-
1
-
-
0014421640
-
Structure of porcine cholecystokinin-pancreozymin
-
Mutt, V., Jorpes, J. Structure of porcine cholecystokinin-pancreozymin. Eur J Biochem 1968, 6: 156-62.
-
(1968)
Eur J Biochem
, vol.6
, pp. 156-162
-
-
Mutt, V.1
Jorpes, J.2
-
2
-
-
0017088941
-
Immunochemical evidence of cholecystokinin-like peptides in brain
-
Dockray, G.J.R. Immunochemical evidence of cholecystokinin-like peptides in brain. Nature 1976, 264: 568-70.
-
(1976)
Nature
, vol.264
, pp. 568-570
-
-
Dockray, G.J.R.1
-
3
-
-
0021039777
-
Cholecystokinin octapeptide (CCK 26-33), nonsulfated octapeptide and tetrapeptide (CCK 30-33) in rat brain: Analysis by high pressure liquid chromatography (HPLC) and radioimmunoassay (RIA)
-
Frey, P. Cholecystokinin octapeptide (CCK 26-33), nonsulfated octapeptide and tetrapeptide (CCK 30-33) in rat brain: analysis by high pressure liquid chromatography (HPLC) and radioimmunoassay (RIA). Neurochem Int 1983, 5: 811-5.
-
(1983)
Neurochem Int
, vol.5
, pp. 811-815
-
-
Frey, P.1
-
4
-
-
0024155485
-
Cholecystokinin-58 is the major molecular form in man, dog and cat but not in pig, beef and rat intestine
-
Eberlein, G.A., Eysselein, V.E., Goebell, H. Cholecystokinin-58 is the major molecular form in man, dog and cat but not in pig, beef and rat intestine. Peptides 1988, 9: 993-8.
-
(1988)
Peptides
, vol.9
, pp. 993-998
-
-
Eberlein, G.A.1
Eysselein, V.E.2
Goebell, H.3
-
5
-
-
0002946295
-
Molecular forms and regional distribution of cholecystokinin in the central nervous system
-
Bradwein, J., Vasar, E. (Eds.). RG Landes Companies
-
Rehfeld, J.H., Nielsen, F.C. Molecular forms and regional distribution of cholecystokinin in the central nervous system. In: Cholecystokinin and Anxiety. Bradwein, J., Vasar, E. (Eds.). RG Landes Companies 1995, 33-56.
-
(1995)
Cholecystokinin and Anxiety
, pp. 33-56
-
-
Rehfeld, J.H.1
Nielsen, F.C.2
-
6
-
-
0018101373
-
Isolation, structure and biological activity of two cholecystokinin octapeptides from sheep brain
-
Dockray, G.J., Gregory, R.A., Hutchinson, J.B. et al. Isolation, structure and biological activity of two cholecystokinin octapeptides from sheep brain. Nature 1978: 359-61.
-
(1978)
Nature
, pp. 359-361
-
-
Dockray, G.J.1
Gregory, R.A.2
Hutchinson, J.B.3
-
7
-
-
0017694572
-
Immunohistochemical localization in rabbit brain of a peptide resembling the COOH-terminal octapeptide of cholecystokinin
-
Muller, J.E., Straus, E., Yalow, R.S. Immunohistochemical localization in rabbit brain of a peptide resembling the COOH-terminal octapeptide of cholecystokinin. Proc Natl Acad Sci USA 1977, 74: 3035-7.
-
(1977)
Proc Natl Acad Sci USA
, vol.74
, pp. 3035-3037
-
-
Muller, J.E.1
Straus, E.2
Yalow, R.S.3
-
8
-
-
0002912489
-
Gastrin
-
Walsh, J.H., Dockray, G.J. (Eds.). Raven Press: New York
-
Walsh, J.H. Gastrin. In: Gut Peptides. Walsh, J.H., Dockray, G.J. (Eds.). Raven Press: New York 1994, 75-121.
-
(1994)
Gut Peptides
, pp. 75-121
-
-
Walsh, J.H.1
-
9
-
-
0028351918
-
The tumor biology of gastrin and cholecystokinin
-
Rehfeld, J.F., Van Solinge, W. W. The tumor biology of gastrin and cholecystokinin. Adv Cancer Res 1994, 63: 295-347.
-
(1994)
Adv Cancer Res
, vol.63
, pp. 295-347
-
-
Rehfeld, J.F.1
Van Solinge, W.W.2
-
10
-
-
0344762858
-
TIPS receptors nomenclature supplement
-
Watson, S., Abbott, A. TIPS receptors nomenclature supplement. Trends Pharmacol Sci 1992, Suppl 11.
-
(1992)
Trends Pharmacol Sci
, Issue.11 SUPPL.
-
-
Watson, S.1
Abbott, A.2
-
11
-
-
0026535933
-
Expression cloning and characterization of the canine parietal cell gastrin receptor
-
Kopin, A.S., Lee, Y.M., McBride, L.J. et al. Expression cloning and characterization of the canine parietal cell gastrin receptor. Proc Natl Acad Sci USA 1992, 89, 3605-9.
-
(1992)
Proc Natl Acad Sci USA
, vol.89
, pp. 3605-3609
-
-
Kopin, A.S.1
Lee, Y.M.2
McBride, L.J.3
-
12
-
-
0026672627
-
Brain and gastrointestinal cholecystokinin receptor family: Structure and functional expression
-
Wank, S.A., Pisegna, J.R., Weerth, A.D. Brain and gastrointestinal cholecystokinin receptor family: structure and functional expression. Proc Natl Acad Sci USA 1992, 89: 8691-5.
-
(1992)
Proc Natl Acad Sci USA
, vol.89
, pp. 8691-8695
-
-
Wank, S.A.1
Pisegna, J.R.2
Weerth, A.D.3
-
13
-
-
0000745560
-
Distinct cholecystokinin receptors in brain and pancreas
-
Innis, R.B., Snyder, S.H. Distinct cholecystokinin receptors in brain and pancreas. Proc Natl Acad Sci USA 1980, 77: 6917-28.
-
(1980)
Proc Natl Acad Sci USA
, vol.77
, pp. 6917-6928
-
-
Innis, R.B.1
Snyder, S.H.2
-
14
-
-
0021039340
-
Cholecystokinin in the central nervous system: A minireview
-
Beinfeld, M.C. Cholecystokinin in the central nervous system: a minireview. Neuropeptides 1983, 3: 411-427.
-
(1983)
Neuropeptides
, vol.3
, pp. 411-427
-
-
Beinfeld, M.C.1
-
16
-
-
0025411361
-
Autoradiographical detection of cholecystokinin-A receptors in primate brain using 1251-bolton hunter CCK-8 and 3H-MK-329
-
Hill, D.R., Shaw, T.M., Graham, W., Woodruff, G.N. Autoradiographical detection of cholecystokinin-A receptors in primate brain using 1251-Bolton Hunter CCK-8 and 3H-MK-329. J Neurosci 1990, 10: 1070-81.
