Bivalency as a principle for proteasome inhibition

Proceedings of the National Academy of Sciences of the United States of America

Volumn 96, Issue 10, 1999, Pages 5418-5422

  Loidl, Günther ^a   Groll, Michael ^a   Musiol, Hans Jürgen ^a   Huber, Robert ^a   Moroder, Luis ^a  

^a MAX PLANCK INSTITUTE OF BIOCHEMISTRY   (Germany)

Author keywords

Polyoxyethylene; X ray structures

Indexed keywords

POLYOXYETHYLENE; PROTEASOME; PROTEASOME INHIBITOR;

ARTICLE; ENZYME ACTIVE SITE; ENZYME INHIBITION; ENZYME SPECIFICITY; ENZYME SUBSTRATE; INHIBITION KINETICS; MOLECULAR RECOGNITION; NONHUMAN; PRIORITY JOURNAL; SACCHAROMYCES CEREVISIAE; X RAY ANALYSIS;

ALDEHYDES; BINDING SITES; CYSTEINE ENDOPEPTIDASES; DRUG DESIGN; ENZYME INHIBITORS; MODELS, MOLECULAR; MULTIENZYME COMPLEXES; PEPTIDES; POLYETHYLENE GLYCOLS; PROTEASOME ENDOPEPTIDASE COMPLEX; PROTEIN FOLDING; SACCHAROMYCES CEREVISIAE; SUBSTRATE SPECIFICITY; X-RAY DIFFRACTION;

SACCHAROMYCES CEREVISIAE;

EID: 0033545942     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.96.10.5418     Document Type: Article

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