-
1
-
-
0020375151
-
-
For a review see: (a)
-
For a review see: (a) Nagai, Y.; Irie, A.; Nakamura, H.; Hino, K.; Uno, H.; Nishimura, H. J. Med. Chem. 1982, 25, 1065-1070.
-
(1982)
J. Med. Chem.
, vol.25
, pp. 1065-1070
-
-
Nagai, Y.1
Irie, A.2
Nakamura, H.3
Hino, K.4
Uno, H.5
Nishimura, H.6
-
5
-
-
0025718829
-
-
(b)
-
(b) Room, P.; Tielemans, A.J. P. C.; de Boer, T.; Van Delft, A.M.L.; Jeroen, J.A.D.M. Eur. J. Pharmacol. 1991, 205, 233-240.
-
(1991)
Eur. J. Pharmacol.
, vol.205
, pp. 233-240
-
-
Room, P.1
Tielemans, A.J.P.C.2
De Boer, T.3
Van Delft, A.M.L.4
Jeroen, J.A.D.M.5
-
6
-
-
0030610198
-
-
(a)
-
(a) Andree, B.; Halldin, C.; Vrijmoed, M.; Farde, L. Psycopharmacol. 1997, 113, 339-345.
-
(1997)
Psycopharmacol.
, vol.113
, pp. 339-345
-
-
Andree, B.1
Halldin, C.2
Vrijmoed, M.3
Farde, L.4
-
7
-
-
0028917659
-
-
(b)
-
(b) Maduskuie, T. P.; Wilde, R. G.; Billheimer, J.; Cromley, D. A.; Germain, S.; Gillies, P. J.; Higley, C. A.; Johnson, A. L.; Penner, P. J. Med. Chem. 1995, 38, 1067-1083.
-
(1995)
J. Med. Chem.
, vol.38
, pp. 1067-1083
-
-
Maduskuie, T.P.1
Wilde, R.G.2
Billheimer, J.3
Cromley, D.A.4
Germain, S.5
Gillies, P.J.6
Higley, C.A.7
Johnson, A.L.8
Penner, P.9
-
8
-
-
0011830151
-
-
(a)
-
(a) Domínguez, E.; Mtez. de Marigorta, E.; Olivera, R.; SanMartin, R. Synlett 1995, 955-956.
-
(1995)
Synlett
, pp. 955-956
-
-
Domínguez, E.1
Mtez. De Marigorta, E.2
Olivera, R.3
Sanmartin, R.4
-
9
-
-
0000228798
-
-
(b)
-
(b) Domínguez, E.; Ibeas, E.; Mtez. de Marigorta, E.; Palacios, J. K.; SanMartin, R. J. Org. Chem. 1996, 61, 5435-5439.
-
(1996)
J. Org. Chem.
, vol.61
, pp. 5435-5439
-
-
Domínguez, E.1
Ibeas, E.2
Mtez. De Marigorta, E.3
Palacios, J.K.4
Sanmartin, R.5
-
10
-
-
0032563819
-
-
(a)
-
(a) Olivera, R.; Pascual, S.; Herrero, M.; SanMartin, R.; Domínguez, E. Tetrahedron Lett. 1998, 39, 7155-7158.
-
(1998)
Tetrahedron Lett.
, vol.39
, pp. 7155-7158
-
-
Olivera, R.1
Pascual, S.2
Herrero, M.3
Sanmartin, R.4
Domínguez, E.5
-
11
-
-
0033597153
-
-
(b)
-
(b) Olivera, R.; SanMartin, R.; Pascual, S.; Herrero, M.; Domínguez, E. Tetrahedron Lett. 1999, 40, 3479-3480.
-
(1999)
Tetrahedron Lett.
, vol.40
, pp. 3479-3480
-
-
Olivera, R.1
Sanmartin, R.2
Pascual, S.3
Herrero, M.4
Domínguez, E.5
-
13
-
-
0033597748
-
-
(b)
-
(b) Hartwig, J. F.; Kawatsura, M.; Hauck, S. I.; Shaghnessy, K. H.; Alcázar-Román, L. M. J. Org. Chem. 1999, 64, 5575-5580.
-
(1999)
J. Org. Chem.
, vol.64
, pp. 5575-5580
-
-
Hartwig, J.F.1
Kawatsura, M.2
Hauck, S.I.3
Shaghnessy, K.H.4
Alcázar-Román, L.M.5
-
14
-
-
0029886443
-
-
(a)
-
(a) de la Fuente, M.C.; Castedo, L.; Domínguez, D. Tetrahedron 1996, 52, 4917-4924.
-
(1996)
Tetrahedron
, vol.52
, pp. 4917-4924
-
-
De La Fuente, M.C.1
Castedo, L.2
Domínguez, D.3
-
15
-
-
0032565912
-
-
(b)
-
(b) Rossi, R; Bellina, F.; Ciucci, D.; Carpita, A.; Fanelli, C. Tetrahedron 1998, 54, 7595-7614.
