Diltiazem causes open channel block of recombinant 5-HT3 receptors

Journal of Physiology

Volumn 519, Issue 3, 1999, Pages 713-722

  Gunthorpe, Martin J ^a,c   Lummis, Sarah C R ^a,b  

^a MRC LABORATORY OF MOLECULAR BIOLOGY   (United Kingdom)

^b Department of Biochemistry ^*  (United Kingdom)

^c GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

5 HYDROXYINDOLE; CALCIUM CHANNEL BLOCKING AGENT; DILTIAZEM; RECOMBINANT RECEPTOR; SEROTONIN 3 ANTAGONIST; SEROTONIN 3 RECEPTOR;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DESENSITIZATION; DRUG MECHANISM; DRUG RECEPTOR BINDING; EMBRYO CELL; KIDNEY CELL; NONHUMAN; PRIORITY JOURNAL; VOLTAGE CLAMP;

CELL LINE; DILTIAZEM; HUMANS; INDOLES; ION CHANNEL GATING; KINETICS; PERFUSION; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT3; RECOMBINANT PROTEINS;

EID: 0033199048     PISSN: 00223751     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1469-7793.1999.0713n.x     Document Type: Article

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