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Volumn 56, Issue 2, 2000, Pages 145-151

Modulation of midazolam 1-hydroxylation activity in vitro by neurotransmitters and precursors

Author keywords

CYP3A; Indoleamines; Metabolism

Indexed keywords

ADRENALIN; CYTOCHROME P450 3A; CYTOCHROME P450 ISOENZYME; MIDAZOLAM; NEUROTRANSMITTER; SEROTONIN;

EID: 0034129703     PISSN: 00316970     EISSN: None     Source Type: Journal    
DOI: 10.1007/s002280050733     Document Type: Article
Times cited : (19)

References (45)
  • 1
    • 0031776805 scopus 로고    scopus 로고
    • Modulation of CYP1A2 enzyme activity by indoleamines. Inhibition by serotonin and tryptamine
    • Agúndez JAG, Gallardo L, Martínez C, Gervasini G, Bonítez J (1998) Modulation of CYP1A2 enzyme activity by indoleamines. Inhibition by serotonin and tryptamine. Pharmacogenetics 8: 251-258
    • (1998) Pharmacogenetics , vol.8 , pp. 251-258
    • Agúndez, J.A.G.1    Gallardo, L.2    Martínez, C.3    Gervasini, G.4    Bonítez, J.5
  • 2
    • 0024309378 scopus 로고
    • Comparative effects of two antimycotic agents, ketoconazole and terfenadine on the metabolism of tolbutamide, ethinyloestradiol, clyclosporin and ethoxycoumarin by human liver microsomes in vitro
    • Back DJ, Stevenson P, Tjia JF (1989) Comparative effects of two antimycotic agents, ketoconazole and terfenadine on the metabolism of tolbutamide, ethinyloestradiol, clyclosporin and ethoxycoumarin by human liver microsomes in vitro. Br J Clin Pharmacol 28: 166-170
    • (1989) Br J Clin Pharmacol , vol.28 , pp. 166-170
    • Back, D.J.1    Stevenson, P.2    Tjia, J.F.3
  • 4
    • 0021273321 scopus 로고
    • 5-Hydroxytryptophol in human cerebrospinal fluid: Conjugation, concentration gradient, relationship to 5-hydroxyindoleacetic acid, and influence of hereditary factors
    • Beck O, Borg S, Edman G, Fyro B, Oxenstierna G, Sedvall G (1984a) 5-hydroxytryptophol in human cerebrospinal fluid: conjugation, concentration gradient, relationship to 5-hydroxyindoleacetic acid, and influence of hereditary factors. J Neurochem 43: 58-61
    • (1984) J Neurochem , vol.43 , pp. 58-61
    • Beck, O.1    Borg, S.2    Edman, G.3    Fyro, B.4    Oxenstierna, G.5    Sedvall, G.6
  • 5
    • 0021361430 scopus 로고
    • Measurement of 5-hydroxytryptophol and 5-hydroxyindoleacetic acid in human and rat brain and plasma
    • Beck O, Borg S, Jonsson G, Lundman A, Valverius P (1984b) Measurement of 5-hydroxytryptophol and 5-hydroxyindoleacetic acid in human and rat brain and plasma. J Neural Transm 59: 57-67
    • (1984) J Neural Transm , vol.59 , pp. 57-67
    • Beck, O.1    Borg, S.2    Jonsson, G.3    Lundman, A.4    Valverius, P.5
  • 6
    • 0027244082 scopus 로고
    • Purification of multiple forms of cytochrome P450 from a human brain and reconstitution of catalytic activities
    • Bhamre S, Anandatheeraavarada HK, Shankar SK, Boyd MR, Ravindranath V (1993) Purification of multiple forms of cytochrome P450 from a human brain and reconstitution of catalytic activities. Arch Biochem Biophys 310: 251-255
    • (1993) Arch Biochem Biophys , vol.310 , pp. 251-255
    • Bhamre, S.1    Anandatheeraavarada, H.K.2    Shankar, S.K.3    Boyd, M.R.4    Ravindranath, V.5
  • 7
    • 0031811037 scopus 로고    scopus 로고
    • Analysis of midazolam and metabolites in plasma by high performance liquid chromatography. A probe of CYP3A
    • Carrillo JA, Ramos SI, Agúndez JAG, Martínez C, Benítez J (1998) Analysis of midazolam and metabolites in plasma by high performance liquid chromatography. A probe of CYP3A. Ther Drug Monit 20: 319-324
    • (1998) Ther Drug Monit , vol.20 , pp. 319-324
    • Carrillo, J.A.1    Ramos, S.I.2    Agúndez, J.A.G.3    Martínez, C.4    Benítez, J.5
  • 8
    • 0024603850 scopus 로고
    • Metabolism of cyclosporin A; IV: Purification and identification of the rifampin-inducible human liver cytochrome P-450 (cyclosporin A oxidase) as a product of P450IIIA gene subfamily