-
(1990)
J Neurosci
, vol.10
, pp. 1070-1081
-
-
Hill, D.R.1
Shaw, T.M.2
Graham, W.3
Woodruff, G.N.4
-
17
-
-
0023947651
-
CCK-A receptors in the rat interpeduncular nucleus: Evidence for a presynaptic location
-
Hill, D.R., Shaw, T.M., Dourish, C.T., Woodruff, G.N. CCK-A receptors in the rat interpeduncular nucleus: evidence for a presynaptic location. Brain Res 1990, 454: 101-5.
-
(1990)
Brain Res
, vol.454
, pp. 101-105
-
-
Hill, D.R.1
Shaw, T.M.2
Dourish, C.T.3
Woodruff, G.N.4
-
18
-
-
0022657202
-
Two brain cholecystokinin receptors: Implications for behavioral actions
-
Moran, T.H., Robinson, P.H., Goldrich, M.S., McHugh, P.R. Two brain cholecystokinin receptors: implications for behavioral actions. Brain Res 1986, 362: 175-9.
-
(1986)
Brain Res
, vol.362
, pp. 175-179
-
-
Moran, T.H.1
Robinson, P.H.2
Goldrich, M.S.3
McHugh, P.R.4
-
19
-
-
0025019446
-
Hormones in colon cancer: Past and prospective studies
-
Singh, P., Townsend, C. M., Thompson, J.C., Naraayan, S., Guo, Y.S. Hormones in colon cancer: past and prospective studies. Cancer J 1990, 3: 28-33.
-
(1990)
Cancer J
, vol.3
, pp. 28-33
-
-
Singh, P.1
Townsend, C.M.2
Thompson, J.C.3
Naraayan, S.4
Guo, Y.S.5
-
21
-
-
0027379255
-
The human gastrin/cholecystokinin type B receptor gene: Alternative splice donor site in exon 4 generates two variant mRNAs
-
Song, I., Brown, R.B., Wiltshire, R.N., Gantz, I., Trent, J.M., Yamada, T. The human gastrin/cholecystokinin type B receptor gene: alternative splice donor site in exon 4 generates two variant mRNAs. Proc Natl Acad Sci USA 1993, 90: 9085-9.
-
(1993)
Proc Natl Acad Sci USA
, vol.90
, pp. 9085-9089
-
-
Song, I.1
Brown, R.B.2
Wiltshire, R.N.3
Gantz, I.4
Trent, J.M.5
Yamada, T.6
-
22
-
-
0014218864
-
Antisecretory action of some new compounds free of anti-cholinergic actions
-
Rovati, A.L., Casula, P.L., Dare, G. Antisecretory action of some new compounds free of anti-cholinergic actions. Minerva Med 1967, 58: 3651-3.
-
(1967)
Minerva Med
, vol.58
, pp. 3651-3653
-
-
Rovati, A.L.1
Casula, P.L.2
Dare, G.3
-
23
-
-
0028950584
-
Therapeutic potential of cholecystokinin-B antagonists
-
Rassmussen, K. Therapeutic potential of cholecystokinin-B antagonists. Exp Opin Invest Drugs 1995, 4: 313-22.
-
(1995)
Exp Opin Invest Drugs
, vol.4
, pp. 313-322
-
-
Rassmussen, K.1
-
24
-
-
0031667266
-
Update on nonpeptide CCK-B receptor antagonists
-
Revel, L., Makovec, F. Update on nonpeptide CCK-B receptor antagonists. Drugs Fut 1998, 23: 751-66.
-
(1998)
Drugs Fut
, vol.23
, pp. 751-766
-
-
Revel, L.1
Makovec, F.2
-
25
-
-
0028860738
-
Gastrin antagonists and gastrointestinal tumors
-
Watson, S.A. Gastrin antagonists and gastrointestinal tumors. Exp Opin Invest Drugs 1995, 4: 1253-66.
-
(1995)
Exp Opin Invest Drugs
, vol.4
, pp. 1253-1266
-
-
Watson, S.A.1
-
27
-
-
0022516131
-
A study of the cerebral cortex cholecystokinin receptor using two radiolabelled probes: Evidence for a common CCK 8 and CCK 4 cholecystokinin binding site
-
Clark, C.R., Daum, P., Hughes, J. A study of the cerebral cortex cholecystokinin receptor using two radiolabelled probes: evidence for a common CCK 8 and CCK 4 cholecystokinin binding site. J Neurochem 1986, 46: 1094-101.
-
(1986)
J Neurochem
, vol.46
, pp. 1094-1101
-
-
Clark, C.R.1
Daum, P.2
Hughes, J.3
-
30
-
-
0024475075
-
3H]L-365260: A new potent and selective brain cholecystokinin (CCK-B) and gastrin receptor antagonist radioligand
-
3H]L-365260: a new potent and selective brain cholecystokinin (CCK-B) and gastrin receptor antagonist radioligand. Mol Pharmacol 1989, 35: 803-8.
-
(1989)
Mol Pharmacol
, vol.35
, pp. 803-808
-
-
Chang, R.S.1
Chen, T.B.2
Bock, M.G.3
-
31
-
-
0027339688
-
3H]-PD-140376: A novel and highly selective antagonist radioligand for the cholecystokininB/gastrin receptor in guinea pig cerebral cortex and gastric mucosa
-
3H]-PD-140376: a novel and highly selective antagonist radioligand for the cholecystokininB/gastrin receptor in guinea pig cerebral cortex and gastric mucosa. Mol Pharmacol 1993, 43: 595-602.
-
(1993)
Mol Pharmacol
, vol.43
, pp. 595-602
-
-
Hunter, J.C.1
Suman-Chauman, N.2
Meecham, K.G.3
-
33
-
-
0027460545
-
The human brain cholecystokinin-B/gastrin receptor
-
Lee, Y.M., Beinborn, M., McBride, E.W., Lu, M., Kolakowski, L.F., Kopin, A.F. The human brain cholecystokinin-B/gastrin receptor. J Biol Chem 1993, 268: 8164-9.
-
(1993)
J Biol Chem
, vol.268
, pp. 8164-8169
-
-
Lee, Y.M.1
Beinborn, M.2
McBride, E.W.3
Lu, M.4
Kolakowski, L.F.5
Kopin, A.F.6
-
34
-
-
0029761351
-
Pharmacological characterization of a Chinese hamster ovary cell line transfected with the human CCK-B receptor gene
-
Dunlop, J., Brammer, N., Ennis, C. Pharmacological characterization of a Chinese hamster ovary cell line transfected with the human CCK-B receptor gene. Neuropeptides 1996, 30: 359-63.
-
(1996)
Neuropeptides
, vol.30
, pp. 359-363
-
-
Dunlop, J.1
Brammer, N.2
Ennis, C.3
-
35
-
-
0018886835
-
Binding of cholecystokinin to high affinity receptors on isolated rat pancreatic acini
-
Sankaran, H., Goldfine, I.D., Deveney, C.W., Wong, K.Y., Williams, J.A. Binding of cholecystokinin to high affinity receptors on isolated rat pancreatic acini. J Biol Chem 1980, 255: 1849-53.
