(±)-4-[(N-allyl-cis-3-methyl-4-piperidinyl)phenylamino]-N,N-diethylbenza mide displays selective binding for the delta opioid receptor

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 20, 1999, Pages 3053-3056

  Thomas, James B ^a   Herault, Xavier M ^a   Rothman, Richard B ^b   Burgess, Jason P ^a   Mascarella, S Wayne ^a   Xu, Heng ^b   Horel, Robert B ^b   Dersch, Christina M ^b   Carroll, F Ivy ^a  

^a RTI INTERNATIONAL   (United States)

^b NIDA Addiction Research Center   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 [(N ALLYL CIS 3 METHYL 4 PIPERDINYL) PHENYLAMINO] N,N DIETHYLBENZAMIDE; 4 [(N ALLYL TRANS 3 METHYL 4 PIPERDINYL) PHENYLAMINO] N,N DIETHYLBENZAMIDE; BINALTORPHIMINE; DELTA OPIATE RECEPTOR; DELTA OPIATE RECEPTOR AGONIST; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; KAPPA OPIATE RECEPTOR; MU OPIATE RECEPTOR; NALTRINDOLE; OPIATE ANTAGONIST; RADIOLIGAND; UNCLASSIFIED DRUG; 4 ((N ALLYL 3 METHYL 4 PIPERIDINYL)PHENYLAMINO) N,N DIETHYLBENZAMIDE; 4 (ALPHA (4 ALLYL 2,5 DIMETHYL 1 PIPERAZINYL) 3 METHOXYBENZYL) N,N DIETHYLBENZAMIDE; 4 [ALPHA (4 ALLYL 2,5 DIMETHYL 1 PIPERAZINYL) 3 HYDROXYBENZYL] N,N DIETHYLBENZAMIDE; 4-((N-ALLYL-3-METHYL-4-PIPERIDINYL)PHENYLAMINO)-N,N-DIETHYLBENZAMIDE; 4-(ALPHA-(4-ALLYL-2,5-DIMETHYL-1-PIPERAZINYL)-3-METHOXYBENZYL)-N,N-DIETHYLBENZAMIDE; BENZAMIDE DERIVATIVE; PIPERAZINE DERIVATIVE; PIPERIDINE DERIVATIVE;

ARTICLE; BINDING AFFINITY; BINDING KINETICS; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; STRUCTURE ANALYSIS; CHEMISTRY; DRUG POTENTIATION; METABOLISM; RADIOASSAY;

BENZAMIDES; PIPERAZINES; PIPERIDINES; RADIOLIGAND ASSAY; RECEPTORS, OPIOID, DELTA;

EID: 0033581463     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00525-9     Document Type: Article

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