Stereoselective pharmacokinetics of desbutylhalofantrine, a metabolite of halofantrine, in the rat after administration of the racemic metabolite or parent drug

Biopharmaceutics and Drug Disposition

Volumn 21, Issue 9, 2000, Pages 365-371

  Brocks, Dion R ^a  

^a WESTERN UNIVERSITY OF HEALTH SCIENCES   (United States)

Author keywords

Halofantrine; Plasma; Stereoselectivity

Indexed keywords

DEBUTYLHALOFANTRINE; DRUG METABOLITE; HALOFANTRINE; HALOTHANE; PHENANTHRENE DERIVATIVE; QUINIDINE;

ANIMAL EXPERIMENT; ANIMAL MODEL; AREA UNDER THE CURVE; ARTICLE; CONTROLLED STUDY; DISTRIBUTION VOLUME; DRUG BIOAVAILABILITY; DRUG BLOOD LEVEL; DRUG CLEARANCE; DRUG DETERMINATION; DRUG METABOLISM; ENANTIOMER; MALE; NONHUMAN; RACEMIC MIXTURE; RAT; STEREOCHEMISTRY;

ANIMALS; ANTIMALARIALS; MALE; PHENANTHRENES; RATS; RATS, SPRAGUE-DAWLEY; STEREOISOMERISM;

EID: 0034429628     PISSN: 01422782     EISSN: None     Source Type: Journal    
DOI: 10.1002/bdd.251     Document Type: Article

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