Synthesis and PKC isozyme surrogate binding of indothiolactam-V, a new thioamide analogue of tumor promoting indolactam-V

Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 18, 2000, Pages 2087-2090

  Nakagawa, Yu ^a   Irie, Kazuhiro ^a   Ohigashi, Hajime ^a   Hayashi, Hideo ^b   Wender, Paul A ^c  

^a KYOTO UNIVERSITY   (Japan)

^b Osaka City University   (Japan)

^c STANFORD UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMIDE; INDOLACTAM V; INDOTHIOLACTAM V; ISOENZYME; PROTEIN KINASE C; THIOAMIDE; TUMOR PROMOTER; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG BINDING; ENZYME ACTIVATION; ENZYME BINDING; ENZYME MODIFICATION; NONHUMAN; STREPTOMYCES; TUMOR PROMOTION;

BINDING, COMPETITIVE; CARCINOGENS; ENZYME ACTIVATION; INDOLES; ISOENZYMES; LACTAMS; MAGNETIC RESONANCE SPECTROSCOPY; PEPTIDE FRAGMENTS; PHORBOL 12,13-DIBUTYRATE; PROTEIN BINDING; PROTEIN KINASE C; THIOAMIDES;

ACTINOBACTERIA (CLASS); STREPTOMYCES; UNCULTURED ACTINOMYCETE;

EID: 0033822235     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(00)00411-X     Document Type: Article

References (26)