-
(1998)
Tetrahedron
, vol.54
, pp. 7595-7614
-
-
Rossi, R.1
Bellina, F.2
Ciucci, D.3
Carpita, A.4
Fanelli, C.5
-
17
-
-
0032483549
-
-
(b)
-
(b) Sawyer, J. S.; Schmittling, E. A.; Palkowitz, J. A.; Smith, W. J. J. Org. Chem. 1998, 63, 6338-6343.
-
(1998)
J. Org. Chem.
, vol.63
, pp. 6338-6343
-
-
Sawyer, J.S.1
Schmittling, E.A.2
Palkowitz, J.A.3
Smith, W.J.4
-
18
-
-
0033534565
-
-
(c)
-
(c) Boger, D. L.; Castle, S. L.; Miyazaki, S.; Wu, J. H.; Beresis, R. T.; Loiseleur, O. J. Org. Chem, 1999, 64, 70-80.
-
(1999)
J. Org. Chem
, vol.64
, pp. 70-80
-
-
Boger, D.L.1
Castle, S.L.2
Miyazaki, S.3
Wu, J.H.4
Beresis, R.T.5
Loiseleur, O.6
-
22
-
-
0030760929
-
-
(a)
-
(a) Widenhoefer, R. A.; Zhong, H. A.; Buchwald, S. L. J. Am. Chem. Soc. 1997, 119, 6787-6795.
-
(1997)
J. Am. Chem. Soc.
, vol.119
, pp. 6787-6795
-
-
Widenhoefer, R.A.1
Zhong, H.A.2
Buchwald, S.L.3
-
25
-
-
0033531744
-
-
(b)
-
(b) Mann, G.; Incarvito, C.; Rheingold, A. L.; Hartwig, J. F. J. Am. Chem. Soc. 1999, 121, 3223-3225.
-
(1999)
J. Am. Chem. Soc.
, vol.121
, pp. 3223-3225
-
-
Mann, G.1
Incarvito, C.2
Rheingold, A.L.3
Hartwig, J.F.4
-
26
-
-
0033549049
-
-
(c)
-
(c) Araynos, A.; Old, D. W.; Kiyomori, A.; Wolfe, J. P.; Sadighi, J. P.; Buchwald, S. L. J. Am. Chem. Soc. 1999, 121, 4369-4378.
-
(1999)
J. Am. Chem. Soc.
, vol.121
, pp. 4369-4378
-
-
Araynos, A.1
Old, D.W.2
Kiyomori, A.3
Wolfe, J.P.4
Sadighi, J.P.5
Buchwald, S.L.6
-
27
-
-
0032510084
-
-
Pinchart, A.; Dallaire, C.; Gingras, M. Tetrahedron Lett. 1998, 39, 543-546.
-
(1998)
Tetrahedron Lett.
, vol.39
, pp. 543-546
-
-
Pinchart, A.1
Dallaire, C.2
Gingras, M.3
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28
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85037967947
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PhD Thesis, University of the Basque Country
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Olivera, R. PhD Thesis, University of the Basque Country, 2000.
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(2000)
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Olivera, R.1
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29
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85037966445
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BINAP: 2,2′-Bis(diphenylphosphino)-1,1′-binaphthyl.
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BINAP: 2,2′-Bis(diphenylphosphino)-1,1′-binaphthyl.
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30
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85037966099
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DPPF: 1,1'-bis(diphenylphosphino)ferrocene
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DPPF: 1,1'-bis(diphenylphosphino)ferrocene.
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32
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85037968897
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Note
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2 as eluent, providing dibenzoxepine 3a (0.109 g, 69%) as a white powder.
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33
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85037956311
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2O: C, 81.27; H, 4.55; N, 9.03. Found: C, 81.39; H, 4.64; N, 9.17.
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2O: C, 81.27; H, 4.55; N, 9.03. Found: C, 81.39; H, 4.64; N, 9.17.
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35
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85037969723
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The observed GC/MS yields for dibenzoxepinopyrazole 3b were 64 and 51% when DPPF and BINAP were the chelating ligands, respectively. The difference between the observed and isolated yields is adduced to the resinous nature of the product and the substrate, which made the purification of the target compound considerably difficult.
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The observed GC/MS yields for dibenzoxepinopyrazole 3b were 64 and 51% when DPPF and BINAP were the chelating ligands, respectively. The difference between the observed and isolated yields is adduced to the resinous nature of the product and the substrate, which made the purification of the target compound considerably difficult.
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36
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85037961494
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Similar intermediates have been proposed in the arylation of alkoxides and phenoxides. See Ref. 11b-c
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Similar intermediates have been proposed in the arylation of alkoxides and phenoxides. See Ref. 11b-c.
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