Mechanistic studies to evaluate the enhanced antiproliferation of human keratinocytes by 1α,25-dihydroxyvitamin D3-3-bromoacetate, a Covalent modifier of vitamin D receptor, compared to 1α,25-dihydroxyvitamin D3

Archives of Biochemistry and Biophysics

Volumn 370, Issue 1, 1999, Pages 34-44

  Chen, Ming L ^a   Ray, Swapna ^a   Swamy, Narasimha ^a   Holick, Michael F ^a   Ray, Rahul ^a  

^a BOSTON UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

1 ,25 dihydroxyvitamin D3 3 bromoacetate; Affinity labeling analog of 1 ,25 dihydroxyvitamin D3; Affinity labeling, kinetic and stoichiometric studies; Antiproliferation of human keratinocytes; Transcriptional mechanism of antiproliferation

Indexed keywords

CALCITRIOL; CALCITRIOL DERIVATIVE; OSTEOCALCIN; OXYGENASE; VITAMIN D RECEPTOR;

AFFINITY LABELING; ANIMAL CELL; ARTICLE; CELL PROLIFERATION; CONFORMATIONAL TRANSITION; DRUG ACTIVITY; DRUG MECHANISM; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG TARGETING; ENZYME INDUCTION; GENE CONTROL; GENETIC TRANSCRIPTION; HUMAN; HUMAN CELL; KERATINOCYTE; NONHUMAN; PRIORITY JOURNAL; PROTEIN CONFORMATION;

ANIMALIA;

EID: 0033215382     PISSN: 00039861     EISSN: None     Source Type: Journal    
DOI: 10.1006/abbi.1999.1353     Document Type: Article

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