-
6
-
-
85034129924
-
-
note
-
This is the average distance in the HIV-1 protease structures with the PDB codes 1HVI, 1HVJ, 1HVK, and 1HVL.
-
-
-
-
7
-
-
0028328704
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-
Hosur, M. V.; Bhat, T. N.; Kempf, D. J.; Baldwin E. T.; Liu, B.; Gulnik, S.; Wideburg, N. E.; Norbeck, D. W.; Appelt, K.; Erickson, J. W. J. Am. Chem. Soc. 1994, 116, 847.
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8
-
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0028113650
-
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(a) Thompson, S. K.; Murthy, K. H.; Zhao, B.; Winborne, E.; Green, D. W.; Fisher, S. M.; DesJarlais, R. L.; Tomaszek,T. A., Jr.; Meek, T. D.; Gleason, J. G.; Abdel-Meguid, S. S. J. Med. Chem. 1994, 37, 3100.
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9
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0028116504
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(b) Abdel-Meguid, S. S.; Metcalf, B. W.; Carr, T. J.; Demarsh, P.; DesJarlais, R. L.; Fisher, S.; Green, D. W.; Ivanoff, L.; Lambert, D. M.; Murthy, K. H. M.; Petteway, S. R., Jr.; Pitts, W. J.; Tomaszek, T. A. Jr.; Winborne, E.; Zhao, B.; Dreyer, G. B.; Meek, T. D. Biochemistry 1994, 33, 11671.
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10
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12944322516
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Thaisrivongs, S.17
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11
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0001241103
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(d) Han, Q.; Chang, C.-H.; Li, R.; Ru, Y.; Jadhav, P. K.; Lam, P. Y. S. J. Med. Chem. 1998, 41, 2019.
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12
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15644373221
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(e) De Lucca, G. V.; Kim, U. T.; Liang, J.; Cordova, B.; Klabe, R. M.; Garber, S.; Bacheler, L. T.; Lam, G. N.; Wright, M. R.; Logue, K. A.; Erickson-Viitanen, S.; Ko, S. S.; Trainer, G. L. J. Med. Chem. 1998, 41, 2411.
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Trainer, G.L.13
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14
-
-
85034150100
-
-
note
-
Spectra are included with the Supporting Information.
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-
-
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15
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0025274362
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Richards, A. D.; Phylip, L. H.; Farmerie, W. G.; Scarborough, P. E.; Alvarez, A.; Dunn, B. M.; Hirel, P.-H.; Konvalinka, J.; Strop, P.; Pavlickova, L.; Kostka, V.; Kay, J. J. Biol. Chem. 1990, 265, 7733. Our inhibitor assays were done at 320 nm instead of 300 nm because this wavelength minimized background variations.
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17
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85034135112
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-
note
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i values will be published at a later date.
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19
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23
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85034124313
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Copper(II) chelates as a new generation of non-peptide inhibitors of the human immunodeficiency virus
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Richmond, VA, June 14-18; Abstract A-21
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13044290051
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