    • Combalbert J, Fabre I, Fabre G, et al. (1989) Metabolism of cyclosporin A; IV: purification and identification of the rifampin-inducible human liver cytochrome P-450 (cyclosporin A oxidase) as a product of P450IIIA gene subfamily. Drug Metab Dispos 17: 197-207
    • (1989) Drug Metab Dispos , vol.17 , pp. 197-207
    • Combalbert, J.1    Fabre, I.2    Fabre, G.3
  • 9
    • 0019973616 scopus 로고
    • Changes in platelet function and blood serotonin level in migraine patients during treatment with femoxetine
    • Dalsgaard-Nielsen J, le Fèvre Honorè P, Zeeberg I (1982) Changes in platelet function and blood serotonin level in migraine patients during treatment with femoxetine. Acta Neurol Scand 66: 191-198
    • (1982) Acta Neurol Scand , vol.66 , pp. 191-198
    • Dalsgaard-Nielsen, J.1    Le Fèvre Honorè, P.2    Zeeberg, I.3
  • 10
    • 0025344378 scopus 로고
    • Cytochrome P450 isoenzymes, epoxide hydrolase and glutathione transferases in rat and human hepatic and extra-hepatic tissues
    • De Waziers I, Cugnene PH, Yang CS, Leroux JP, Beaune PH (1990) Cytochrome P450 isoenzymes, epoxide hydrolase and glutathione transferases in rat and human hepatic and extra-hepatic tissues. J Pharmacol Exp Ther 253: 387-394
    • (1990) J Pharmacol Exp Ther , vol.253 , pp. 387-394
    • De Waziers, I.1    Cugnene, P.H.2    Yang, C.S.3    Leroux, J.P.4    Beaune, P.H.5
  • 11
    • 0026445458 scopus 로고
    • Adrenaline: Relationship between infusion rate, plasma concentration, metabolic and haemodynamic effects in volunteers
    • Ensinger H, Lindner KH, Dirks B, Kilian J, Grunert A, Ahnefeld FW (1992) Adrenaline: relationship between infusion rate, plasma concentration, metabolic and haemodynamic effects in volunteers. Eur J Anaesthesiol 9: 435-446
    • (1992) Eur J Anaesthesiol , vol.9 , pp. 435-446
    • Ensinger, H.1    Lindner, K.H.2    Dirks, B.3    Kilian, J.4    Grunert, A.5    Ahnefeld, F.W.6
  • 12
    • 0027443245 scopus 로고
    • Regiospecific expression of cytochrome P-450s and microsomal epoxide hydrolase in human brain tissue
    • Farin FM, Omiecinski CJ (1993) Regiospecific expression of cytochrome P-450s and microsomal epoxide hydrolase in human brain tissue. J Toxicol Environ Health 40: 317-335
    • (1993) J Toxicol Environ Health , vol.40 , pp. 317-335
    • Farin, F.M.1    Omiecinski, C.J.2
  • 14
    • 0025999285 scopus 로고
    • In vitro forecasting of drugs which may interfere with the biotransformation of midazolam
    • Gascon MP, Dayer P (1991) In vitro forecasting of drugs which may interfere with the biotransformation of midazolam. Eur J Clin Pharmacol 41: 573-578
    • (1991) Eur J Clin Pharmacol , vol.41 , pp. 573-578
    • Gascon, M.P.1    Dayer, P.2
  • 15
    • 0028234586 scopus 로고
    • Regioselective biotransformation of midazolam by members of the human cytochrome P450 3A (CYP3A) sub-family
    • Gorski JC, Hall SD, Jones DR, VandenBranden M, Wrighton SA (1994) Regioselective biotransformation of midazolam by members of the human cytochrome P450 3A (CYP3A) sub-family. Biochem Pharmacol 47: 1643-1653
    • (1994) Biochem Pharmacol , vol.47 , pp. 1643-1653
    • Gorski, J.C.1    Hall, S.D.2    Jones, D.R.3    VandenBranden, M.4    Wrighton, S.A.5
  • 16
    • 0029776066 scopus 로고    scopus 로고
    • Inhibition of human cytochrome P450-3A isoforms by fluoxetine and norfluoxetine: In vitro and in vivo studies
    • Greenblatt DJ, von Moltke LL, Schmider J, Harmatz JS, Shader RI (1996) Inhibition of human cytochrome P450-3A isoforms by fluoxetine and norfluoxetine: in vitro and in vivo studies. J Clin Pharmacol 36: 792-798
    • (1996) J Clin Pharmacol , vol.36 , pp. 792-798
    • Greenblatt, D.J.1    Von Moltke, L.L.2    Schmider, J.3    Harmatz, J.S.4    Shader, R.I.5
  • 17
    • 0022998708 scopus 로고
