메뉴 건너뛰기




Volumn 39, Issue 4, 1999, Pages 184-190

Effect of selective estrogen receptor modulators on estrogen-sensitive tissues;Wirkung von selektiven ostrogen-rezeptor-modulatoren auf ostrogensensitive gewebe

Author keywords

Breast cancer; Droloxifene; Endometrium; Estrogen receptor; Idoxifene; Raloxifene; Selective estrogen receptor modulators; Tamoxifen; Toremifene

Indexed keywords

DROLOXIFENE; IDOXIFENE; RALOXIFENE; SELECTIVE ESTROGEN RECEPTOR MODULATOR; TAMOXIFEN; TOREMIFENE;

EID: 0033401268     PISSN: 10188843     EISSN: None     Source Type: Journal    
DOI: 10.1159/000022308     Document Type: Review
Times cited : (3)

References (41)
  • 1
    • 0025062215 scopus 로고
    • Role of the two activating domains of the oestrogen receptor in the cell-type and promoter-context dependent agonistic activity of the anti-oestrogen 4-hydroxytamoxifen
    • Berry M, Metzger D, Chambon P: Role of the two activating domains of the oestrogen receptor in the cell-type and promoter-context dependent agonistic activity of the anti-oestrogen 4-hydroxytamoxifen. EMBO J 1990;9:2811-2818.
    • (1990) EMBO J , vol.9 , pp. 2811-2818
    • Berry, M.1    Metzger, D.2    Chambon, P.3
  • 4
    • 0030593681 scopus 로고    scopus 로고
    • ERβ identification and characterization of a novel human estrogen receptor
    • Mosselman S, Polman J, Dijkema R: ERβ identification and characterization of a novel human estrogen receptor. FEBS Lett 1996;392: 49-53.
    • (1996) FEBS Lett , vol.392 , pp. 49-53
    • Mosselman, S.1    Polman, J.2    Dijkema, R.3
  • 5
    • 0030775052 scopus 로고    scopus 로고
    • In search of optimal long-term female hormone replacement: The potential of selective estrogen receptor modulators
    • Mitlak B, Cohen F: In search of optimal long-term female hormone replacement: The potential of selective estrogen receptor modulators. Horm Res 1997;48:155-163.
    • (1997) Horm Res , vol.48 , pp. 155-163
    • Mitlak, B.1    Cohen, F.2
  • 6
    • 0032134252 scopus 로고    scopus 로고
    • Therapeutic potential of selective estrogen receptor modulators
    • Gustafsson J: Therapeutic potential of selective estrogen receptor modulators. Curr Opin Chem Biol 1998;2:508-511.
    • (1998) Curr Opin Chem Biol , vol.2 , pp. 508-511
    • Gustafsson, J.1
  • 8
    • 0031037365 scopus 로고    scopus 로고
    • Behavioral effects of estrogen receptor gene disruption in male mice
    • Ogawa S, Lubahn D, Korach K, Pfaff D: Behavioral effects of estrogen receptor gene disruption in male mice. Proc Natl Acad Sci USA 1997;94:1476-1481.
    • (1997) Proc Natl Acad Sci USA , vol.94 , pp. 1476-1481
    • Ogawa, S.1    Lubahn, D.2    Korach, K.3    Pfaff, D.4
  • 9
    • 0031024192 scopus 로고    scopus 로고
    • Estrogen receptors are essential for female sexual receptivity
    • Rissman E, Early A, Taylor J, Korach K, Lubahn D: Estrogen receptors are essential for female sexual receptivity. Endocrinology 1997; 138:507-510.
    • (1997) Endocrinology , vol.138 , pp. 507-510
    • Rissman, E.1    Early, A.2    Taylor, J.3    Korach, K.4    Lubahn, D.5
  • 12
    • 0028233383 scopus 로고
    • Estrogen receptor associated proteins: Possible mediators of hormone-induced transcription
    • Halachmi S, Marden E. Martin G, MacKay H, Abbondanza C, Brown M: Estrogen receptor associated proteins: Possible mediators of hormone-induced transcription. Science 1993; 264:1455-1458.
    • (1993) Science , vol.264 , pp. 1455-1458
    • Halachmi, S.1    Marden, E.2    Martin, G.3    MacKay, H.4    Abbondanza, C.5    Brown, M.6
  • 14
    • 0030071445 scopus 로고    scopus 로고
    • Tripartite steroid hormone receptor pharmacology: Interaction with multiple effector sites as a basis for the cell-and promoter-specific action of these hormones
