1,4-Diaryl-2-oxo-1,2-dihydro-quinoline-3-carboxylic acids as endothelin receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 14, 1997, Pages 1883-1886

  Mederski, Werner W K R ^a   Osswald, Mathias ^a   Dorsch, Dieter ^a   Christadler, Maria ^a   Schmitges, Claus Jochen ^a   Wilm, Claudia ^a  

^a MERCK KGAA   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

1,2 DIHDYRO 1 (2,5 DIMETHOXYPBENZYL) 6 ETHOXY 4 (4 METHOXYPHENYL) 2 OXO 3 QUINOLINECARBOXYLIC ACID; ENDOTHELIN A RECEPTOR; ENDOTHELIN B RECEPTOR; ENDOTHELIN RECEPTOR; ENDOTHELIN RECEPTOR ANTAGONIST; QUINOLINE DERIVATIVE; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; AORTA; ARTICLE; BINDING AFFINITY; CELL MEMBRANE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; ENDOTHELIUM; IN VITRO STUDY; KIDNEY; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION; SWINE; VASOCONSTRICTION;

ANIMALIA; SUS SCROFA;

EID: 0030793673     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00319-3     Document Type: Article

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