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Angewandte Chemie - International Edition

Volumn 38, Issue 24, 1999, Pages 3743-3748

The design of leadlike combinatorial libraries

(4) Teague, Simon J a Davis, Andrew M a Leeson, Paul D a Oprea, Tudor a

a ASTRAZENECA (United Kingdom)

Author keywords

Bioorganic chemistry; Combinatorial chemistry; Drug research; Structure activity relationships

Indexed keywords

3 [[4 (4 CHLOROPHENYL) 1 PIPERAZINYL]METHYL] 1H PYRROLO[2,3 B]PYRIDINE; 4 AMINOBUTYRIC ACID; 5 DIMETHYLAMINO N (3,4 DIMETHYL 5 ISOXAZOLYL) 1 NAPHTHALENESULFONAMIDE; BACLOFEN; CHLOROTHIAZIDE; CHLORPHENIRAMINE; CIMETIDINE; DOPAMINE; DRUG DERIVATIVE; EPROSARTAN; FUROSEMIDE; HISTAMINE; IPRONIAZID; ISONIAZID; LOSARTAN; MIFEPRISTONE; MUSCARINE; NORADRENALIN; OCTANOL; OXYTOCIN; PILOCARPINE; PROGESTERONE; PROPRANOLOL; SULFANILAMIDE; SULFATHIAZOLE; THIOPERAMIDE; WATER;

ARTICLE; BINDING AFFINITY; DRUG DESIGN; DRUG POTENCY; DRUG RESEARCH; HYDROGEN BOND; LIPOPHILICITY; MOLECULAR WEIGHT; PARTITION COEFFICIENT; PHYSICAL CHEMISTRY; STRUCTURE ACTIVITY RELATION;

EID: 0033576601 PISSN: 14337851 EISSN: None Source Type: Journal
DOI: 10.1002/(SICI)1521-3773(19991216)38:24<3743::AID-ANIE3743>3.0.CO;2-U Document Type: Article

Times cited : (789)

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