Effect of estrogen agonists and antagonists on induction of progesterone receptor in a rat hypothalamic cell line

Endocrinology

Volumn 140, Issue 9, 1999, Pages 3928-3937

  Fitzpatrick, Susan L ^a   Berrodin, Thomas J ^a   Jenkins, Susan F ^a   Sindoni, Deborah M ^a   Deecher, Darlene C ^a   Frail, Donald E ^a  

^a WYETH AYERST RESEARCH   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIESTROGEN; ENCLOMIFENE; ESTRADIOL; ESTROGEN; ESTROGEN RECEPTOR; ETHINYLESTRADIOL; FULVESTRANT; GENISTEIN; MESSENGER RNA; PROGESTERONE RECEPTOR; PROMEGESTONE; RALOXIFENE; TAMOXIFEN; ZUCLOMIFENE;

ANIMAL CELL; ARTICLE; BINDING SITE; CELL TYPE; CONTROLLED STUDY; DNA RESPONSIVE ELEMENT; EMBRYO CELL; ESTROGEN ACTIVITY; GENETIC TRANSFECTION; HORMONAL REGULATION; HORMONE RECEPTOR INTERACTION; HYPOTHALAMUS; MOLECULAR CLONING; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR UPREGULATION; REPORTER GENE; REPRODUCTION; WESTERN BLOTTING;

EID: 0033305436     PISSN: 00137227     EISSN: None     Source Type: Journal    
DOI: 10.1210/endo.140.9.7006     Document Type: Article

References (63)

1. The gonadotropin-releasing hormone (GnRH), neuronal systems: Immunocytochemistry and in situ hybridization
2. Cellular and molecular mechanisms of female reproductive behaviors
3. Hot flashes: Epidemiology and physiology
4. Postmenopausal hot flushes and their management
5. Expression and estrogen regulation of progesterone receptor mRNA in neurons of the mediobasal hypothalamus: An in situ hybridization study
6. Estradiol-induced progestin receptor immunoreactivity is found only in estrogen receptor-immunoreactive cells in guinea pig brain
7. Ovarian steroid regulation of estrogen and progesterone receptor messenger ribonucleic acid in the anteroventral periventricular nucleus of the rat
8. Estradiol induces oxytocin binding sites in rat hypothalamic ventromedial nucleus
9. Expression and region-specific regulation of the oxytocin receptor gene in rat brain
10. c-fos induction by estrogen in specific rat brain areas
11. Progesterone enhances an estradiol-induced increase in Fos immunoreactivity in localized regions of female rat forebrain
12. Estrogen increases proenkephalin messenger ribonucleic acid levels in the ventromedial hypothalamus of the rat
13. Endogenous opioid-immunoreactive neurons of the ventromedial hypothalamic nucleus concentrate estrogen in male and female rats
14. Localized actions of progesterone in hypothalamus involve oxytocin
15. The human oxytocin gene promoter is regulated by estrogens
16. Regulation of neural oxytocin gene expression by gonadal steroids in pubertal rats
17. Hormonal and neurotransmitter regulation of GnRH gene expression and related reproductive behaviors
18. Regulation of gonadotropin-releasing hormone gene expression in vivo and in vitro
19. Multimodal influence of estrogen upon gonadotropin-releasing hormone neurons
20. Cloning of a novel estrogen receptor expressed in rat prostate and ovary
21. ERβ: Identification and characterization of a novel human estrogen receptor
22. Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptor α and β
23. Comparative distribution of estrogen receptor-α and -β mRNA in the rat central nervous system
24. Cloning, chromosomal localization, and functional analysis of the murine estrogen receptor β
25. Mouse estrogen receptor β forms estrogen response element-binding heterodimers with estrogen receptor α
26. Human estrogen receptor β binds DNA in a manner similar to and dimerizes with estrogen receptor α
27. Evidence for the colocalization of estrogen receptor-β mRNA and estrogen receptor-α immunoreactivity in neurons of the rat forebrain
28. Regulation of progesterone receptor messenger ribonucleic acid in the rat medial preoptic nucleus by estrogenic and antiestrogenic compounds: An in situ hybridization study
29. Characterization of the hormone responsive element involved in the regulation of the progesterone receptor gene
30. Identification of multiple, widely spaced estrogen-responsive regions in the rat progesterone receptor gene
31. Responses in the brain of estrogen receptor alpha-disrupted mice
32. Basic guide to the mechanisms of antiestrogen action
33. Analysis of estrogen receptor function in vitro reveals three distinct classes of antiestrogens
34. Estrogen receptor ligands modulate its interaction with DNA
35. Human estrogen receptor transactivational capacity is determined by both cellular and promoter context and mediated by two functionally distinct intramolecular regions
36. Stability of the ligand-estrogen receptor interaction depends on estrogen response element flanking sequences and cellular factors
37. Co-activators and co-repressors in the integration of transcriptional responses
38. Immortalization of hypothalamic GnRH neurons by genetically targeted tumorigenesis
39. Steroid binding and metabolism in the luteinizing hormone-releasing hormone producing neuronal cell line GT1-1
40. Expression of functional estrogen receptors and galanin messenger ribonucleic acid in immortalized luteinizing hormone-releasing hormone neurons: Estrogenic control of galanin gene expression
41. The effects of estradiol on the growth patterns of estrogen receptor-positive hypothalamic cell lines
42. Cloning of estrogen-regulated messenger ribonucleic acids from rat uterus
43. Regulation of the human glucocorticoid receptor by long-term and chronic treatment with glucocorticoid
44. Accurate transcription initiation by RNA polymerase II in a soluble extract from isolated mammalian nuclei
45. Complete amino acid sequence of the human progesterone receptor deduced from cloned cDNA
46. Human progesterone receptors: Synthesis, structure, and phosphorylation
47. Estrogen and progesterone receptors in human uterus and oviduct
48. Induction of progestin receptors by estradiol in the forebrain of estrogen receptor-α gene-disrupted mice
49. Effects of brain antiestrogen implants on maternal behavior and on postpartum estrus in pregnant rats
50. Regulation of estrogen-stimulated lordosis behavior and hypothalamic progestin receptor induction by antiestrogens in female rats
51. Antiestrogens: Effects of tamoxifen, nafoxidine, and CI-628 on sexual behavior, cytoplasmic receptors, and nuclear binding of estrogen
52. Antagonism of central estrogen action by intracerebral implants of tamoxifen
53. An assessment of agonist/antagonist effects of tamoxifen in the female mouse brain
54. Antagonism of sexual behavior in female rats by ventromedial hypothalamic implants of antiestrogen
55. Suppression of spontaneous LH surges in estrogen-treated ovariectomized rats by microimplants of antiestrogens into the preoptic brain
56. Symptoms associated with tamoxifen treatment in postmenopausal women
57. A controlled trial of raloxifene (LY139481) HCl: Impact on bone turnover and serum lipid profile in healthy postmenopausal women
58. Pharmacokinetics, pharmacological and antitumour effects of the specific anti-oestrogen ICI 182780 in women with advanced breast cancer
59. ICI 182,780: A pure antiestrogen that affects behaviors and energy balance in rats without acting in the brain
60. Genistein, a specific inhibitor of tyrosine-specific protein kinases
61. Evidence for an erbstatin-sensitive tyrosine kinase functioning in ascidian egg activation
62. Dietary phytoestrogens
63. Clinical review 92: Phytoestrogens