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85037517381
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(h) Takamura, M.; Hamashima, Y.; Usuda, H.; Kanai, M.; Shibasaki, M. Submitted for publication.
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85037497547
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note
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All ketoimines were prepared by reaction of the appropriate ketone and amine in dichloromethane in the presence of 3 Å sieves. Full experimental details are provided as Supporting Information.
-
-
-
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29
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-
85037521439
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-
note
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Solutions of hydrogen cyanide were generated prior to the Strecker reaction by combination of equimolar amounts of TMSCN and methanol in toluene at 5°C for 2 h.
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30
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33748737484
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85007975161
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The absolute stereochemistry of 6 was assigned by comparison of its optical rotation with literature values: (a) Terashima, S.; Yamada, S. I. Chem. Pharm. Bull. 1968, 15, 1953.
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Spiegler, C.8
Mueller, K.9
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