-
(1980)
J Biol Chem
, vol.255
, pp. 1849-1853
-
-
Sankaran, H.1
Goldfine, I.D.2
Deveney, C.W.3
Wong, K.Y.4
Williams, J.A.5
-
38
-
-
0027204042
-
Activation of CCK-B receptors elevates cytosolic Ca2+ levels in a pituitary cell line
-
Kuwahara, T., Nagase, H., Takamiya, M., Yoshizaki, H., Nakano, A., Arisawa, M. Activation of CCK-B receptors elevates cytosolic Ca2+ levels in a pituitary cell line. Peptides 1993, 14: 801-5.
-
(1993)
Peptides
, vol.14
, pp. 801-805
-
-
Kuwahara, T.1
Nagase, H.2
Takamiya, M.3
Yoshizaki, H.4
Nakano, A.5
Arisawa, M.6
-
39
-
-
0028180038
-
Characterization of CCKB receptors on GH3 pituitary cells: Receptor activation is linked to Ca2+ mobilization
-
Smith, A.J., Patel, S., Freedman, S.B. Characterization of CCKB receptors on GH3 pituitary cells: receptor activation is linked to Ca2+ mobilization. Eur J Pharmacol 1994, 267: 215-23.
-
(1994)
Eur J Pharmacol
, vol.267
, pp. 215-223
-
-
Smith, A.J.1
Patel, S.2
Freedman, S.B.3
-
40
-
-
0029796566
-
Antagonistic effect of YM022, an antiulcer agent in rats, on human cholecystokinin (CCK)B/gastrin receptor
-
Koizumi, T., Saita, Y., Miyake, A., Nishida, A., Yazawa, H., Honda, K. Antagonistic effect of YM022, an antiulcer agent in rats, on human cholecystokinin (CCK)B/gastrin receptor. Jpn J Pharmacol 1996, 71: 307-13.
-
(1996)
Jpn J Pharmacol
, vol.71
, pp. 307-313
-
-
Koizumi, T.1
Saita, Y.2
Miyake, A.3
Nishida, A.4
Yazawa, H.5
Honda, K.6
-
41
-
-
0023885148
-
Excitatory effects of cholecystokinin in rat hippocampus: Pharmacological response compatible with central or B-type CCK receptors
-
Bohme, G.A., Stutzman, J.M., Blanchard, J.C. Excitatory effects of cholecystokinin in rat hippocampus: pharmacological response compatible with central or B-type CCK receptors. Brain Res 1988, 451: 309-18.
-
(1988)
Brain Res
, vol.451
, pp. 309-318
-
-
Bohme, G.A.1
Stutzman, J.M.2
Blanchard, J.C.3
-
42
-
-
0025160491
-
Investigation of behavioral and electrophysiological responses induced by selective stimulation of CCKB receptors by using a new highly potent CCK analog, BC 264
-
Daugè, G.A., Bohme, J.N. Crawley, C. et al. Investigation of behavioral and electrophysiological responses induced by selective stimulation of CCKB receptors by using a new highly potent CCK analog, BC 264. Synapse 1990, 6: 73-80.
-
(1990)
Synapse
, vol.6
, pp. 73-80
-
-
Daugè, G.A.1
Bohme, J.N.2
Crawley, C.3
-
43
-
-
70449173508
-
Continuous recording of acid gastric secretion in the rat
-
Gosh, M.N., Shild, H.O. Continuous recording of acid gastric secretion in the rat. Br J Pharmacol Chemother 1958, 13: 54-61.
-
(1958)
Br J Pharmacol Chemother
, vol.13
, pp. 54-61
-
-
Gosh, M.N.1
Shild, H.O.2
-
44
-
-
0001274018
-
Studies on gastrin
-
Lai, K.S. Studies on gastrin. Gut 1964, 5: 327-32.
-
(1964)
Gut
, vol.5
, pp. 327-332
-
-
Lai, K.S.1
-
45
-
-
0027521751
-
The gastrin/cholecystokinin-B receptor antagonist L-365,260 reduces basal acid secretion and prevents gastrointestinal damage induced by aspirin, ethanol and cysteamine in the rat
-
Pendley, C.E., Fitzpatrick, L.R., Ewing, R.W., Molino, B.F., Martin, G.E. The gastrin/cholecystokinin-B receptor antagonist L-365,260 reduces basal acid secretion and prevents gastrointestinal damage induced by aspirin, ethanol and cysteamine in the rat. J Pharmacol Exp Ther 1993, 1348-54.
-
(1993)
J Pharmacol Exp Ther
, pp. 1348-1354
-
-
Pendley, C.E.1
Fitzpatrick, L.R.2
Ewing, R.W.3
Molino, B.F.4
Martin, G.E.5
-
46
-
-
0026525948
-
L-365260, a potent gastrin/CCK-B receptor antagonist, suppress gastric acid secretion induced by histamine and betanechol as well as pentagastrin in rat
-
Nishida, A., Yuki, H., Tsutsumi, R. et al. L-365260, a potent gastrin/CCK-B receptor antagonist, suppress gastric acid secretion induced by histamine and betanechol as well as pentagastrin in rat. Jpn J Pharmacol 1992, 58: 137-45.
-
(1992)
Jpn J Pharmacol
, vol.58
, pp. 137-145
-
-
Nishida, A.1
Yuki, H.2
Tsutsumi, R.3
-
47
-
-
0014441168
-
Response of rats with chronic gastric fistulas to subcutaneous injection of histamine, ICI-50123 and insulin
-
Lee, Y.H, Thompson, J.H. Response of rats with chronic gastric fistulas to subcutaneous injection of histamine, ICI-50123 and insulin. Am J Dig Dis 1969, 14: 14-29.
-
(1969)
Am J Dig Dis
, vol.14
, pp. 14-29
-
-
Lee, Y.H.1
Thompson, J.H.2
-
48
-
-
0024337187
-
Gastrin is a major mediator of the gastric phase of acid secretion in dogs: Proof by monoclonal antibody neutralization
-
Kovac, T.O.G., Walsh, J.H., Maxwell, V. et al. Gastrin is a major mediator of the gastric phase of acid secretion in dogs: proof by monoclonal antibody neutralization. Gastroenterology 1989, 97: 1406-13.
-
(1989)
Gastroenterology
, vol.97
, pp. 1406-1413
-
-
Kovac, T.O.G.1
Walsh, J.H.2
Maxwell, V.3
-
49
-
-
0005614316
-
Uber die absonderung der fundusdrusen des magens
-
Heidenhain, R. Uber die absonderung der fundusdrusen des magens. Pfluegers Arch 1879, 19: 148-66.
