Benzodiazepine compounds as inhibitors of the Src protein tyrosine kinase: Screening of a combinatorial library of 1,4-benzodiazepines

Archives of Biochemistry and Biophysics

Volumn 368, Issue 2, 1999, Pages 394-400

  Ramdas, Latha ^a   Bunnin, Barry A ^b   Plunkett, Matthew J ^b   Sun, Gongqin ^a   Ellman, Jonathan ^b   Gallick, Gary ^a   Budde, Raymond J A ^a  

^a UNIVERSITY OF TEXAS MD ANDERSON CANCER CENTER   (United States)

^b UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

Benzodiazepines; Combinatorial library; Inhibitor; Multiple inhibition; Protein tyrosine kinase; Src

Indexed keywords

ADENOSINE TRIPHOSPHATE MAGNESIUM; BENZODIAZEPINE DERIVATIVE; FIBROBLAST GROWTH FACTOR RECEPTOR; PROTEIN TYROSINE KINASE; TRYPTOPHAN; TYROSINE;

ARTICLE; CANCER CELL CULTURE; CELL GROWTH; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG EFFECT; DRUG STRUCTURE; ENZYME INHIBITION; FIBROBLAST CULTURE; GROWTH INHIBITION; HUMAN; HUMAN CELL; PRIORITY JOURNAL;

EID: 0033567317     PISSN: 00039861     EISSN: None     Source Type: Journal    
DOI: 10.1006/abbi.1999.1313     Document Type: Article

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