Preparation and characterization of cholic acid-derived antimicrobial agents with controlled stabilities

Organic Letters

Volumn 2, Issue 18, 2000, Pages 2837-2840

  Guan, Qunying ^a   Li, Chunhong ^a   Schmidt, Erica J ^b   Boswell, J Scott ^b   Walsh, Joshua P ^b   Allman, Glenn W ^b   Savage, Paul B ^a  

^a Brigham Young University   (United States)

^b BRIGHAM YOUNG UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIINFECTIVE AGENT; CHOLIC ACID DERIVATIVE;

ARTICLE; CELL MEMBRANE PERMEABILITY; DRUG EFFECT; DRUG STABILITY; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; METABOLISM; MICROBIOLOGICAL EXAMINATION; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ANTI-BACTERIAL AGENTS; CELL MEMBRANE PERMEABILITY; CHOLIC ACIDS; DRUG STABILITY; GRAM-NEGATIVE BACTERIA; GRAM-POSITIVE BACTERIA; MICROBIAL SENSITIVITY TESTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0034618315     PISSN: 15237060     EISSN: None     Source Type: Journal    
DOI: 10.1021/ol0062704     Document Type: Article

References (14)

1. For a recent review, see: Epand, R. M.; Vogel, H. J. Biochim. Biophys. Acta 1999, 1462, 11.
2. Shai, Y. Biochim. Biophys. Acta 1999, 1462, 55.
3. Groisman, E. A.; Kayser, J.; Soncini, F. C. J. Bacteriol. 1997, 179, 7040.
4. (a) Li, C.; Budge, L. P.; Driscoll, C. D.; Willardson, B. M.; Allman, G. W.; Savage, P. B. J. Am. Chem. Soc. 1999, 121, 931.
5. (b) Rehman, A.; Li, C.; Budge, L. P.; Street, S. E.; Savage, P. B. Tetrahedron Lett. 1999, 40, 1865.
6. (c) Li, C.; Peters, A. S.; Meredith, E. L.; Allman, G. H.; Savage, P. B. J. Am. Chem. Soc. 1998, 120, 2961.
7. Li, C.; Lewis, M. R.; Gilbert, A. B.; Noel, M. D.; Scoville, D. H.; Allman, G. W.; Savage, P. B. Antimicrob. Agents Chemother. 1999, 43, 1347.
8. 13 cells). Tannock, G. W. In Normal Microfluora. An Introduction to Microbes Inhabiting the Human Body; Tannock, G. W., Ed.; Chapman and Hall: London, 1994; pp 1-36.
9. For example see: (a) Vollaard, E. J.; Clasener, H. A. L. Antimicrob. Agents Chemother. 1994, 38, 409.
10. (b) Hentges, D. J. In Human Intestinal Microflora in Health and Disease; Hentges, D. J., Ed.; Academic Press: New York, 1983; pp 311-328.
11. For example, see: Finegold, S. M.; Mathisen, G. E.; George, W. L. In Human Intestinal Microflora in Health and Disease; Hentges, D. J., Ed.; Academic Press: New York. 1983; pp 356-438.
12. Delves-Broughton, J.; Blackburn, P.; Evans, R. J.; Hugenholtz, J. Antonie van Leeuwenhoek 1996, 69, 193.
13. De Vuyst, L.; Vandamme, E. J. In Bacteriocins of Lactic Acid Bacteria; De Vuyst, L.; Vandamme, E. J., Ed.; Blackie Academic and Professional: Glasgow, 1994; pp 151-221.
14. Matsuzaki, K.; Sugishita, K.; Fugii, N.; Miyajima, K. Biochemistry 1995, 34, 3423.