Affinity of various ligands for GABA(A) receptors containing α4β3γ2, α4γ2, or α1β3γ2 subunits

European Journal of Pharmacology

Volumn 304, Issue 1-3, 1996, Pages 155-162

  Scholze, Petra ^a   Ebert, Veronika ^a   Sieghart, Werner ^a  

^a MEDICAL UNIVERSITY OF VIENNA   (Austria)

Author keywords

benzodiazepine binding site property; GABA(A) receptor subtype, recombinant, 4 3 2S, 4 2S, 1 3 2S

Indexed keywords

2 PHENYL 4 [2 (3 PIPERIDYL)ETHYL]QUINOLINE; 2 PHENYL 5H PYRAZOLO[4,3 C]QUINOLIN 3 ONE; 3 METHYL 6 (3 TRIFLUOROMETHYLPHENYL) 1,2,4 TRIAZOLO[4,3 B]PYRIDAZINE; 4 AMINOBUTYRIC ACID A RECEPTOR; 8 AZIDO 5,6 DIHYDRO 5 METHYL 6 OXO 4H IMIDAZO[1,5 A][1,4]BENZODIAZEPINE 3 CARBOXYLIC ACID ETHYL ESTER; ABECARNIL; ALPRAZOLAM; BENZODIAZEPINE DERIVATIVE; BENZODIAZEPINE RECEPTOR; BETA CARBOLINE DERIVATIVE; CLOBAZAM; CLOTIAZEPAM; CLOXAZOLAM; CYCLOPYRROLONE DERIVATIVE; FLUMAZENIL; GABAERGIC RECEPTOR AFFECTING AGENT; IMIDAZOPYRIDINE DERIVATIVE; IMIDAZOQUINOLINE DERIVATIVE; ISOQUINOLINE DERIVATIVE; N METHYL BETA CARBOLINE 3 CARBOXAMIDE; N SEC BUTYL 1 (2 CHLOROPHENYL) N METHYL 3 ISOQUINOLINECARBOXAMIDE; QUINOLINE DERIVATIVE; RADIOLIGAND; RECEPTOR SUBTYPE; RECEPTOR SUBUNIT; TRIAZOLOPYRIDAZINE DERIVATIVE; UNCLASSIFIED DRUG; UNINDEXED DRUG; ZOLPIDEM; ZOPICLONE; AZIDE; LIGAND; RECOMBINANT PROTEIN;

ARTICLE; BINDING COMPETITION; CONTROLLED STUDY; DRUG POTENCY; EMBRYO; HUMAN; HUMAN CELL; KIDNEY CELL; MOLECULAR CLONING; PRIORITY JOURNAL; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION; ANIMAL; BINDING SITE; CELL CULTURE; CYTOLOGY; DRUG ANTAGONISM; DRUG EFFECT; GENETICS; IN VITRO STUDY; KIDNEY; METABOLISM; PROTEIN BINDING; RADIOASSAY; RAT;

ANIMALS; AZIDES; BENZODIAZEPINES; BINDING SITES; CELLS, CULTURED; CLONING, MOLECULAR; EMBRYO; HUMANS; KIDNEY; LIGANDS; PROTEIN BINDING; RADIOLIGAND ASSAY; RATS; RECEPTORS, GABA-A; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0030598573     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(96)00088-X     Document Type: Article

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