-
(1879)
Pfluegers Arch
, vol.19
, pp. 148-166
-
-
Heidenhain, R.1
-
50
-
-
0000100769
-
Gastric mucosal injury by fatty and acetylsalicylic acids
-
Davenport, H.D. Gastric mucosal injury by fatty and acetylsalicylic acids. Gastroenterology 1964, 46: 245-53.
-
(1964)
Gastroenterology
, vol.46
, pp. 245-253
-
-
Davenport, H.D.1
-
51
-
-
0016257119
-
Inhibition of indomethacin-induced gastric ulceration in the rat by perorally administered synthetic and natural prostaglandin analogues
-
Lippman, W. Inhibition of indomethacin-induced gastric ulceration in the rat by perorally administered synthetic and natural prostaglandin analogues. Prostaglandins 1974, 7: 1-9.
-
(1974)
Prostaglandins
, vol.7
, pp. 1-9
-
-
Lippman, W.1
-
52
-
-
0017699599
-
Duodenal ulcerogens cysteamine, and propionitrile, stimulate serum gastrin levels in the rat
-
Lichetnberger, L.M., Szabo, S., Trier, J.S. Duodenal ulcerogens cysteamine, and propionitrile, stimulate serum gastrin levels in the rat. Gastroenterology 1977, 73: 1305-8.
-
(1977)
Gastroenterology
, vol.73
, pp. 1305-1308
-
-
Lichetnberger, L.M.1
Szabo, S.2
Trier, J.S.3
-
53
-
-
0020036350
-
Mepirizole-induced duodenal ulcers in rat and their pathogenesis
-
Okabe, S., Ishihara, Y., Inoo, H., Tanaka, H. Mepirizole-induced duodenal ulcers in rat and their pathogenesis. Dig Dis Sci 1982, 27: 242-9.
-
(1982)
Dig Dis Sci
, vol.27
, pp. 242-249
-
-
Okabe, S.1
Ishihara, Y.2
Inoo, H.3
Tanaka, H.4
-
54
-
-
0022586951
-
Hypergastrinemia produces trophic effect in stomach but not in pancreas and intestine
-
Håkanson, R., Blom, H., Carlsson, E., Larsson, B., Ryberg, B., Sundler, F. Hypergastrinemia produces trophic effect in stomach but not in pancreas and intestine. Regul Pept 1986, 13: 225-33.
-
(1986)
Regul Pept
, vol.13
, pp. 225-233
-
-
Håkanson, R.1
Blom, H.2
Carlsson, E.3
Larsson, B.4
Ryberg, B.5
Sundler, F.6
-
55
-
-
0027005524
-
The biology and pathobiology of the ECL cells
-
Håkanson, R., Tielemans, Y., Chen, D. et al. The biology and pathobiology of the ECL cells. Yale J Biol Med 1992, 65: 761-74.
-
(1992)
Yale J Biol Med
, vol.65
, pp. 761-774
-
-
Håkanson, R.1
Tielemans, Y.2
Chen, D.3
-
56
-
-
0025733774
-
Gastrin and cholecystokinin receptors on histamine- and somatostatin-containing cells from rabbit fundic mucosa. Characterization by means of selective antagonists L-364,718 and L-365,260
-
Roche, S., Gusdinar, T., Bali, J.P., Magous, R. Gastrin and cholecystokinin receptors on histamine- and somatostatin-containing cells from rabbit fundic mucosa. Characterization by means of selective antagonists L-364,718 and L-365,260. Biochem Pharmacol 1991, 42: 771-6.
-
(1991)
Biochem Pharmacol
, vol.42
, pp. 771-776
-
-
Roche, S.1
Gusdinar, T.2
Bali, J.P.3
Magous, R.4
-
57
-
-
0025883797
-
Cholecystokinin-B (gastrin) receptor regulates gastrin histamine release and acid secretion
-
Sandvik, A.K., Waldum, H.L. Cholecystokinin-B (gastrin) receptor regulates gastrin histamine release and acid secretion. Am J Physiol 1991, 260: G925-G928.
-
(1991)
Am J Physiol
, vol.260
-
-
Sandvik, A.K.1
Waldum, H.L.2
-
58
-
-
0021812468
-
Toxicological studies on omeprazole
-
Ekman, L., Hansson, E., Havu, N., Carlsson, E., Lundbeg, G. Toxicological studies on omeprazole. Scand J Gastroenterol 1985, 20:, Suppl. 108: 53-69.
-
(1985)
Scand J Gastroenterol
, vol.20
, Issue.108 SUPPL.
, pp. 53-69
-
-
Ekman, L.1
Hansson, E.2
Havu, N.3
Carlsson, E.4
Lundbeg, G.5
-
59
-
-
0022394794
-
Association of long-lasting unsurmountable histamine H2 blockade and gastric carcinoid tumors in the rat
-
Poynter, C., Pick, R.C., Harcourt, R.A. et al. Association of long-lasting unsurmountable histamine H2 blockade and gastric carcinoid tumors in the rat. Gut 1985, 26: 1284-95.
-
(1985)
Gut
, vol.26
, pp. 1284-1295
-
-
Poynter, C.1
Pick, R.C.2
Harcourt, R.A.3
-
60
-
-
0027301098
-
Histamine secretion from rat enterochromaffin-like cells
-
Prinz, C., Kaimura, M., Scott, D.R., Mercier, M., Helander, H.F., Sachs, G. Histamine secretion from rat enterochromaffin-like cells. Gastroenterology 1993, 105: 449-61.
-
(1993)
Gastroenterology
, vol.105
, pp. 449-461
-
-
Prinz, C.1
Kaimura, M.2
Scott, D.R.3
Mercier, M.4
Helander, H.F.5
Sachs, G.6
-
61
-
-
0029957166
-
Evaluation of the specificity and potency of a series of cholecystokinin-B/gastrin receptor antagonists in vivo
-
Ding, X-Q., Håkanson, R. Evaluation of the specificity and potency of a series of cholecystokinin-B/gastrin receptor antagonists in vivo. Pharmacol Toxicol 1996, 79: 124-30.
-
(1996)
Pharmacol Toxicol
, vol.79
, pp. 124-130
-
-
Ding, X.-Q.1
Håkanson, R.2
-
62
-
-
0028807324
-
Gastrin receptor antagonist YM-022 prevents hypersecretion after long-term acid suppression
-
Nishida, A., Kobayashi, A., Azukawa, S. et al. Gastrin receptor antagonist YM-022 prevents hypersecretion after long-term acid suppression. Am J Physiol 1995, 269: G699-G705.
-
(1995)
Am J Physiol
, vol.269
-
-
Nishida, A.1
Kobayashi, A.2
Azukawa, S.3
-
63
-
-
0026671301
-
Effect of gastric receptor blockade on endocrine cells in rats during achlorhydria
-
Eissle, R., Parberg, H., Koop, H. et al. Effect of gastric receptor blockade on endocrine cells in rats during achlorhydria. Gastroenterology 1992, 103: 1596-601.
