Facilitation of acetylcholine release by SK-951, a benzofuran derivative, via the 5-hydroxytryptamine4 receptor in guinea pig stomach

Japanese Journal of Pharmacology

Volumn 82, Issue 2, 2000, Pages 138-143

  Takeda, Motohiro ^a   Tsukamoto, Katsura ^a   Sakurai Yamashita, Yasuko ^b   Suzuki, Tsunemasa ^a   Taniyama, Kohtaro ^b  

^a SANWA KAGAKU KENKYUSHO CO LTD   (Japan)

^b NAGASAKI UNIVERSITY SCHOOL OF MEDICINE   (Japan)

Author keywords

5 Hydroxytryptamine4 receptor; Acetylcholine release; Guinea pig stomach; SK 951; 125I SB207710 binding

Indexed keywords

1 METHYL 3 INDOLECARBOXYLIC ACID [1 [2 (METHYLSULFONYLAMINO)ETHYL] 4 PIPERIDINYLMETHYL] ESTER; 4 AMINO 5 CHLORO 2,3 DIHYDRO 2 METHYL N [2 (8 PYRROLIZIDINYL)ETHYL]BENZO[B]FURAN 7 CARBOXAMIDE; 8 AMINO 7 CHLORO 1,4 BENZODIOXAN 5 CARBOXYLIC ACID 1 BUTYL 4 PIPERIDINYLMETHYL ESTER; 8 AMINO 7 IODO 1,4 BENZODIOXAN 5 CARBOXYLIC ACID 1 BUTYL 4 PIPERIDINYLMETHYL ESTER; ACETYLCHOLINE; ATROPINE; BENZOFURAN DERIVATIVE; CALCIUM; SEROTONIN; SEROTONIN 4 RECEPTOR; TETRODOTOXIN; TRITIUM; UNCLASSIFIED DRUG;

ACETYLCHOLINE RELEASE; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG INHIBITION; DRUG RECEPTOR BINDING; GASTROINTESTINAL DISEASE; GASTROINTESTINAL MOTILITY; GUINEA PIG; IN VITRO STUDY; MALE; NONHUMAN; STOMACH; STOMACH MUSCLE;

EID: 0034014836     PISSN: 00215198     EISSN: None     Source Type: Journal    
DOI: 10.1254/jjp.82.138     Document Type: Article

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