Coupling efficacy and selectivity of the human μ-opioid receptor expressed as receptor-Gα fusion proteins in Escherichia coli

Journal of Neurochemistry

Volumn 75, Issue 3, 2000, Pages 1190-1199

  Stanasila, Laura ^a,b,c   Lim, William K ^a,b   Neubig, Richard R ^a,b   Pattus, Franc ^a,b  

^a UNIVERSITÉ DE STRASBOURG   (France)

^b UNIVERSITY OF MICHIGAN MEDICAL SCHOOL   (United States)

^c University of Lausanne Departement de Pharmacologie et de Toxicologie   (Switzerland)

Author keywords

Opioid receptor; Escherichia coli; G protein coupled receptors; Pharmacology; Receptor G protein fusion

Indexed keywords

DIPRENORPHINE; ENDOMORPHIN 1; ENKEPHALIN; HYBRID PROTEIN; MU OPIATE RECEPTOR;

ARTICLE; CARBOXY TERMINAL SEQUENCE; CHIMERA; CONFORMATIONAL TRANSITION; COUPLING FACTOR; ESCHERICHIA COLI; GASTROINTESTINAL MOTILITY; LIGAND BINDING; NEUROMODULATION; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN FAMILY; RECEPTOR AFFINITY; RECEPTOR DOWN REGULATION;

ANIMALS; BRAIN; CATTLE; DIPRENORPHINE; ENKEPHALIN, ALA(2)-MEPHE(4)-GLY(5)-; ESCHERICHIA COLI; GTP-BINDING PROTEIN ALPHA SUBUNIT, GI2; GTP-BINDING PROTEIN ALPHA SUBUNITS, GI-GO; GTP-BINDING PROTEINS; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HETEROTRIMERIC GTP-BINDING PROTEINS; HUMANS; KINETICS; MORPHINE; OLIGOPEPTIDES; PROTO-ONCOGENE PROTEINS; RADIOLIGAND ASSAY; RECEPTORS, OPIOID, MU; RECOMBINANT FUSION PROTEINS; TRITIUM;

EID: 0033836350     PISSN: 00223042     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1471-4159.2000.0751190.x     Document Type: Article

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