Benzofuro[3,2-b]pyridines as mixed ET(A)/ET(B) and selective ET(B) endothelin receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 4, 1999, Pages 619-622

  Mederski, Werner W K R ^a   Osswald, Mathias ^a   Dorsch, Dieter ^a   Christadler, Maria ^a   Schmitges, Claus Jochen ^a   Wilm, Claudia ^a  

^a MERCK KGAA   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOFURAN DERIVATIVE; BENZOFURO[3,2 B]PYRIDINE DERIVATIVE; ENDOTHELIN; ENDOTHELIN A RECEPTOR ANTAGONIST; ENDOTHELIN B RECEPTOR ANTAGONIST; PYRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; BLOOD VESSEL REACTIVITY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG SYNTHESIS; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION;

ANIMALS; ENDOTHELIN-1; ENDOTHELIUM, VASCULAR; KIDNEY; PYRIDINES; RABBITS; RATS; RECEPTOR, ENDOTHELIN A; RECEPTOR, ENDOTHELIN B; RECEPTORS, ENDOTHELIN; STRUCTURE-ACTIVITY RELATIONSHIP; SWINE;

EID: 0033593861     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00040-2     Document Type: Article

References (13)

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