1-Aminomethylisoquinoline-4-carboxylates as novel dipeptidylpeptidase IV inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 14, 2000, Pages 1555-1558

  Coppola, Gary M ^a   Zhang, Y Larry ^a   Schuster, Herbert F ^a   Russell, Mary E ^a   Hughes, Thomas E ^a  

^a NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1 AMINOMETHYLISOQUINOLINE 4 CARBOXYLIC ACID; CARBOXYLIC ACID DERIVATIVE; DIPEPTIDYL PEPTIDASE IV; ENZYME INHIBITOR; ISOQUINOLINE DERIVATIVE; SDZ 029 576; UNCLASSIFIED DRUG;

ARTICLE; DRUG INHIBITION; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; STRUCTURE ACTIVITY RELATION;

ANTIGENS, CD26; CARBOXYLIC ACIDS; COLONIC NEOPLASMS; HUMANS; INDICATORS AND REAGENTS; ISOQUINOLINES; KINETICS; MOLECULAR STRUCTURE; PROTEASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP; TUMOR CELLS, CULTURED;

EID: 0034679748     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(00)00286-9     Document Type: Article

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