메뉴 건너뛰기




Volumn 99, Issue 1-2, 2000, Pages 91-100

Pharmacology of recombinant human GABA(A) receptor subtypes measured using a novel pH-based high-throughput functional efficacy assay

Author keywords

Benzodiazepines; Fluorescence; GABA; L(tk ) cells; pH regulation

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; BENZODIAZEPINE DERIVATIVE; BICUCULLINE; CARBOXYFLUORESCEIN; DIAZEPAM; HYDROGEN POTASSIUM ADENOSINE TRIPHOSPHATASE; LIGAND; RECEPTOR SUBTYPE;

EID: 0034733467     PISSN: 01650270     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0165-0270(00)00219-3     Document Type: Article
Times cited : (11)

References (29)
  • 2
    • 0030762991 scopus 로고    scopus 로고
    • Ion pumps in epithelial cells: Sorting, stabilization, and polarity
    • Caplan M.J. Ion pumps in epithelial cells: sorting, stabilization, and polarity. Am. J. Physiol. 272:1997;G1304-G1313.
    • (1997) Am. J. Physiol. , vol.272 , pp. 1304-G1313
    • Caplan, M.J.1
  • 3
    • 33750879837 scopus 로고    scopus 로고
    • Sodium-independent inward chloride pumping in rat cardiac ventricular cells
    • Chipperfield A.R., Davis J.P.L., Harper A.A. Sodium-independent inward chloride pumping in rat cardiac ventricular cells. Am. J. Physiol. 272:1997;735-739.
    • (1997) Am. J. Physiol , vol.272 , pp. 735-739
    • Chipperfield, A.R.1    Davis, J.P.L.2    Harper, A.A.3
  • 7
    • 0021895468 scopus 로고
    • Transport of sodium and chloride across rat gastric mucosa in vitro
    • Jackson M.J., Norris S.H. Transport of sodium and chloride across rat gastric mucosa in vitro. J. Physiol. (Lond.). 360:1985;293-310.
    • (1985) J. Physiol. (Lond.) , vol.360 , pp. 293-310
    • Jackson, M.J.1    Norris, S.H.2
  • 8
    • 0020684357 scopus 로고
    • Direct effect of metolazone on sodium-dependent transport across the renal brush border membrane
    • Kempson S.A., Kowalski J.C., Puschett J.B. Direct effect of metolazone on sodium-dependent transport across the renal brush border membrane. J. Lab. Clin. Med. 101:1983;308-316.
    • (1983) J. Lab. Clin. Med. , vol.101 , pp. 308-316
    • Kempson, S.A.1    Kowalski, J.C.2    Puschett, J.B.3
  • 12
    • 0031856385 scopus 로고    scopus 로고
    • Rapid assessment of ligand actions with nicotinic acetylcholine receptors using calcium dynamics and FLIPR
    • Kuntzweiler T.A., Arneric S.P., Donnelly-Roberts D.L. Rapid assessment of ligand actions with nicotinic acetylcholine receptors using calcium dynamics and FLIPR. Drug. Dev. Res. 44:1998;14-20.
    • (1998) Drug. Dev. Res. , vol.44 , pp. 14-20
    • Kuntzweiler, T.A.1    Arneric, S.P.2    Donnelly-Roberts, D.L.3
  • 13
    • 0026724785 scopus 로고
    • +-ATPase in vascular smooth muscle cells
    • +-ATPase in vascular smooth muscle cells. Am. J. Physiol. 262:1992;H1955-H1958.
    • (1992) Am. J. Physiol. , vol.262 , pp. 1955-H1958
    • McCabe, R.D.1    Young, D.B.2
  • 16
    • 0025644867 scopus 로고
    • Intracellular ion activities and membrane transport in parietal cells measured with fluorescent dyes
    • Negulescu P.A., Machen T.E. Intracellular ion activities and membrane transport in parietal cells measured with fluorescent dyes. Methods. Enzymol. 192:1990;38-81.
    • (1990) Methods. Enzymol. , vol.192 , pp. 38-81
    • Negulescu, P.A.1    Machen, T.E.2
  • 17
    • 0024246930 scopus 로고