    • Katzenellenbogen J, O'Malley B, Katzenellenbogen B: Tripartite steroid hormone receptor pharmacology: Interaction with multiple effector sites as a basis for the cell-and promoter-specific action of these hormones. Mol Endocrinol 1996;10:119-131.
    • (1996) Mol Endocrinol , vol.10 , pp. 119-131
    • Katzenellenbogen, J.1    O'Malley, B.2    Katzenellenbogen, B.3
  • 15
    • 0029841146 scopus 로고    scopus 로고
    • Identification of an estrogen response element activated by metabolites of 17β-estradiol and raloxifene
    • Yang N, Venugopalan M, Hardikar S, Glasebrook A: Identification of an estrogen response element activated by metabolites of 17β-estradiol and raloxifene. Science 1996;273:1222-1225.
    • (1996) Science , vol.273 , pp. 1222-1225
    • Yang, N.1    Venugopalan, M.2    Hardikar, S.3    Glasebrook, A.4
  • 16
    • 0032508294 scopus 로고    scopus 로고
    • Interim analysis of the incidence of breast cancer in the Royal Marsden Hospital tamoxifen randomised chemoprevention trial
    • Powles T, Eeles R, Ashley S: Interim analysis of the incidence of breast cancer in the Royal Marsden Hospital tamoxifen randomised chemoprevention trial. Lancet 1998;352:98-101.
    • (1998) Lancet , vol.352 , pp. 98-101
    • Powles, T.1    Eeles, R.2    Ashley, S.3
  • 17
    • 0032246469 scopus 로고    scopus 로고
    • Tamoxifen in the treatment of patients with breast cancer: Results of the latest meta-analysis of prospective randomized clinical trials
    • Sevelda P: Tamoxifen in the treatment of patients with breast cancer: Results of the latest meta-analysis of prospective randomized clinical trials. Gynäkol Geburtshilfliche Rundsch 1998;38:81-84.
    • (1998) Gynäkol Geburtshilfliche Rundsch , vol.38 , pp. 81-84
    • Sevelda, P.1
  • 18
    • 0028053224 scopus 로고
    • Risk of endometrial cancer after tamoxifen treatment of breast cancer
    • Leeuwen F, Benraadt J: Risk of endometrial cancer after tamoxifen treatment of breast cancer. Lancet 1994;343:448-452.
    • (1994) Lancet , vol.343 , pp. 448-452
    • Leeuwen, F.1    Benraadt, J.2
  • 19
    • 0031746719 scopus 로고    scopus 로고
    • Abnormalities detected on transvaginal ultrasonography in tamoxifen-treated postmenopausal breast cancer patients may represent endometrial cystic atrophy
    • McGonigle K, Shaw S, Vasilev S, Odom-Maryon T, Roy S, Simpson J: Abnormalities detected on transvaginal ultrasonography in tamoxifen-treated postmenopausal breast cancer patients may represent endometrial cystic atrophy. Am J Obstet Gynecol 1998;178:1145-1150.
    • (1998) Am J Obstet Gynecol , vol.178 , pp. 1145-1150
    • McGonigle, K.1    Shaw, S.2    Vasilev, S.3    Odom-Maryon, T.4    Roy, S.5    Simpson, J.6
  • 20
    • 0031901924 scopus 로고    scopus 로고
    • The role of transvaginal ultrasound in the investigation of women with post-menopausal bleeding
    • Briley M, Lindsell D: The role of transvaginal ultrasound in the investigation of women with post-menopausal bleeding. Clin Radiol 1998; 53:502-505.
    • (1998) Clin Radiol , vol.53 , pp. 502-505
    • Briley, M.1    Lindsell, D.2
  • 21
    • 0031982689 scopus 로고    scopus 로고
    • Uterine side effects of tamoxifen: A need for systematic pretreatment screening
    • Berlière M, Charles A, Galant C, Donnez J: Uterine side effects of tamoxifen: A need for systematic pretreatment screening. Obstet Gynecol 1998;94:40-41.
    • (1998) Obstet Gynecol , vol.94 , pp. 40-41
    • Berlière, M.1    Charles, A.2    Galant, C.3    Donnez, J.4
  • 22
    • 0031013929 scopus 로고    scopus 로고
    • Comparative effects of droloxifene, tamoxifen and estrogen on bone, serum cholesterol, and uterine histology in the ovariectomized rat model
    • Ke H, Chen K, Simmons H, Qi H, Crawford D: Comparative effects of droloxifene, tamoxifen and estrogen on bone, serum cholesterol, and uterine histology in the ovariectomized rat model. Bone 1997;20:31-39.