-
(1992)
Gastroenterology
, vol.103
, pp. 1596-1601
-
-
Eissle, R.1
Parberg, H.2
Koop, H.3
-
64
-
-
0026010280
-
Studies of isolated parietal and enterochromaffin-like cells from the rat
-
Brenna, E., Waldum, H.L. Studies of isolated parietal and enterochromaffin-like cells from the rat. Scan J Gastroenterol 1991, 26: 1295-306.
-
(1991)
Scan J Gastroenterol
, vol.26
, pp. 1295-1306
-
-
Brenna, E.1
Waldum, H.L.2
-
65
-
-
0025936503
-
Inhibitory effects of the gastrin receptor antagonist (L-365,260) on gastrointestinal tumor cell
-
Watson, S., Durrant, L., Elston, P. Morris, D. Inhibitory effects of the gastrin receptor antagonist (L-365,260) on gastrointestinal tumor cell. Cancer 1991, 68: 1255-60.
-
(1991)
Cancer
, vol.68
, pp. 1255-1260
-
-
Watson, S.1
Durrant, L.2
Elston, P.3
Morris, D.4
-
66
-
-
0031903962
-
Gastrin-17 and G17-gly induce proliferation of LoVo cells through the CCK B/gastrin receptor
-
Artru, P., Attoub, S., Levasseur, S., Lewin, M.J., Bado, A. Gastrin-17 and G17-gly induce proliferation of LoVo cells through the CCK B/gastrin receptor. Gastroenterol Clin Biol 1998, 22: 607-12.
-
(1998)
Gastroenterol Clin Biol
, vol.22
, pp. 607-612
-
-
Artru, P.1
Attoub, S.2
Levasseur, S.3
Lewin, M.J.4
Bado, A.5
-
67
-
-
0029958939
-
Gastrin receptor antagonist CI-988 inhibits growth of human colon cancer in vivo and in vitro
-
Romani, R., Howes, L.G., Morris, D.L. Gastrin receptor antagonist CI-988 inhibits growth of human colon cancer in vivo and in vitro. Aust N Z J Surg 1996, 66: 235-7.
-
(1996)
Aust N Z J Surg
, vol.66
, pp. 235-237
-
-
Romani, R.1
Howes, L.G.2
Morris, D.L.3
-
68
-
-
0027181967
-
Differential mode of action of high- and low-affinity CCK/gastrin receptor antagonists in growth inhibition of gastrin-responsive human gastric adenocarcinoma cells in vitro
-
Piontek, M.K., Hengels, K.J. Differential mode of action of high- and low-affinity CCK/gastrin receptor antagonists in growth inhibition of gastrin-responsive human gastric adenocarcinoma cells in vitro. Anticancer Res 1993, 13: 715-20.
-
(1993)
Anticancer Res
, vol.13
, pp. 715-720
-
-
Piontek, M.K.1
Hengels, K.J.2
-
69
-
-
0026684688
-
Therapeutic effect of the gastrin receptor antagonist, CR 2093 on gastrointestinal tumor cell growth
-
Watson, S.A., Crosbee, D.M., Morris, D.L. et al. Therapeutic effect of the gastrin receptor antagonist, CR 2093 on gastrointestinal tumor cell growth. Br J Cancer 1992, 65: 879-83.
-
(1992)
Br J Cancer
, vol.65
, pp. 879-883
-
-
Watson, S.A.1
Crosbee, D.M.2
Morris, D.L.3
-
70
-
-
0031964306
-
Biochemical and pharmacological profiles of loxiglumide, a novel cholecystokinin-A receptor antagonist
-
Fukamizu, Y., Nakaijma, T., Kimura, K. et al. Biochemical and pharmacological profiles of loxiglumide, a novel cholecystokinin-A receptor antagonist. Arzneim-Forsch Drug Res 1998, 48: 58-64.
-
(1998)
Arzneim-Forsch Drug Res
, vol.48
, pp. 58-64
-
-
Fukamizu, Y.1
Nakaijma, T.2
Kimura, K.3
-
71
-
-
0029035591
-
RP 73870, a gastrin/cholecystokinin-B receptor antagonist with potent antiulcer activity in the rat
-
Pendley, C.E., Fitzpatrick, L.R., Capolino, A.L. et al. RP 73870, a gastrin/cholecystokinin-B receptor antagonist with potent antiulcer activity in the rat. J Pharmacol Exp Ther 1995, 273: 1015-22.
-
(1995)
J Pharmacol Exp Ther
, vol.273
, pp. 1015-1022
-
-
Pendley, C.E.1
Fitzpatrick, L.R.2
Capolino, A.L.3
-
72
-
-
0027988272
-
5-Phenyl-3-ureidobenzazepin-2-ones as cholecystokinin-B receptor antagonists
-
Lowe, J.A., Hageman, D.L., Drodza, S.E. et al. 5-Phenyl-3-ureidobenzazepin-2-ones as cholecystokinin-B receptor antagonists. J Med Chem 1994, 37: 3789-811.
-
(1994)
J Med Chem
, vol.37
, pp. 3789-3811
-
-
Lowe, J.A.1
Hageman, D.L.2
Drodza, S.E.3
-
73
-
-
0026515186
-
Structure-antigastrin activity relationships of new (R)-4-benzamido-5-oxopentanoic acid derivatives
-
Makovec, F., Peris, W., Revel, L., Giovanetti, R., Mennuni, L. Rovati, L.C. Structure-antigastrin activity relationships of new (R)-4-benzamido-5-oxopentanoic acid derivatives. J Med Chem 1992, 35: 28-38.
-
(1992)
J Med Chem
, vol.35
, pp. 28-38
-
-
Makovec, F.1
Peris, W.2
Revel, L.3
Giovanetti, R.4
Mennuni, L.5
Rovati, L.C.6
-
74
-
-
0028276292
-
Selectivity and potency of new basic CCK-B antagonists
-
Rovati, L.C., D'Amato, M., Peris, W., Revel, L., Makovec, F. Selectivity and potency of new basic CCK-B antagonists. Ann NY Acad Sci 1994, 713: 395-7.
-
(1994)
Ann Ny Acad Sci
, vol.713
, pp. 395-397
-
-
Rovati, L.C.1
D'Amato, M.2
Peris, W.3
Revel, L.4
Makovec, F.5
-
76
-
-
0031779556
-
CR 2945: A novel CCKB receptor antagonist with anxiolytic-like activity
-
Revel, L., Mennuni, L., Garofalo, P., Makovec, F. CR 2945: a novel CCKB receptor antagonist with anxiolytic-like activity. Behav Pharmacol 1988, 9: 183-194.
-
(1988)
Behav Pharmacol
, vol.9
, pp. 183-194
-
-
Revel, L.1
Mennuni, L.2
Garofalo, P.3
Makovec, F.4
-
77
-
-
0031965829
-
Synthesis of phenoxyacetic acid derivatives as highly potent antagonists of gastrin/cholecystokinin-B receptors
-
Takeda, Y., Kawagoe, K., Yokomizo, A. et al. Synthesis of phenoxyacetic acid derivatives as highly potent antagonists of gastrin/cholecystokinin-B receptors. Chem Pharm Bull 1998, 46: 434-44.
