Synthesis, kinetic characterization and X-ray analysis of peptide aldehydes as inhibitors of the 20S proteasomes from Thermoplasma acidophilum and Saccharomyces cerevisiae

Biological Chemistry

Volumn 378, Issue 8, 1997, Pages 893-898

  Escherich, Achim ^a   Ditzel, Lars ^a   Musiol, Hans Jürgen ^a   Groll, Michael ^a   Huber, Robert ^a   Moroder, Luis ^a  

^a MAX PLANCK INSTITUTE OF BIOCHEMISTRY   (Germany)

Author keywords

Inhibition; Peptide aldehydes; Proteasome; X ray structures

Indexed keywords

ALDEHYDE DERIVATIVE; CHYMOTRYPSIN; PEPTIDE; PROTEASOME; PROTEINASE INHIBITOR;

ANALYSIS; ARCHAEBACTERIUM; ARTICLE; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME KINETICS; INHIBITION KINETICS; NONHUMAN; PRIORITY JOURNAL; SACCHAROMYCES CEREVISIAE; SYNTHESIS; X RAY CRYSTALLOGRAPHY;

ARCHAEA; SACCHAROMYCES CEREVISIAE; THERMOPLASMA ACIDOPHILUM;

EID: 0030861790     PISSN: 14316730     EISSN: None     Source Type: Journal    
DOI: 10.1515/bchm.1997.378.8.893     Document Type: Article

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