    • (1997) Bone , vol.20 , pp. 31-39
    • Ke, H.1    Chen, K.2    Simmons, H.3    Qi, H.4    Crawford, D.5
  • 23
    • 0032052776 scopus 로고    scopus 로고
    • Antiestrogen stimulated human endometrial cancer growth: Laboratory and clinical considerations
    • Tonetti D, O'Regan R, Tanjore S, England G: Antiestrogen stimulated human endometrial cancer growth: Laboratory and clinical considerations. J Steroid Biochem Mol Biol 1998;65: 181-189.
    • (1998) J Steroid Biochem Mol Biol , vol.65 , pp. 181-189
    • Tonetti, D.1    O'Regan, R.2    Tanjore, S.3    England, G.4
  • 24
    • 0025301011 scopus 로고
    • Antiestrogenic and antitumor properties of the new triphenylethylene derivative toremifen in the rat
    • Di Salle E, Zaccheo T, Ornati G: Antiestrogenic and antitumor properties of the new triphenylethylene derivative toremifen in the rat. J Chem Biochem 1990;36:203-206.
    • (1990) J Chem Biochem , vol.36 , pp. 203-206
    • Di Salle, E.1    Zaccheo, T.2    Ornati, G.3
  • 25
    • 0026345105 scopus 로고    scopus 로고
    • Pyrrolidino-4-iodotamoxifen and 4-iodotamoxifen: New analogues of the antioestrogen for the treatment of breast cancer
    • 191
    • Changer S, McCague R, Lugmani Y: Pyrrolidino-4-iodotamoxifen and 4-iodotamoxifen: New analogues of the antioestrogen for the treatment of breast cancer. Cancer Res 191;51: 5851-5858.
    • Cancer Res , vol.51 , pp. 5851-5858
    • Changer, S.1    McCague, R.2    Lugmani, Y.3
  • 26
    • 0031725563 scopus 로고    scopus 로고
    • Idoxifene: A novel selective estrogen receptor modulator prevents bone loss and lowers cholesterol levels in ovariectomized rats and decreases uterine weight in intact rats
    • Nuttall M, Bradbeer J, Stroup G, Nadeau D, Hoffman S, Zhao H, Rehm S, Gowen M: Idoxifene: A novel selective estrogen receptor modulator prevents bone loss and lowers cholesterol levels in ovariectomized rats and decreases uterine weight in intact rats. Endocrinology 1998;139:5224-5233.
    • (1998) Endocrinology , vol.139 , pp. 5224-5233
    • Nuttall, M.1    Bradbeer, J.2    Stroup, G.3    Nadeau, D.4    Hoffman, S.5    Zhao, H.6    Rehm, S.7    Gowen, M.8
  • 27
    • 0030256256 scopus 로고    scopus 로고
    • Identification of rhesus macaques with spontaneous endometriosis
    • Rippy M, Lee D, Pearson S, Bernai C: Identification of rhesus macaques with spontaneous endometriosis. J Med Primatol 1996;25:346-355.
    • (1996) J Med Primatol , vol.25 , pp. 346-355
    • Rippy, M.1    Lee, D.2    Pearson, S.3    Bernai, C.4
  • 28
    • 0003237519 scopus 로고    scopus 로고
    • Video mapping to assess efficacy of an antiestrogen (raloxifen) on spontaneous endometriosis in the rhesus monkey: Macaca mulatta
    • Kuehl T (ed). Temple, Texas A & M University Health Science Center
    • Fanning P, Kuehl T, Lee R, Pearson S: Video mapping to assess efficacy of an antiestrogen (raloxifen) on spontaneous endometriosis in the rhesus monkey: Macaca mulatta; in Kuehl T (ed): Bunkley Day Proceedings. Temple, Texas A & M University Health Science Center, 1996, vol 6, pp 51-61.
    • (1996) Bunkley Day Proceedings , vol.6 , pp. 51-61
    • Fanning, P.1    Kuehl, T.2    Lee, R.3    Pearson, S.4
  • 29
    • 0013666830 scopus 로고    scopus 로고
    • Raloxifen causes rapid regressions of abdominal wall leiomyomas in the estrogen induced pig model
    • Porter K, Tsibris J, Porter G: Raloxifen causes rapid regressions of abdominal wall leiomyomas in the estrogen induced pig model (abstract). J Soc Gynecol Invest 1996;3(suppl): 147.
    • (1996) J Soc Gynecol Invest , vol.3 , Issue.SUPPL. , pp. 147
    • Porter, K.1    Tsibris, J.2    Porter, G.3
  • 30
    • 0029952875 scopus 로고    scopus 로고
    • Inhibition of estrogen-stimulated growth of uterine leiomyomas by selective estrogen receptor modulators
