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Volumn 66, Issue 10, 2001, Pages 785-791

Synthesis and biological evaluation of novel daunorubicin-estrogen conjugates

(8) Kasiotis, Konstantinos M a Magiatis, Prokopios b Pratsinis, Harris b Skaltsounis, Alexios Leandros b Abadji, Vasiliki b Charalambous, Avgui c Moutsatsou, Paraskevi b Haroutounian, Serkos A a

a AGRICULTURAL UNIVERSITY OF ATHENS (Greece)

b UNIVERSITY OF ATHENS MEDICAL SCHOOL (Greece)

c ELPEN Pharmaceutical Co Inc (Greece)

Author keywords

Cytotoxic activity; Daunorubicin conjugates; Estrogen receptor binding; Steroidal and non steroidal estrogen ligand; Synthesis

Indexed keywords

DAUNORUBICIN DERIVATIVE; DAUNORUBICIN ESTROGEN CONJUGATE; ESTROGEN; ESTROGEN RECEPTOR; UNCLASSIFIED DRUG;

ADULT; AGED; ANTINEOPLASTIC ACTIVITY; ARTICLE; BINDING AFFINITY; CANCER CELL; CYTOTOXICITY; DRUG CONJUGATION; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; FEMALE; HUMAN; HUMAN CELL; MALE; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY;

ADULT; AGED; AGED, 80 AND OVER; ANIMALS; ANTINEOPLASTIC AGENTS; CELL LINE; DAUNORUBICIN; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG SCREENING ASSAYS, ANTITUMOR; ESTROGENS; FEMALE; HUMANS; LIGANDS; MALE; MICE; MIDDLE AGED; MOLECULAR STRUCTURE; RECEPTORS, ESTROGEN;

EID: 0034884460 PISSN: 0039128X EISSN: None Source Type: Journal
DOI: 10.1016/S0039-128X(01)00110-6 Document Type: Article

Times cited : (37)

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