-
(1998)
Chem Pharm Bull
, vol.46
, pp. 434-444
-
-
Takeda, Y.1
Kawagoe, K.2
Yokomizo, A.3
-
78
-
-
0031013735
-
Dual CCK-A and CCK-B receptor antagonists (I). C9-methyl-1,4-benzodiazepines
-
Tabuchi, S. et al. Dual CCK-A and CCK-B receptor antagonists (I). C9-methyl-1,4-benzodiazepines. Bioorg Med Chem Lett 1997, 7: 169-74.
-
(1997)
Bioorg Med Chem Lett
, vol.7
, pp. 169-174
-
-
Tabuchi, S.1
-
79
-
-
0344762842
-
Dual cholecystokinin (CCK)-A and -B receptor antagonist: Synthesis and structure-activity relationships of 9-methyl-5-alkyl-1,4-benzodiazepines
-
Nov 19-21, Tsukuba, Abst 1-P-26
-
nd Conf Drug Discov (Nov 19-21, Tsukuba) 1997, Abst 1-P-26.
-
(1997)
nd Conf Drug Discov
-
-
Satoh, Y.1
-
80
-
-
0345625369
-
Anxiolytic activity of GV 150013, a new potent and selective cholecystokinin-B (CCK-B) antagonist
-
Abst P-10-24
-
Trist, G. et al. Anxiolytic activity of GV 150013, a new potent and selective cholecystokinin-B (CCK-B) antagonist. Eur Neuropsychopharmacol 1996, 6 (Suppl 3): Abst P-10-24.
-
(1996)
Eur Neuropsychopharmacol
, vol.6
, Issue.3 SUPPL.
-
-
Trist, G.1
-
81
-
-
0345193323
-
Synthesis of new 1,5-benzodiazepines as potent and selective CCK-B antagonist
-
Sept 8-12, Maastricht: Abst P-6.57
-
th Symp Med Chem (Sept 8-12, Maastricht) 1996: Abst P-6.57.
-
(1996)
th Symp Med Chem
-
-
Ursini, A.1
-
82
-
-
0029899545
-
Analysis of variation in L-365,260 competition curves in radioligand binding assays
-
Harper, E.A., Roberts, S.P., Shankley, N.P., Black, J.W. Analysis of variation in L-365,260 competition curves in radioligand binding assays. Br J Pharmacol 1996, 118: 1717-26.
-
(1996)
Br J Pharmacol
, vol.118
, pp. 1717-1726
-
-
Harper, E.A.1
Roberts, S.P.2
Shankley, N.P.3
Black, J.W.4
-
83
-
-
0028323564
-
Second-generation benzydiazepine CCK-B antagonists. Development of subnanomolar analogs with selectivity and water solubility
-
Bock, M.G., Di Pardo, R.M., Mellin, E.C. et al. Second-generation benzydiazepine CCK-B antagonists. Development of subnanomolar analogs with selectivity and water solubility. J Med Chem 1994, 37: 722-4.
-
(1994)
J Med Chem
, vol.37
, pp. 722-724
-
-
Bock, M.G.1
Di Pardo, R.M.2
Mellin, E.C.3
-
84
-
-
0028865233
-
Potent, selective, water-soluble benzodiazepine-based CCKB receptor antagonists that contain lipophilic carboxylate surrogates
-
Chambers, M.S. et al. Potent, selective, water-soluble benzodiazepine-based CCKB receptor antagonists that contain lipophilic carboxylate surrogates. Bioorg Med Chem Lett 1995, 5: 2303-8.
-
(1995)
Bioorg Med Chem Lett
, vol.5
, pp. 2303-2308
-
-
Chambers, M.S.1
-
85
-
-
0030043963
-
Controlled modification of acidity in cholecystokinin B receptor antagonists: N-(1,4-Benzodiazepin-3-yl)-N′-[3-(tetrazol-5-ylamino) phenyl]ureas
-
Castro, J.L., Ball, R.G., Broughton, H.B., et al. Controlled modification of acidity in cholecystokinin B receptor antagonists: N-(1,4-Benzodiazepin-3-yl)-N′-[3-(tetrazol-5-ylamino) phenyl]ureas. J Med Chem 1996, 39: 842-849.
-
(1996)
J Med Chem
, vol.39
, pp. 842-849
-
-
Castro, J.L.1
Ball, R.G.2
Broughton, H.B.3
-
86
-
-
0028314649
-
b/gastrin receptor antagonists containing a cationic solubilizing group
-
B/gastrin receptor antagonists containing a cationic solubilizing group. J Med Chem 1994, 37: 719-21.
-
(1994)
J Med Chem
, vol.37
, pp. 719-721
-
-
Showell, G.A.1
Bourrain, S.2
Neduvelil, J.G.3
-
87
-
-
15444358348
-
5-(piperidin-2-yl)- and 5-(homopiperidin-2-yl)-1,4-benzodiazepines: High-affinity, basic ligands for the cholecystokinin-B receptor
-
Castro, J.L., Broughton, H.B., Russel, M.G.N. et al. 5-(piperidin-2-yl)- and 5-(homopiperidin-2-yl)-1,4-benzodiazepines: high-affinity, basic ligands for the cholecystokinin-B receptor. J Med Chem 1997, 40: 2491-501.
-
(1997)
J Med Chem
, vol.40
, pp. 2491-2501
-
-
Castro, J.L.1
Broughton, H.B.2
Russel, M.G.N.3
-
88
-
-
0009750236
-
A novel series of non-peptide CCK and gastrin antagonists: Medicinal chemistry and electrophysiological demonstration of antagonism
-
Dourish C.T., S.J. Cooper (Eds.). Oxford University Press: London
-
Howbert, J.J., Lobb, K.L., Brown, F.R. et al. A novel series of non-peptide CCK and gastrin antagonists: medicinal chemistry and electrophysiological demonstration of antagonism. In: Multiple Cholecystokinin Receptors - Progress Towards CNS Therapeutic Targets. Dourish C.T., S.J. Cooper (Eds.). Oxford University Press: London 1992, 28-37.
-
(1992)
Multiple Cholecystokinin Receptors - Progress Towards CNS Therapeutic Targets
, pp. 28-37
-
-
Howbert, J.J.1
Lobb, K.L.2
Brown, F.R.3
-
91
-
-
0028800435
-
Peptoid CCK receptor antagonists: Pharmacological evaluation of CCKA, CCKB and mixed CCKA/B receptor antagonists
-
Singh, L., Field, M.J., Hill, D.R., et al. Peptoid CCK receptor antagonists: pharmacological evaluation of CCKA, CCKB and mixed CCKA/B receptor antagonists. Eur J Pharmacol 1995, 286: 185-91.
