Dicarba-closo-dodecaboranes as a pharmacophore. Novel potent retinoidal agonist

Chemical and Pharmaceutical Bulletin

Volumn 47, Issue 4, 1999, Pages 585-587

  Endo, Yasuyuki ^a   Iijma, Toru ^a   Kagechika, Hiroyuki ^a   Ohta, Kiminori ^a   Kawachi, Emiko ^a   Shudo, Koichi ^a  

^a UNIVERSITY OF TOKYO   (Japan)

Author keywords

Carborane; Dicarba closo dodecaborane; Differentiation; Hydrophobic moiety; Retinoid

Indexed keywords

4 [3 (1,2 DICARBA CLOSO DODECABORAN 1 YL)PHENYLAMINO]BENZOIC ACID; 4 [4 (1,2 DICARBA CLOSO DODECABORAN 1 YL)PHENYLAMINO]BENZOIC ACID; CARBORANE DERIVATIVE; DA 013; HX 630; RETINOIC ACID RECEPTOR; RETINOID DERIVATIVE; RETINOID X RECEPTOR; TAMIBAROTENE; UNCLASSIFIED DRUG;

ARTICLE; CELL DIFFERENTIATION; CELL STRAIN HL 60; CONTROLLED STUDY; DRUG ACTIVITY; DRUG POTENCY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; HYDROPHOBICITY; PHARMACOPHORE; PROMYELOCYTIC LEUKEMIA;

EID: 0032894447     PISSN: 00092363     EISSN: None     Source Type: Journal    
DOI: 10.1248/cpb.47.585     Document Type: Article

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