4-Aminoquinolines: Novel nociceptin antagonists with analgesic activity

Journal of Medicinal Chemistry

Volumn 43, Issue 24, 2000, Pages 4667-4677

  Shinkai, H ^a   Ito, T ^a   Iida, T ^a   Kitao, Y ^a   Yamada, H ^a   Uchida, I ^a  

^a JT Inc   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOQUINOLINE DERIVATIVE; ANALGESIC AGENT; NALOXONE; NOCICEPTIN RECEPTOR ANTAGONIST; UNCLASSIFIED DRUG;

ALLODYNIA; ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CONTROLLED STUDY; DRUG MECHANISM; DRUG STRUCTURE; DRUG SYNTHESIS; HOT PLATE TEST; MALE; MOUSE; NONHUMAN; RAT;

ADENOSINE MONOPHOSPHATE; AMINOQUINOLINES; ANALGESICS; ANIMALS; BENZAMIDES; CELL LINE; DRUG EVALUATION, PRECLINICAL; HUMANS; MALE; MICE; MICE, INBRED ICR; NALOXONE; NARCOTIC ANTAGONISTS; OPIOID PEPTIDES; PAIN MEASUREMENT; RADIOLIGAND ASSAY; RECEPTORS, OPIOID, DELTA; RECEPTORS, OPIOID, KAPPA; RECEPTORS, OPIOID, MU; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0034736150     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm0002073     Document Type: Article

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