-
(1995)
Eur J Pharmacol
, vol.286
, pp. 185-191
-
-
Singh, L.1
Field, M.J.2
Hill, D.R.3
-
92
-
-
0027489992
-
Cholecystokinin peptidomimetics as selective CCK-B antagonists: Design, synthesis and in vitro and in vivo biochemical properties
-
Blommaert, A.G., Weng, J.H., Dorville, A. et al. Cholecystokinin peptidomimetics as selective CCK-B antagonists: design, synthesis and in vitro and in vivo biochemical properties. J Med Chem 1993, 36: 2868-77.
-
(1993)
J Med Chem
, vol.36
, pp. 2868-2877
-
-
Blommaert, A.G.1
Weng, J.H.2
Dorville, A.3
-
93
-
-
0031048074
-
Structure-based design of new constrained cyclic agonists of the cholecystokinin CCK-B receptor
-
Blommaert, A.G., Dhotel, H., Ducos, B. et al. Structure-based design of new constrained cyclic agonists of the cholecystokinin CCK-B receptor. J Med Chem 1997, 40: 647-658.
-
(1997)
J Med Chem
, vol.40
, pp. 647-658
-
-
Blommaert, A.G.1
Dhotel, H.2
Ducos, B.3
-
94
-
-
0028225773
-
The ureidoacetamides, a novel family of non-peptide CCK-B/gastrin antagonists
-
Bohme, G.A., Bertrand, P., Guyon, C. et al. The ureidoacetamides, a novel family of non-peptide CCK-B/gastrin antagonists. Ann NY Acad Sci 1994, 713: 118-20.
-
(1994)
Ann Ny Acad Sci
, vol.713
, pp. 118-120
-
-
Bohme, G.A.1
Bertrand, P.2
Guyon, C.3
-
95
-
-
0001760209
-
RPR 101367, a new potent and selective non-peptide CCK-B receptor antagonist
-
Abst 241P
-
Bertrand, P. et al. RPR 101367, a new potent and selective non-peptide CCK-B receptor antagonist. Br J Pharmacol 1995, 116(Suppl): Abst 241P.
-
(1995)
Br J Pharmacol
, vol.116
, Issue.SUPPL.
-
-
Bertrand, P.1
-
96
-
-
0030861916
-
Synthesis and pharmacological properties of ureidomethylcarbamoylphenylketone derivatives. A new potent and subtype-selective nonpeptide CCK-B/gastrin receptor antagonists, S-0509
-
Hagishita, S., Murakami, Y., Seno, K. et al. Synthesis and pharmacological properties of ureidomethylcarbamoylphenylketone derivatives. A new potent and subtype-selective nonpeptide CCK-B/gastrin receptor antagonists, S-0509. Bioorg Med Chem 1997, 5: 1695-714.
-
(1997)
Bioorg Med Chem
, vol.5
, pp. 1695-1714
-
-
Hagishita, S.1
Murakami, Y.2
Seno, K.3
-
97
-
-
14444288026
-
(3R)-N-(tert-butylcarbonylmethyl)-2,3-dihydro-2-oxo-5-(2-pyridyl)-1H-1,4- benzodiazepin-3-yl-N′-(3-(methylamino)phenyl)urea (YF476): A potent and orally active gastrin/CCK-B antagonist
-
Semple, G., Ryder, H., Rooker, D.P. et al. (3R)-N-(tert-butylcarbonylmethyl)-2,3-dihydro-2-oxo-5-(2-pyridyl)-1H-1,4- benzodiazepin-3-yl)-N′-(3-(methylamino)phenyl)urea (YF476): a potent and orally active gastrin/CCK-B antagonist. J Med Chem 1997, 40: 331-41.
-
(1997)
J Med Chem
, vol.40
, pp. 331-341
-
-
Semple, G.1
Ryder, H.2
Rooker, D.P.3
-
98
-
-
8044235636
-
YF476 is a new potent and selective gastrin/cholecystokinin-B receptor antagonist in vitro and in vivo
-
Takinami, Y., Yuki, H., Nishida, A. et al. YF476 is a new potent and selective gastrin/cholecystokinin-B receptor antagonist in vitro and in vivo. Aliment Pharmacol Ther 1997, 11: 113-20.
-
(1997)
Aliment Pharmacol Ther
, vol.11
, pp. 113-120
-
-
Takinami, Y.1
Yuki, H.2
Nishida, A.3
-
99
-
-
0344048483
-
Substituted 1,4-benzodiazepin-2-one derivatives as potent selective and orally active gastrin/CCK-B antagonists
-
Aug 20-24: Abst MEDI 166
-
th ACS Natl Meet (Aug 20-24) 1995: Abst MEDI 166.
-
(1995)
th ACS Natl Meet
-
-
Satoh, M.1
-
100
-
-
0030036247
-
Biological activity of analogues of YM022. Novel (3-amino substituted phenyl) urea derivatives of 1,4-benzodiazepin-2-one as gastrin/cholecystokinin-B receptor antagonists
-
Satoh, M., Okamoto, Y., Koshio, H. et al. Biological activity of analogues of YM022. Novel (3-amino substituted phenyl) urea derivatives of 1,4-benzodiazepin-2-one as gastrin/cholecystokinin-B receptor antagonists. Chem Pharm Bull 1996, 44: 1412-4.
-
(1996)
Chem Pharm Bull
, vol.44
, pp. 1412-1414
-
-
Satoh, M.1
Okamoto, Y.2
Koshio, H.3
-
101
-
-
0029558218
-
New 1,4-benzodiazepin-2-one derivatives as gastrin/cholecystokinin-B antagonists
-
Satoh, M., Kondoh, Y., Okamoto, Y. et al. New 1,4-benzodiazepin-2-one derivatives as gastrin/cholecystokinin-B antagonists. Chem Pharm Bull 1995, 43: 2159-67.
-
(1995)
Chem Pharm Bull
, vol.43
, pp. 2159-2167
-
-
Satoh, M.1
Kondoh, Y.2
Okamoto, Y.3
-
102
-
-
0030070863
-
Structure-antigastrin activity relationships of new spiroglumide amido acid derivatives
-
Makovec, F., Peris, W., Frigerio, S. et al. Structure-antigastrin activity relationships of new spiroglumide amido acid derivatives. J Med Chem 1996, 39: 135-42.
-
(1996)
J Med Chem
, vol.39
, pp. 135-142
-
-
Makovec, F.1
Peris, W.2
Frigerio, S.3
-
103
-
-
0028199905
-
Evaluation of a series of novel CCKB antagonists using a functional assay in the rat central nervous system
-
Boden, P.R, Pinnock, R.D., Pritchard, M.C., Woodruff, G.N. Evaluation of a series of novel CCKB antagonists using a functional assay in the rat central nervous system. Br J Pharmacol 1994, 112: 666-70.