    • Characterization of rat and human liver microsomal cytochrome P-450 forms involved in nifedipine oxidation, a prototype for genetic polymorphism in oxidative drug metabolism
    • Guengerich FP, Martin MV, Beaune PH, Kremers P, Wolff T, Waxman DJ (1986) Characterization of rat and human liver microsomal cytochrome P-450 forms involved in nifedipine oxidation, a prototype for genetic polymorphism in oxidative drug metabolism. J Biol Chem 261: 5051-5060
    • (1986) J Biol Chem , vol.261 , pp. 5051-5060
    • Guengerich, F.P.1    Martin, M.V.2    Beaune, P.H.3    Kremers, P.4    Wolff, T.5    Waxman, D.J.6
  • 18
    • 0030460183 scopus 로고    scopus 로고
    • Effect of quinapril therapy on blood pressure and serotonin change in patients with mild to moderate hypertension
    • Huang JL, Cheng FC, Chen YT, Ting CT (1996) Effect of quinapril therapy on blood pressure and serotonin change in patients with mild to moderate hypertension. Chung Hua I Hsueh Tsa Chih 58: 329-334
    • (1996) Chung Hua I Hsueh Tsa Chih , vol.58 , pp. 329-334
    • Huang, J.L.1    Cheng, F.C.2    Chen, Y.T.3    Ting, C.T.4
  • 20
    • 0026662330 scopus 로고
    • Brain cytochrome P450 and testosterone metabolism by rat brain subcellular fractions: Presence of cytochrome P450 3A immunoreactive protein in rat brain mitochondria
    • Jayyosi Z, Cooper KO, Thomas PE (1992) Brain cytochrome P450 and testosterone metabolism by rat brain subcellular fractions: presence of cytochrome P450 3A immunoreactive protein in rat brain mitochondria. Arch Biochem Biophys 298: 265-270
    • (1992) Arch Biochem Biophys , vol.298 , pp. 265-270
    • Jayyosi, Z.1    Cooper, K.O.2    Thomas, P.E.3
  • 21
    • 0342468270 scopus 로고    scopus 로고
    • Detection of a CYP3A5 allelic variant: A candidate for the polymorphic expression of the protein?
    • Jounaïdi Y, Hyrailles V, Gervot L, Mauril P (1996) Detection of a CYP3A5 allelic variant: a candidate for the polymorphic expression of the protein? Biochem Biophys Res Commun 221: 466-470
    • (1996) Biochem Biophys Res Commun , vol.221 , pp. 466-470
    • Jounaïdi, Y.1    Hyrailles, V.2    Gervot, L.3    Mauril, P.4
  • 26
  • 28
    • 0032520750 scopus 로고    scopus 로고
    • Regional distribution of individual forms of cytochrome P450 mRNA in normal adult human brain
    • McFayden MCE, Melvin WT, Murray GI (1998) Regional distribution of individual forms of cytochrome P450 mRNA in normal adult human brain. Biochem Pharmacol 55: 825-830
    • (1998) Biochem Pharmacol , vol.55 , pp. 825-830
    • McFayden, M.C.E.1    Melvin, W.T.2    Murray, G.I.3
  • 29
    • 0025980557 scopus 로고
    • Determination of melatonin and monoamines in rat pineal using reversed-phase ion-interaction chromotography with fluorescence detection
    • Mills MH, Finlay DC, Haddad PR (1991) Determination of melatonin and monoamines in rat pineal using reversed-phase ion-interaction chromotography with fluorescence detection. J Chromatogr 564: 93-102
    • (1991) J Chromatogr , vol.564 , pp. 93-102
    • Mills, M.H.1    Finlay, D.C.2    Haddad, P.R.3
  • 30
    • 0027243182 scopus 로고
    • Tryptamine: A metabolite of tryptophan implicated in various neurophyschiatric disorders
    • Mosseau DD (1993) Tryptamine: a metabolite of tryptophan implicated in various neurophyschiatric disorders. Metab Brain Dis 8: 1-44
    • (1993) Metab Brain Dis , vol.8 , pp. 1-44
    • Mosseau, D.D.1
  • 33
    • 0016322145 scopus 로고
    • Dietary regulation of brain tryptophan metabolism by plasma ratio of free tryptophan and neutral amino acids in humans
    • Perez-Cruet J, Chase TN, Murphy DL (1974) Dietary regulation of brain tryptophan metabolism by plasma ratio of free tryptophan and neutral amino acids in humans. Nature 248: 693-695
    • (1974) Nature , vol.248 , pp. 693-695
    • Perez-Cruet, J.1    Chase, T.N.2    Murphy, D.L.3
  • 35
    • 0018832488 scopus 로고
