Inhibition mechanism of cathepsin L-specific inhibitors based on the crystal structure of papain-CLIK148 complex

Biochemical and Biophysical Research Communications

Volumn 266, Issue 2, 1999, Pages 411-416

  Tsuge, Hideaki ^a   Nishimura, Tomohiro ^a   Tada, Yukio ^b   Asao, Tetsuji ^b   Turk, Dusan ^c   Turk, Vito ^c   Katunuma, Nobuhiko ^a  

^a TOKUSHIMA BUNRI UNIVERSITY   (Japan)

^b TAIHO PHARMACEUTICAL CO LTD   (Japan)

^c JO EF STEFAN INSTITUTE   (Slovenia)

Author keywords

Cathepsin L; Inhibitor; Papain; X ray crystallography

Indexed keywords

CATHEPSIN L; ENZYME INHIBITOR; PAPAIN; PYRIDINE;

AMINO TERMINAL SEQUENCE; ARTICLE; CHEMICAL STRUCTURE; COMPLEX FORMATION; CRYSTAL STRUCTURE; HYDROPHOBICITY; PRIORITY JOURNAL;

EID: 0033590204     PISSN: 0006291X     EISSN: None     Source Type: Journal    
DOI: 10.1006/bbrc.1999.1830     Document Type: Article

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