Interaction of local anaesthetics with recombinant μ, κ, and δ opioid receptors expressed in Chinese hamster ovary cells

British Journal of Anaesthesia

Volumn 85, Issue 5, 2000, Pages 740-746

  Hirota, K ^a   Okawa, H ^a   Appadu, B L ^a   Grandy, D K ^b   Lambert, D G ^a  

^a LEICESTER ROYAL INFIRMARY   (United Kingdom)

^b OREGON HEALTH AND SCIENCE UNIVERSITY   (United States)

Author keywords

Anaesthetics local; Measurement techniques, radioligand binding; Metabolism, cAMP

Indexed keywords

ADENYLATE CYCLASE; BUPIVACAINE; CALCIUM ION; CYCLIC AMP; DELTA OPIATE RECEPTOR; DIPRENORPHINE; ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE]; KAPPA OPIATE RECEPTOR; LIDOCAINE; LOCAL ANESTHETIC AGENT; MU OPIATE RECEPTOR; NALOXONE; OPIATE; OPIATE RECEPTOR; PRILOCAINE; PROCAINE; RECOMBINANT RECEPTOR; SPIRADOLINE; TETRACAINE; TRITIUM;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CELL LINE; CHO CELL; CONTROLLED STUDY; DRUG ACTIVITY; DRUG MECHANISM; DRUG POTENTIATION; DRUG PROTEIN BINDING; FEMALE; GENETIC TRANSFECTION; HAMSTER; ISOMER; ISOTOPE LABELING; LOCAL ANESTHESIA; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION;

EID: 0033754257     PISSN: 00070912     EISSN: None     Source Type: Journal    
DOI: 10.1093/bja/85.5.740     Document Type: Article

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