NVP-DPP728 (1-[[[2-[(5-cyanopyridin-2-yl)amino]ethyl] amino] acetyl]-2- cyano-(S)-pyrrolidine), a slow-binding inhibitor of dipeptidyl peptidase IV

Biochemistry

Volumn 38, Issue 36, 1999, Pages 11597-11603

  Hughes, Thomas E ^a   Mone, Manisha D ^a   Russell, Mary E ^a   Weldon, Stephen C ^a   Villhauer, Edwin B ^a  

^a NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1 [[[2 [(5 CYANOPYRIDIN 2 YL)AMINO]ETHYL]AMINO]ACETYL] 2 CYANO PYRROLIDINE; DIPEPTIDYL PEPTIDASE IV; GLUCAGON LIKE PEPTIDE 1; INSULIN; NITRILE; PYRROLIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CATTLE; DEGRADATION; DISSOCIATION CONSTANT; ENZYME INHIBITION; HUMAN; HUMAN CELL; NONHUMAN; POLYACRYLAMIDE GEL ELECTROPHORESIS; PRIORITY JOURNAL;

ANIMALS; ANTIGENS, CD26; CACO-2 CELLS; CATTLE; DRUG STABILITY; HUMANS; NITRILES; PROTEASE INHIBITORS; PYRROLIDINES;

ANIMALIA; BOS TAURUS; BOVINAE;

EID: 0033533402     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi990852f     Document Type: Article

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