-
1
-
-
0021153959
-
Central cardiovascular effects of the α-adrenergic drugs. Differences between catecholamines and imidazolines
-
Bousquet P., Feldman J., Schwartz J. Central cardiovascular effects of the α-adrenergic drugs. Differences between catecholamines and imidazolines. J. Pharmacol. Exp. Ther. 230:1984;232-236.
-
(1984)
J. Pharmacol. Exp. Ther.
, vol.230
, pp. 232-236
-
-
Bousquet, P.1
Feldman, J.2
Schwartz, J.3
-
3
-
-
0028990748
-
1-imidazoline receptor. Definition, characterization, distribution, and trans-membrane signaling
-
1-imidazoline receptor. Definition, characterization, distribution, and trans-membrane signaling. Ann. N.Y. Acad. Sci. 763:1995;22-42.
-
(1995)
Ann. N.Y. Acad. Sci.
, vol.763
, pp. 22-42
-
-
Ernsberger, P.1
Graves, M.E.2
Graff, L.M.3
Zakieh, N.4
Nguyen, P.5
-
4
-
-
0030639995
-
1-imidazoline receptor: From binding site to therapeutic target in cardiovascular disease
-
Suppl.
-
1-imidazoline receptor: from binding site to therapeutic target in cardiovascular disease. J. Hypertens. 15(1):1997;S9-S23. Suppl.
-
(1997)
J. Hypertens.
, vol.15
, Issue.1
, pp. 9-S23
-
-
Ernsberger, P.1
Friedman, J.E.2
Koletsky, R.J.3
-
6
-
-
0026043081
-
Regulation of sigma receptors and responsiveness to guanine nucleotides following repeated exposure to haloperidol: Further evidence for multiple sigma binding sites
-
Itzhak Y., Stein I. Regulation of sigma receptors and responsiveness to guanine nucleotides following repeated exposure to haloperidol: further evidence for multiple sigma binding sites. Brain Res. 566:1991;166-172.
-
(1991)
Brain Res.
, vol.566
, pp. 166-172
-
-
Itzhak, Y.1
Stein, I.2
-
7
-
-
0030582657
-
Cloning and functional expression of the human type 1 sigma receptor (hSigmaR1)
-
Kekuda R., Prasad P.D., Fei Y.J., Leibach F.H., Ganapathy V. Cloning and functional expression of the human type 1 sigma receptor (hSigmaR1). Biochem. Biophys. Res. Commun. 229:1996;553-558.
-
(1996)
Biochem. Biophys. Res. Commun.
, vol.229
, pp. 553-558
-
-
Kekuda, R.1
Prasad, P.D.2
Fei, Y.J.3
Leibach, F.H.4
Ganapathy, V.5
-
8
-
-
0028269271
-
Agmatine: An endogenous clonidine-displacing substance in the brain
-
Li G., Regunathan S., Barrow C.J., Eshraghi J., Cooper R., Reis D.J. Agmatine: an endogenous clonidine-displacing substance in the brain. Science. 263:1994;966-969.
-
(1994)
Science
, vol.263
, pp. 966-969
-
-
Li, G.1
Regunathan, S.2
Barrow, C.J.3
Eshraghi, J.4
Cooper, R.5
Reis, D.J.6
-
9
-
-
0017064976
-
The effects of morphine and nalorphine-like drugs in the nondependent and morphine-dependent chronic spinal dog
-
Martin W.R., Eades C.G., Thomson J.A., Happler R.E., Gilbert P.E. The effects of morphine and nalorphine-like drugs in the nondependent and morphine-dependent chronic spinal dog. J. Pharmacol. Exp. Ther. 197:1976;517-532.
-
(1976)
J. Pharmacol. Exp. Ther.
, vol.197
, pp. 517-532
-
-
Martin, W.R.1
Eades, C.G.2
Thomson, J.A.3
Happler, R.E.4
Gilbert, P.E.5
-
10
-
-
0026778766
-
Keeping an eye on the I site: Imidazoline preferring receptors
-
Michel M.C., Ernsberger P. Keeping an eye on the I site: imidazoline preferring receptors. Trends Pharmacol. Sci. 13:1992;369-370.