    • Relationships in healthy volunteers between concentrations of monoamine metabolites in cerebrospinal fluid and family history of psychiatric morbidity
    • Sedvall G, Fyro B, Gullberg B, Nyback H, Wiesel FA, Wode-Helgodt B (1980) Relationships in healthy volunteers between concentrations of monoamine metabolites in cerebrospinal fluid and family history of psychiatric morbidity. Br J Psychiatry 136: 366-374
    • (1980) Br J Psychiatry , vol.136 , pp. 366-374
    • Sedvall, G.1    Fyro, B.2    Gullberg, B.3    Nyback, H.4    Wiesel, F.A.5    Wode-Helgodt, B.6
  • 37
    • 0028237729 scopus 로고
    • Interindividual variations in human liver cytochromes P450 enzymes involved in the oxidations of drugs, carcinogens and toxic chemicals: Studies with liver microsomes of 30 Japanese and 30 Caucasians
    • Shimada T, Yamazaki H, Mimura M, Inui Y, Guenguerich FP (1994) Interindividual variations in human liver cytochromes P450 enzymes involved in the oxidations of drugs, carcinogens and toxic chemicals: studies with liver microsomes of 30 Japanese and 30 Caucasians. J Pharmacol Exp Ther 270: 414-423
    • (1994) J Pharmacol Exp Ther , vol.270 , pp. 414-423
    • Shimada, T.1    Yamazaki, H.2    Mimura, M.3    Inui, Y.4    Guenguerich, F.P.5
  • 39
    • 0029743080 scopus 로고    scopus 로고
    • Midazolam hydroxylation by human liver microsomes in vitro: Inhibition by fluoxetine, norfluoxetine, and by azole antifungal agents
    • von Moltke LL, Greenblatt DJ, Schmider J, Duan SX, Wright CE, Harmatz JS, Shader RI (1996) Midazolam hydroxylation by human liver microsomes in vitro: inhibition by fluoxetine, norfluoxetine, and by azole antifungal agents. J Clin Pharmacol 36: 783-791
    • (1996) J Clin Pharmacol , vol.36 , pp. 783-791
    • Von Moltke, L.L.1    Greenblatt, D.J.2    Schmider, J.3    Duan, S.X.4    Wright, C.E.5    Harmatz, J.S.6    Shader, R.I.7
  • 41
    • 0028071759 scopus 로고
    • Noninvasive test of CYP3A enzymes
    • Watkins PB (1994) Noninvasive test of CYP3A enzymes. Pharmacogenetics 4: 171-184
    • (1994) Pharmacogenetics , vol.4 , pp. 171-184
    • Watkins, P.B.1
  • 42
    • 0028361593 scopus 로고
    • Inhibition of human CYP3A catalyzed 1′-hydroxy midazolam formation by ketoconazole, nifedipine, erythromycin, cimetidine and nizatidine
    • Wrighton SA, Ring BJ (1994) Inhibition of human CYP3A catalyzed 1′-hydroxy midazolam formation by ketoconazole, nifedipine, erythromycin, cimetidine and nizatidine. Pharm Res 11: 921-924
    • (1994) Pharm Res , vol.11 , pp. 921-924
    • Wrighton, S.A.1    Ring, B.J.2
  • 43
    • 0026750647 scopus 로고
    • The human hepatic cytochromes P450 involved in drug metabolism
    • Wrighton SA, Stevens JC (1992) The human hepatic cytochromes P450 involved in drug metabolism. Crit Rev Toxicol 22: 1-21
    • (1992) Crit Rev Toxicol , vol.22 , pp. 1-21
    • Wrighton, S.A.1    Stevens, J.C.2
  • 44
    • 0027168405 scopus 로고
    • Oxidation of the antihistaminic drug terfenadine in human liver microsomes: Role of cytochrome P-450 3A(4) in N-dealkylation and C-hydroxylation
    • Yun CH, Okerholm RA, Guengerich FP (1993) Oxidation of the antihistaminic drug terfenadine in human liver microsomes: role of cytochrome P-450 3A(4) in N-dealkylation and C-hydroxylation. Drug Metab Dispos 21: 403-409
    • (1993) Drug Metab Dispos , vol.21 , pp. 403-409
    • Yun, CH.1    Okerholm, R.A.2    Guengerich, F.P.3
  • 45
    • 0018908458 scopus 로고
    • Integrated concentration of epinephrine and norepinephrine in normal subjects and in patients with mild essential hypertension
    • Zadik Z, Hamilton BP, Kowarski AA (1980) Integrated concentration of epinephrine and norepinephrine in normal subjects and in patients with mild essential hypertension. J Clin Endocrinol Metab 50: 842-845
    • (1980) J Clin Endocrinol Metab , vol.50 , pp. 842-845
    • Zadik, Z.1    Hamilton, B.P.2    Kowarski, A.A.3


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