-
(1994)
Br J Pharmacol
, vol.112
, pp. 666-670
-
-
Boden, P.R.1
Pinnock, R.D.2
Pritchard, M.C.3
Woodruff, G.N.4
-
104
-
-
0026740897
-
Characterization of antigastrin activity in vivo of CR2194, a new R-4-benzamido-5-oxo-pentanoic acid derivative
-
Revel, L., Ferrari, F., Makovec, F., Rovati, L.C., Impicciatore, M. Characterization of antigastrin activity in vivo of CR2194, a new R-4-benzamido-5-oxo-pentanoic acid derivative. Eur J Pharmacol 1992, 216: 217-24.
-
(1992)
Eur J Pharmacol
, vol.216
, pp. 217-224
-
-
Revel, L.1
Ferrari, F.2
Makovec, F.3
Rovati, L.C.4
Impicciatore, M.5
-
106
-
-
0024520619
-
A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-B) ligand: L-365,260
-
Lotti, V.J., Chang, R.S.L. A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-B) ligand: L-365,260. Eur J Pharmacol 1989, 162: 273-80.
-
(1989)
Eur J Pharmacol
, vol.162
, pp. 273-280
-
-
Lotti, V.J.1
Chang, R.S.L.2
-
107
-
-
0027939411
-
Biological properties of the benzodiazepine amidine derivative L-740,093, a cholecystokinin-B/gastrin receptor antagonist with high affinity in vitro and high potency in vivo
-
Patel, S., Smith, A.J., Chapman, K.L. et al. Biological properties of the benzodiazepine amidine derivative L-740,093, a cholecystokinin-B/gastrin receptor antagonist with high affinity in vitro and high potency in vivo. Mol Pharmacol 1994, 46: 943-8.
-
(1994)
Mol Pharmacol
, vol.46
, pp. 943-948
-
-
Patel, S.1
Smith, A.J.2
Chapman, K.L.3
-
108
-
-
0028290641
-
Pharmacological profile of (R)-1-[2,3-dihydro-1-(2′-methyl-phenacyl)-2-oxo-5-phenyl-1H-1,4- benzodiazepin-3-yl]-3-(3-methylphenyl)urea (YM022), a new potent and selective gastrin/cholecystokinin-B receptor antagonist, in vitro and in vivo
-
Nishida, A., Miyata, K., Tsutsumi, R. et al. Pharmacological profile of (R)-1-[2,3-dihydro-1-(2′-methyl-phenacyl)-2-oxo-5-phenyl-1H-1,4- benzodiazepin-3-yl]-3-(3-methylphenyl)urea (YM022), a new potent and selective gastrin/cholecystokinin-B receptor antagonist, in vitro and in vivo. J Pharmacol Exp Ther 1994, 269: 725-31.
-
(1994)
J Pharmacol Exp Ther
, vol.269
, pp. 725-731
-
-
Nishida, A.1
Miyata, K.2
Tsutsumi, R.3
-
110
-
-
0026092714
-
Rationally designed "dipeptoid" analogues of CCK. Alpha-methyltryptophan derivatives as highly selective and orally active gastrin and CCK-B antagonists with potent anxiolvtic properties
-
Horwell, D.C., Hughes, J., Hunter, J.C. et al. Rationally designed "dipeptoid" analogues of CCK. alpha-methyltryptophan derivatives as highly selective and orally active gastrin and CCK-B antagonists with potent anxiolvtic properties. J Med Chem 1991, 34: 404-14.
-
(1991)
J Med Chem
, vol.34
, pp. 404-414
-
-
Horwell, D.C.1
Hughes, J.2
Hunter, J.C.3
-
111
-
-
15444340232
-
Second generation "peptoid" CCK-B receptor antagonists: Identification and development of N-(adamantyloxycarbonyl)-alpha-methyl-(R)-tryptophan derivative (CI-1015) with an improved pharmacokinetic profile
-
Trivedi, B.K., Padia, J.K., Holmes, A. et al. Second generation "peptoid" CCK-B receptor antagonists: identification and development of N-(adamantyloxycarbonyl)-alpha-methyl-(R)-tryptophan derivative (CI-1015) with an improved pharmacokinetic profile. J Med Chem 1998, 41: 38-45.
-
(1998)
J Med Chem
, vol.41
, pp. 38-45
-
-
Trivedi, B.K.1
Padia, J.K.2
Holmes, A.3
-
112
-
-
0345625367
-
Antisecretory effects of YF476, gastrin/CCK_B receptor antagonist, in beagle dogs with gastric fistula
-
Abst P-405
-
Takemoto, Y. et al. Antisecretory effects of YF476, gastrin/CCK_B receptor antagonist, in beagle dogs with gastric fistula. Jpn J Pharmacol 1997, 73 (Suppl 1): Abst P-405.
-
(1997)
Jpn J Pharmacol
, vol.73
, Issue.1 SUPPL.
-
-
Takemoto, Y.1
-
113
-
-
0030951677
-
YM022, a potent and selective gastrin/CCK-B receptor antagonist, inhibits peptone meal-induced gastric acid secretion in Heidenhain pouch dogs
-
Yuki, H., Nishida, A., Miyake, A. et al. YM022, a potent and selective gastrin/CCK-B receptor antagonist, inhibits peptone meal-induced gastric acid secretion in Heidenhain pouch dogs. Dig Dis Sci 1997, 42: 707-4.
-
(1997)
Dig Dis Sci
, vol.42
, pp. 707-714
-
-
Yuki, H.1
Nishida, A.2
Miyake, A.3
-
114
-
-
15144360265
-
Effects of YF476, a potent and selective gastrin/CCK-B receptor antagonist, on gastric acid secretion in beagle dogs with gastric fistula
-
Takemoto, T., Yuki, H., Nishida, A. Effects of YF476, a potent and selective gastrin/CCK-B receptor antagonist, on gastric acid secretion in beagle dogs with gastric fistula. Arzneim-Forsch Drug Res 1998, 48: 403-7.
-
(1998)
Arzneim-Forsch Drug Res
, vol.48
, pp. 403-407
-
-
Takemoto, T.1
Yuki, H.2
Nishida, A.3
-
115
-
-
0027996070
-
YM022, [(R)-1-]2,3-dihydro-1-(2′-methyl-phenacyl)-2-oxo-5-phenyl-1H-1,4- benzodiazepin-3-yl-3-(3-ethylphenyl)urea, a potent and selective gastrin/cholecystokinin-B receptor antagonist, prevents gastric and duodenal lesions in rats
-
Nishida, A., Takinami, Y., Yuki, H. et al. YM022, [(R)-1-]2,3-dihydro-1-(2′-methyl-phenacyl)-2-oxo-5-phenyl-1H-1,4- benzodiazepin-3-yl]-3-(3-ethylphenyl)urea), a potent and selective gastrin/cholecystokinin-B receptor antagonist, prevents gastric and duodenal lesions in rats. J Pharmacol Exp Ther 1994, 270: 1256-61.
-
(1994)
J Pharmacol Exp Ther
, vol.270
, pp. 1256-1261
-
-
Nishida, A.1
Takinami, Y.2
Yuki, H.3
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