-
(1992)
Trends Pharmacol. Sci.
, vol.13
, pp. 369-370
-
-
Michel, M.C.1
Ernsberger, P.2
-
12
-
-
0030949390
-
The mysteries of sigma receptors: New family members reveal a role in cholesterol synthesis
-
Moebius F.F., Striessnig J., Glossman H. The mysteries of sigma receptors: new family members reveal a role in cholesterol synthesis. Trends Pharmacol. Sci. 18:1997;67-70.
-
(1997)
Trends Pharmacol. Sci.
, vol.18
, pp. 67-70
-
-
Moebius, F.F.1
Striessnig, J.2
Glossman, H.3
-
13
-
-
0030759252
-
Imidazoline receptors: Basic knowledge, recent advances and future prospects for therapy and diagnosis
-
Molderings G.J. Imidazoline receptors: basic knowledge, recent advances and future prospects for therapy and diagnosis. Drug Future. 22:1997;757-772.
-
(1997)
Drug Future
, vol.22
, pp. 757-772
-
-
Molderings, G.J.1
-
15
-
-
0028199907
-
The effects of sigma ligands and neuropeptide Y on N-methyl-D-aspartate-induced neuronal activation of CA3 dorsal hippocampus neurons are differentially affected by pertussin toxin
-
Monnet F.P., Debonnel G., Bergeron R., Gronier B., de Montigny C. The effects of sigma ligands and neuropeptide Y on N-methyl-D-aspartate-induced neuronal activation of CA3 dorsal hippocampus neurons are differentially affected by pertussin toxin. Br. J. Pharmacol. 112:1994;709-715.
-
(1994)
Br. J. Pharmacol.
, vol.112
, pp. 709-715
-
-
Monnet, F.P.1
Debonnel, G.2
Bergeron, R.3
Gronier, B.4
De Montigny, C.5
-
16
-
-
0033602524
-
Design, synthesis, structure-activity relationships, and biological characterization of novel arylalkoxyphenylalkylamine σ ligands as potential antipsychotic drugs
-
Nakazato A., Ohta K., Sekiguchi Y., Okuyama S., Chaki S., Kawashima Y., Hatayama K. Design, synthesis, structure-activity relationships, and biological characterization of novel arylalkoxyphenylalkylamine σ ligands as potential antipsychotic drugs. J. Med. Chem. 42:1999;1076-1087.
-
(1999)
J. Med. Chem.
, vol.42
, pp. 1076-1087
-
-
Nakazato, A.1
Ohta, K.2
Sekiguchi, Y.3
Okuyama, S.4
Chaki, S.5
Kawashima, Y.6
Hatayama, K.7
-
17
-
-
0031008545
-
Imidazoline receptor: Qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity
-
Pigini M., Bousquet P., Carotti A., Dontenwill M., Giannella M., Moriconi R., Piergentili A., Quaglia W., Tayebati S.K., Brasili L. Imidazoline receptor: qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity. Bioorg. Med. Chem. 5:1997;843-856.
-
(1997)
Bioorg. Med. Chem.
, vol.5
, pp. 843-856
-
-
Pigini, M.1
Bousquet, P.2
Carotti, A.3
Dontenwill, M.4
Giannella, M.5
Moriconi, R.6
Piergentili, A.7
Quaglia, W.8
Tayebati, S.K.9
Brasili, L.10
-
18
-
-
0032217337
-
2 imidazoline receptor: The role of lipophilicity in quantitative structure-activity relationship models
-
2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models. Bioorg. Med. Chem. 6:1998;2245-2260.
-
(1998)
Bioorg. Med. Chem.
