Modulation of GABAA receptor-mediated currents by phenazepam and its metabolites

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 364, Issue 1, 2001, Pages 1-8

  Kopanitsa, M V ^a   Zhuk, O V ^a   Zinkovsky, V G ^a   Krishtal, O A ^a  

^a BOGOMOLETZ INSTITUTE OF PHYSIOLOGY   (Ukraine)

Author keywords

1,4 Benzodiazepine metabolites; Benzophenone; GABAA receptor; Patch clamp; Phenazepam; Purkinje neurone; Quinazoline; Whole cell

Indexed keywords

3 HYDROXYPHENAZEPAM; 4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; 5 BROMO (2 CHLOROPHENYL) 2 AMINOBENZOPHENONE; 6 BROMO (2 CHLOROPHENYL)QUINAZOLIN 2 ONE; BENZODIAZEPIN 2 ONE DERIVATIVE; CHLORIDE ION; DIAZEPAM; DRUG METABOLITE; PHENAZEPAM; UNCLASSIFIED DRUG; 3-HYDROXYPHENAZEPAM; ANXIOLYTIC AGENT; BENZODIAZEPINE DERIVATIVE; BENZODIAZEPINE RECEPTOR AFFECTING AGENT;

ANIMAL CELL; ARTICLE; CHLORIDE CURRENT; CONTROLLED STUDY; DRUG EFFECT; DRUG MECHANISM; DRUG RECEPTOR BINDING; GABAERGIC SYSTEM; ION CURRENT; NONHUMAN; PATCH CLAMP; PURKINJE CELL; RAT; RECEPTOR DOWN REGULATION; ANIMAL; CELL MEMBRANE POTENTIAL; CHEMICAL STRUCTURE; CHEMISTRY; METABOLISM; NERVE CELL;

ANIMALS; ANTI-ANXIETY AGENTS; BENZODIAZEPINES; DIAZEPAM; GABA MODULATORS; MEMBRANE POTENTIALS; MOLECULAR STRUCTURE; NEURONS; PURKINJE CELLS; RATS; RECEPTORS, GABA-A;

EID: 0034743335     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/s002100100403     Document Type: Article

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