

Indexed keywords

1 (2 METHOXYPHENYL) 4 (4 PHTHALIMIDOBUTYL)PIPERAZINE; 1 [2 (4 AMINOPHENYL)ETHYL] 4 (3 TRIFLUOROMETHYLPHENYL)PIPERAZINE; 2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 5 METHYLURAPIDIL; 8 [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] 8 AZASPIRO[4.5]DECANE 7,9 DIONE; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1A ADRENERGIC RECEPTOR; ALPHA 1B ADRENERGIC RECEPTOR; ALPHA 1D ADRENERGIC RECEPTOR; BEMESETRON; CLOZAPINE; CYANOPINDOLOL; CYPROHEPTADINE; KETANSERIN; METHYSERGIDE; METOCLOPRAMIDE; MIANSERIN; NORADRENALIN BITARTRATE; RAUWOLSCINE; RISPERIDONE; RITANSERIN; SEROTONIN 1A AGONIST; SEROTONIN 1A ANTAGONIST; SEROTONIN 2A ANTAGONIST; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; SEROTONIN CREATININE SULFATE; SPIPERONE; SPIROXATRINE; UNINDEXED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CAROTID ARTERY; COMPARATIVE STUDY; CONCENTRATION RESPONSE; CONTROLLED STUDY; DOG; DRUG SELECTIVITY; IC 50; MALE; NONHUMAN; RAT; RECEPTOR BINDING; TAIL ARTERY; THORACIC AORTA;

EID: 0034937635     PISSN: 00215198     EISSN: None     Source Type: Journal    
DOI: 10.1254/jjp.86.189     Document Type: Article

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