Preparation of L-N(α)-Fmoc-4-[di-(tert- butyl)phosphonomethyl]phenylalanine from L-tyrosine

Tetrahedron Asymmetry

Volumn 10, Issue 19, 1999, Pages 3727-3734

  Yao, Zhu Jun ^a   Gao, Yang ^a   Burke Jr , Terrence R ^a  

^a NATIONAL INSTITUTES OF HEALTH   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 (PHOSPHONOMETHYL)PHENYLALANINE; AMINO ACID DERIVATIVE; N ALPHA (9 FLUORENYLMETHOXYCARBONYL) 4 [(DI TERT BUTYL)PHOSPHONOMETHYL]PHENYLALANINE; PROTEIN TYROSINE KINASE; TYROSINE; UNCLASSIFIED DRUG;

ARTICLE; ENANTIOMER; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; RACEMIC MIXTURE; SIGNAL TRANSDUCTION; STEREOCHEMISTRY; SYNTHESIS;

EID: 0033461799     PISSN: 09574166     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0957-4166(99)00385-7     Document Type: Article

References (18)

1. Burke Jr., T. R.; Yao, Z.-J.; Smyth, M. S.; Ye, B. Curr. Pharm. Des. 1997, 3, 291-304.
2. Domchek, S. M.; Auger, K. R.; Chatterjee, S.; Burke, T. R.; Shoelson, S. E. Biochemistry 1992, 31, 9865-9870.
3. Yao, Z.-J.; King, C. R.; Cao, T.; Kelley, J.; Milne, G. W. A.; Voigt, J. H.; Burke Jr., T. R. J. Med. Chem. 1999, 42, 25-35.
4. Schoepfer, J.; Fretz, H.; Gay, B.; Furet, P.; GarciaEcheverria, C.; End, N.; Caravatti, G. Bioorg. Med. Chem. Lett. 1999, 9, 221-226.
5. Marseigne, I.; Roques, B. P. J. Org. Chem. 1988, 53, 3621-3624.
6. Garbay-Jaureguiberry, C.; McCort-Tranchepain, I.; Barbe, B.; Ficheux, D.; Roques, B. P. Tetrahedron: Asymmetry 1992, 3, 637-650.
7. Cushman, M.; Lee, E. S. Tetrahedron Lett. 1992, 33, 1193-1196.
8. Dow, R. L.; Bechle, B. M. Synlett. 1994, 293-294.
9. Burke Jr., T. R.; Russ, P.; Lim, B. Synthesis 1991, 11, 1019-1020.
10. Josien, H.; Matin, A.; Chassaing, G. Tetrahedron Lett. 1991, 32, 6547-6550.
11. Liu, W. Q.; Roques, B. P.; Garbay-Jaureguiberry, C. Tetrahedron: Asymmetry 1995, 6, 647-650.
12. Hartman, G. D.; Halczenko, H. Synth. Commun. 1991, 21, 2103-2107.
13. Yokomatsu, T.; Yamagishi, T.; Matsumoto, K.; Shibuya, S. Tetrahedron 1996, 52, 11725-11738.
14. Rasmussen, J. R.; Slinger, C. J.; Kordish, R. J.; Newman-Evans, D. D. J. Org. Chem. 1981, 46, 4843-4846.
15. Baczko, K.; Liu, W. Q.; Roques, B. P.; GarbayJaureguiberry, C. Tetrahedron 1996, 52, 2021-2030.
16. Whole animal studies with Pmp-containing Grb2 SH2 domain inhibitor 4 are currently in progress.
17. Rink, H. Tetrahedron Lett. 1987, 28, 3787-3790.
18. Burke, T. R.; Yao, Z. J.; Zhao, H.; Milne, G. W. A.; Wu, L.; Zhang, Z. Y.; Voigt, J. H. Tetrahedron 1998, 54, 9981-9994.