    • Fuchs-Young R, Howe S: Inhibition of estrogen-stimulated growth of uterine leiomyomas by selective estrogen receptor modulators. Mol Carcinog 1996;17:151-159.
    • (1996) Mol Carcinog , vol.17 , pp. 151-159
    • Fuchs-Young, R.1    Howe, S.2
  • 31
    • 0342901073 scopus 로고
    • A scale for assessing postmenopausal endometrial proliferation in response to potential or known selective estrogen receptor modulators
    • Giant M, Eisenhut C, Boss S, Draper M: A scale for assessing postmenopausal endometrial proliferation in response to potential or known selective estrogen receptor modulators. Am J Clin Pathol 1995;104:341-342.
    • (1995) Am J Clin Pathol , vol.104 , pp. 341-342
    • Giant, M.1    Eisenhut, C.2    Boss, S.3    Draper, M.4
  • 32
    • 0032247544 scopus 로고    scopus 로고
    • Epidemiologische hinweise auf die bedeutung von hormonen in der karzinogenese
    • Obermaier A, Jirecek S, Leodolter S: Epidemiologische Hinweise auf die Bedeutung von Hormonen in der Karzinogenese. Gynäkol Geburtshilfliche Rundsch 1998;38:73-79.
    • (1998) Gynäkol Geburtshilfliche Rundsch , vol.38 , pp. 73-79
    • Obermaier, A.1    Jirecek, S.2    Leodolter, S.3
  • 33
    • 0017078344 scopus 로고
    • Effect of tamoxifen (ICI 46,474) on initiation and growth of DMBA-induced rat mammary carcinomata
    • Jordan V: Effect of tamoxifen (ICI 46,474) on initiation and growth of DMBA-induced rat mammary carcinomata. Eur J Cancer 1976;12: 419-425.
    • (1976) Eur J Cancer , vol.12 , pp. 419-425
    • Jordan, V.1
  • 34
    • 0347450835 scopus 로고
    • Tamoxifen and contralateral breast cancer
    • Cuzick J, Baum M: Tamoxifen and contralateral breast cancer. Lancet 1985;ii:282.
    • (1985) Lancet , vol.2 , pp. 282
    • Cuzick, J.1    Baum, M.2
  • 36
    • 0028068906 scopus 로고
    • Droloxifene, a new antiestrogen: Its role in metastatic breast cancer
    • Rausching W, Pritchard KI: Droloxifene, a new antiestrogen: Its role in metastatic breast cancer. Breast Cancer Res Treat 1994;31:83-94.
    • (1994) Breast Cancer Res Treat , vol.31 , pp. 83-94
    • Rausching, W.1    Pritchard, K.I.2
  • 37
    • 0028035492 scopus 로고
    • Genotoxicity of tamoxifen, tamoxifen epoxide and toremifene in human lymphoblastoid cells containing human cytochrome P-450
    • Styles G, Davis E, Lim C: Genotoxicity of tamoxifen, tamoxifen epoxide and toremifene in human lymphoblastoid cells containing human cytochrome P-450. Carcinogenesis 1994; 15:5-9.
    • (1994) Carcinogenesis , vol.15 , pp. 5-9
    • Styles, G.1    Davis, E.2    Lim, C.3
  • 38
    • 0029084658 scopus 로고
    • Randomized comparison of tamoxifen and two separate doses of toremifene in postmenopausal patients with metastatic breast cancer
    • Hayes DF, Van Zyl JA, Hacking A: Randomized comparison of tamoxifen and two separate doses of toremifene in postmenopausal patients with metastatic breast cancer. J Clin Oncol 1995;113:2556-2566.
    • (1995) J Clin Oncol , vol.113 , pp. 2556-2566
    • Hayes, D.F.1    Van Zyl, J.A.2    Hacking, A.3
  • 39
    • 0028935148 scopus 로고
    • Idoxifene: Report of a phase I study in patients with metastatic breast cancer
    • Coombes RC, Haynes BP, Dowsett M: Idoxifene: Report of a phase I study in patients with metastatic breast cancer. Cancer Res 1995;55: 1070-1074.
    • (1995) Cancer Res , vol.55 , pp. 1070-1074
    • Coombes, R.C.1    Haynes, B.P.2    Dowsett, M.3
  • 41
    • 0032537396 scopus 로고    scopus 로고
    • Tamoxifen for early breast cancer: An overview of the randomised trials
    • Early Breast Cancer Trial's Collaborative Group: Tamoxifen for early breast cancer: An overview of the randomised trials. Lancet 1998;351:1451-1467.
    • (1998) Lancet , vol.351 , pp. 1451-1467


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.