Photoactivatable α-conotoxins reveal contacts with all subunits as well as antagonist-induced rearrangements in the Torpedo californica acetylcholine receptor

European Journal of Biochemistry

Volumn 268, Issue 13, 2001, Pages 3664-3673

  Kasheverov, Igor ^a   Rozhkova, Anna ^a   Zhmak, Maxim ^a   Utkin, Yuri ^a   Ivanov, Vadim ^a   Tsetlin, Victor I ^a  

^a SHEMYAKIN OVCHINNIKOV INSTITUTE OF BIOORGANIC CHEMISTRY   (Russian Federation)

Author keywords

conotoxins; Acetylcholine receptor; Antagonist induced rearrangements; Photoactivatable derivatives; Physostigmine

Indexed keywords

ALPHA BUNGAROTOXIN; ALPHA CONOTOXIN GI; ALPHA CONOTOXIN MI; CHOLINERGIC RECEPTOR; CONOTOXIN; IODINE 125; PHYSOSTIGMINE; RECEPTOR SUBUNIT; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING SITE; CONFORMATIONAL TRANSITION; CONTROLLED STUDY; CROSS LINKING; DRUG POTENCY; DRUG SYNTHESIS; IRRADIATION; ISOTOPE LABELING; NONHUMAN; PHOTOACTIVATION; PRIORITY JOURNAL; RECEPTOR BINDING; TORPEDO CALIFORNICA;

AMINO ACID SEQUENCE; ANIMALS; BINDING SITES; BUNGAROTOXINS; CONOTOXINS; IODINE RADIOISOTOPES; KINETICS; MOLECULAR SEQUENCE DATA; PHOTOCHEMISTRY; PROTEIN SUBUNITS; RECEPTORS, NICOTINIC; SEQUENCE ALIGNMENT; SEQUENCE HOMOLOGY, AMINO ACID; SPECTROMETRY, MASS, MATRIX-ASSISTED LASER DESORPTION-IONIZATION; SUBSTRATE SPECIFICITY; TORPEDO;

EID: 0034819433     PISSN: 00142956     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1432-1327.2001.02272.x     Document Type: Article

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