, vol.6
, pp. 2245-2260
-
-
Pigini, M.1
Bousquet, P.2
Brasili, L.3
Carrieri, A.4
Cavagna, R.5
Dontenwill, M.6
Gentili, F.7
Giannella, M.8
Leonetti, F.9
Piergentili, A.10
Quaglia, W.11
Carotti, A.12
-
19
-
-
0025923670
-
3H ]-p-aminoclonidine to alpha 2-adrenoceptor state plus a non-adrenergic sites on human platelet plasma membranes
-
3H ]-p-aminoclonidine to alpha 2-adrenoceptor state plus a non-adrenergic sites on human platelet plasma membranes Biochem. Pharmacol. 42:1991;569-584.
-
(1991)
Biochem. Pharmacol.
, vol.42
, pp. 569-584
-
-
Piletz, J.E.1
Andorn, A.C.2
Unnerstall, J.R.3
Halaris, A.4
-
20
-
-
0032492927
-
1 ligand
-
1 ligand. J. Med. Chem. 41:1998;1557-1560.
-
(1998)
J. Med. Chem.
, vol.41
, pp. 1557-1560
-
-
Quaglia, W.1
Giannella, M.2
Piergentili, A.3
Pigini, M.4
Brasili, L.5
Di Toro, R.6
Rossetti, L.7
Spampinato, S.8
Melchiorre, C.9
-
21
-
-
0026567933
-
A proposal for the classification of sigma binding sites
-
Quirion R., Bowen W.D., Itzhak Y., Junien J.L., Musacchio J.M., Rothman R.B., Su T.P., Tam S.W., Taylor D.P. A proposal for the classification of sigma binding sites. Trends. Pharmacol. Sci. 13:1992;85-86.
-
(1992)
Trends. Pharmacol. Sci.
, vol.13
, pp. 85-86
-
-
Quirion, R.1
Bowen, W.D.2
Itzhak, Y.3
Junien, J.L.4
Musacchio, J.M.5
Rothman, R.B.6
Su, T.P.7
Tam, S.W.8
Taylor, D.P.9
-
23
-
-
9844252872
-
Design and synthesis of imidazoline derivatives active on glucose homeostasis in rat model of type II diabetes: 1. Synthesis and biological activities of N-benzyl-N′-(arylalkyl)-2-(4′,5′-dihydro-1′H-imidazol- 2′-yl)piperazines
-
Rondu F., LE Bihan G., Wang X., Lamouri A., Touboul E., Dive G., Bellahsene T., Pfeiffer B., Renard P., Guardiola-Lamaitre B., Manechez D., Penicaud L., Ktorza A., Godfroid J.-J. Design and synthesis of imidazoline derivatives active on glucose homeostasis in rat model of type II diabetes: 1. Synthesis and biological activities of N-benzyl-N′-(arylalkyl)-2-(4′,5′-dihydro-1′H-imidazol- 2′-yl)piperazines. J. Med. Chem. 40:1997;3793-3803.
-
(1997)
J. Med. Chem.
, vol.40
, pp. 3793-3803
-
-
Rondu, F.1
Le Bihan, G.2
Wang, X.3
Lamouri, A.4
Touboul, E.5
Dive, G.6
Bellahsene, T.7
Pfeiffer, B.8
Renard, P.9
Guardiola-Lamaitre, B.10
Manechez, D.11
Penicaud, L.12
Ktorza, A.13
Godfroid, J.-J.14
-
25
-
-
0028795145
-
Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines
-
Vilner B.J., John C.S., Bowen W.D. Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines. Cancer Res. 55:1995;408-413.
-
(1995)
Cancer Res.
, vol.55
, pp. 408-413
-
-
Vilner, B.J.1
John, C.S.2
Bowen, W.D.3
-
26
-
-
0028825010
-
Progress in sigma receptor research
-
Wyrick S.D., Booth R. Progress in sigma receptor research. Drugs Future. 20:1995;1033-1044.
-
(1995)
Drugs Future
, vol.20
, pp. 1033-1044
-
-
Wyrick, S.D.1
Booth, R.2
|