Identification of the cyclosporin-binding site in P-glycoprotein

Biochemistry

Volumn 37, Issue 51, 1998, Pages 18110-18118

  Demeule, Michel ^a   Laplante, Alain ^a   Murphy, Gérard F ^b   Wenger, Roland M ^c   Béliveau, Richard ^a  

^a UNIVERSITÉ DU QUÉBEC À MONTRÉAL   (Canada)

^b Novartis Pharmaceutical Inc   (Canada)

^c NOVARTIS PHARMA AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

2 NITRO 5 THIOCYANATOBENZOIC ACID; AGAROSE; CYANOGEN BROMIDE; CYCLOSPORIN A; DIAZIRINE; GLYCOPROTEIN P; MEMBRANE PROTEIN; N CHLOROSUCCINIMIDE; UNCLASSIFIED DRUG; WHEAT GERM AGGLUTININ;

ANIMAL CELL; ARTICLE; BINDING SITE; CHO CELL; DRUG BINDING; MULTIDRUG RESISTANCE; NONHUMAN; PHOTOAFFINITY LABELING; PREDICTION; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN DEGRADATION; PROTEIN DOMAIN; PROTEIN PURIFICATION;

ANIMALS; AZIRINES; BINDING SITES; CHO CELLS; CRICETINAE; CYCLOSPORINE; CYCLOSPORINS; ELECTROPHORESIS, POLYACRYLAMIDE GEL; MEMBRANE PROTEINS; P-GLYCOPROTEIN; PEPTIDE FRAGMENTS; PHOTOAFFINITY LABELS; SERINE ENDOPEPTIDASES; SUCCINIMIDES; SULFHYDRYL REAGENTS; THIOCYANATES; ULTRAVIOLET RAYS;

EID: 0032559001     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi981992c     Document Type: Article

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