    • +-ATPase, gastric acid secretion and HCl·ethanol-induced gastric lesions in rats
    • +-ATPase, gastric acid secretion and HCl·ethanol-induced gastric lesions in rats. Dig. Dis. Sci. 33:1987;1425-1434.
    • (1987) Dig. Dis. Sci. , vol.33 , pp. 1425-1434
    • Okabe, S.1    Akimoto, Y.2    Yamasaki, S.3    Nagai, H.4
  • 18
    • 0024423323 scopus 로고
    • A-benzodiazepine receptors produced in transfected cells
    • A-benzodiazepine receptors produced in transfected cells. Science. 245:1989a;1389-1392.
    • (1989) Science , vol.245 , pp. 1389-1392
    • Pritchett, D.B.1    Luddens, H.2    Seeburg, P.H.3
  • 20
    • 0028174520 scopus 로고
    • γ-Aminobutyric acid type A receptors in the rat brain can contain both γ2 and γ3 subunits, but γ1 does not exist in combination with another subunit
    • Quirk K., Gillard N.P., Ragan C.I., Whiting P.J., McKernan R.M. γ-Aminobutyric acid type A receptors in the rat brain can contain both γ2 and γ3 subunits, but γ1 does not exist in combination with another subunit. Mol. Pharmacol. 45:1994;1061.
    • (1994) Mol. Pharmacol. , vol.45 , pp. 1061
    • Quirk, K.1    Gillard, N.P.2    Ragan, C.I.3    Whiting, P.J.4    McKernan, R.M.5
  • 21
    • 0030598573 scopus 로고    scopus 로고
    • A receptors containing α4β3γ2, α4β2, or α1β3γ2 subunits
    • A receptors containing α4β3γ2, α4β2, or α1β3γ2 subunits. Eur. J. Pharmacol. 304:1996;155-162.
    • (1996) Eur. J. Pharmacol. , vol.304 , pp. 155-162
    • Scholze, P.1    Ebert, V.2    Sieghart, W.3
  • 23
    • 0034708421 scopus 로고    scopus 로고
    • Functional characterization of bradykinin analogues on Chinese hamster ovary cells expressing recombinant human B1 and B2 bradykinin receptors
    • Simpson P.B., Woollacott A.J., Hill R.G., Seabrook G.R. Functional characterization of bradykinin analogues on Chinese hamster ovary cells expressing recombinant human B1 and B2 bradykinin receptors. Eur. J. Pharmacol. 392:2000;1-9.
    • (2000) Eur. J. Pharmacol. , vol.392 , pp. 1-9
    • Simpson, P.B.1    Woollacott, A.J.2    Hill, R.G.3    Seabrook, G.R.4
  • 25
    • 0025687508 scopus 로고
    • A receptor, but the α1 polypeptide is the principal site of the agonist benzodiazepine photoaffinity labelling reaction
    • A receptor, but the α1 polypeptide is the principal site of the agonist benzodiazepine photoaffinity labelling reaction. J. Biol. Chem. 265:1990;21160.
    • (1990) J. Biol. Chem. , vol.265 , pp. 21160
    • Stephenson, F.A.1    Duggan, M.J.2    Pollard, S.3
  • 26
    • 0029417325 scopus 로고
    • A receptor inverse agonists modulate γ-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site
    • A receptor inverse agonists modulate γ-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site. Mol. Pharmacol. 481:1995;965-969.
    • (1995) Mol. Pharmacol. , vol.481 , pp. 965-969
    • Stevenson, A.1    Wingrove, P.B.2    Whiting, P.J.3    Wafford, K.A.4
  • 29
    • 0026612363 scopus 로고
    • A receptor subunit mRNAs in the rat brain. I. Telencephelon, diencephelon, mesencephalon
    • A receptor subunit mRNAs in the rat brain. I. Telencephelon, diencephelon, mesencephalon. J. Neurosci. 12:1992;1040-1062.
    • (1992) J. Neurosci. , vol.12 , pp. 1040-1062
    • Wisden, W.1    Laurie, D.J.2    Monyer, H.3    Seeburg, P.H.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.