Pyrrolo[3,4-c]-β-carboline-diones as a novel class of inhibitors of the platelet- derived growth factor receptor kinase

European Journal of Medicinal Chemistry

Volumn 35, Issue 4, 2000, Pages 413-427

  Teller, Steffen ^a   Eluwa, Stella ^b   Koller, Markus ^b   Uecker, Andrea ^a   Beckers, Thomas ^c   Baasner, Silke ^c   Böhmer, Frank D ^a   Mahboobi, Siavosh ^b  

^a FRIEDRICH SCHILLER UNIVERSITY JENA   (Germany)

^b UNIVERSITY OF REGENSBURG   (Germany)

^c ASTA MEDICA AG   (Germany)

Author keywords

PDGF receptor; Signal transduction; Tyrosine kinase; carbolines

Indexed keywords

BETA CARBOLINE DERIVATIVE; PLATELET DERIVED GROWTH FACTOR RECEPTOR; PROTEIN KINASE INHIBITOR; PYRROLE DERIVATIVE;

ANIMAL CELL; ARTICLE; AUTOPHOSPHORYLATION; CELL STRAIN 3T3; DRUG ACTIVITY; DRUG EFFECT; DRUG SCREENING; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME SPECIFICITY; NONHUMAN; PROTEIN PHOSPHORYLATION; SIGNAL TRANSDUCTION;

EID: 0034128465     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0223-5234(00)00140-9     Document Type: Article

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