-
1
-
-
0029953826
-
-
1. Plummer, M. S.; Lunney, E. A.; Para, S. K.; Vara Prasad, J. V. N.; Shahripour, A.; Singh, C. J. S.; Humblet, C.; Fergus, J. H.; Marks, J. S.; Sawyer, T. K. Drug Design and Discovery 1996, 13, 75.
-
(1996)
Drug Design and Discovery
, vol.13
, pp. 75
-
-
Plummer, M.S.1
Lunney, E.A.2
Para, S.K.3
Vara Prasad, J.V.N.4
Shahripour, A.5
Singh, C.J.S.6
Humblet, C.7
Fergus, J.H.8
Marks, J.S.9
Sawyer, T.K.10
-
2
-
-
0028346563
-
-
2. Cambier, J. C.; Pleiman, C. M.; Clark, M. R. Annu. Rev. Immunol. 1994, 12, 457.
-
(1994)
Annu. Rev. Immunol.
, vol.12
, pp. 457
-
-
Cambier, J.C.1
Pleiman, C.M.2
Clark, M.R.3
-
3
-
-
0029970787
-
-
3. Kimura, T.; Kihara, H.; Bhattacharyya, S.; Sakamoto, H.; Appella, E.; Siraganian, R. P. J. Biol. Chem. 1996, 271, 27962.
-
(1996)
J. Biol. Chem.
, vol.271
, pp. 27962
-
-
Kimura, T.1
Kihara, H.2
Bhattacharyya, S.3
Sakamoto, H.4
Appella, E.5
Siraganian, R.P.6
-
4
-
-
0030730053
-
-
4. Plummer, M. S.; Holland, D. R.; Shahripour, A.; Lunney, E. A.; Fergus, J. H.; Marks, J. S.; McConnell, B.; Mueller, W. T.; Sawyer, T. K. J. Med. Chem. 1997, 40, 3719.
-
(1997)
J. Med. Chem.
, vol.40
, pp. 3719
-
-
Plummer, M.S.1
Holland, D.R.2
Shahripour, A.3
Lunney, E.A.4
Fergus, J.H.5
Marks, J.S.6
McConnell, B.7
Mueller, W.T.8
Sawyer, T.K.9
-
5
-
-
0026793591
-
-
5. (a) Domchek, S. M.; Auger, K. R.; Chatterjee, S.; Burke, Jr., T. R.; Shoelson, S. E.; Biochemistry, 1992, 31, 9865.
-
(1992)
Biochemistry
, vol.31
, pp. 9865
-
-
Domchek, S.M.1
Auger, K.R.2
Chatterjee, S.3
Burke T.R., Jr.4
Shoelson, S.E.5
-
6
-
-
0028985602
-
-
(b) Wange, R. L.; Isakov, N.; Burke, Jr., T. R.; Otaka, A.; Roller, P. P.; Watts, J. D.; Aebersold, R.; Samelson, L. E. J. Biol. Chem. 1995, 270, 944.
-
(1995)
J. Biol. Chem.
, vol.270
, pp. 944
-
-
Wange, R.L.1
Isakov, N.2
Burke T.R., Jr.3
Otaka, A.4
Roller, P.P.5
Watts, J.D.6
Aebersold, R.7
Samelson, L.E.8
-
7
-
-
0028985602
-
-
(c) Wange, R. L.; Isakov, N.; Burke, Jr., T. R.; Otaka, A.; Roller, P. P.; Watts, J. D.; Aebersold, R.; Samelson, L. E. J. Biol. Chem. 1995, 270, 944.
-
(1995)
J. Biol. Chem.
, vol.270
, pp. 944
-
-
Wange, R.L.1
Isakov, N.2
Burke T.R., Jr.3
Otaka, A.4
Roller, P.P.5
Watts, J.D.6
Aebersold, R.7
Samelson, L.E.8
-
8
-
-
17644445390
-
-
(d) Plummer, M. S.; Lunney, E. A.; Para, K. S.; Shahripour, A.; Stankovic, C. J.; Humblet, C.; Fergus, J. H.; Saltiel, A.; Sawyer, T. K. Bioorg. Med. Chem. 1997, 5, 41.
-
(1997)
Bioorg. Med. Chem.
, vol.5
, pp. 41
-
-
Plummer, M.S.1
Lunney, E.A.2
Para, K.S.3
Shahripour, A.4
Stankovic, C.J.5
Humblet, C.6
Fergus, J.H.7
Saltiel, A.8
Sawyer, T.K.9
-
9
-
-
0030725743
-
-
(e) Furet, P.; Gay, B.; G-Echeverria, C.; Rahuel, J.; Fretz, H.; Schoepfer, J.; Caravatti, G. J. Med. Chem. 1997, 40, 3551.
-
(1997)
J. Med. Chem.
, vol.40
, pp. 3551
-
-
Furet, P.1
Gay, B.2
G-Echeverria, C.3
Rahuel, J.4
Fretz, H.5
Schoepfer, J.6
Caravatti, G.7
-
10
-
-
0030697349
-
-
(f) Revesz, L.; Blum, E.; Manning, U.; Demange, B. J.; Widmer, A.; Zuber, J.-F. Bioorg. Med. Chem. Lett. 1997, 7, 2875.
-
(1997)
Bioorg. Med. Chem. Lett.
, vol.7
, pp. 2875
-
-
Revesz, L.1
Blum, E.2
Manning, U.3
Demange, B.J.4
Widmer, A.5
Zuber, J.-F.6
-
11
-
-
0028308838
-
-
6. (a) Burke, Jr., T. R.; Smyth, M. S.; Otaka, A.; Nomizu, M.; Roller, P. P.; Wolf, G.; Case, R.; Shoelson, S. E. Biochemistry 1994, 33, 6490.
-
(1994)
Biochemistry
, vol.33
, pp. 6490
-
-
Burke T.R., Jr.1
Smyth, M.S.2
Otaka, A.3
Nomizu, M.4
Roller, P.P.5
Wolf, G.6
Case, R.7
Shoelson, S.E.8
-
12
-
-
0027316389
-
-
(b) Burke, Jr., Smyth, M. S.; Otaka, A.; Roller, P. P. Tetrahedron Lett. 1993, 34, 4125.
-
(1993)
Tetrahedron Lett.
, vol.34
, pp. 4125
-
-
Burke, Jr.1
Smyth, M.S.2
Otaka, A.3
Roller, P.P.4
-
13
-
-
0031584893
-
-
2 has also been attributed to a direct interaction of the fluorines with active site residues and not to lower pKa values, see: Chen, L.; Wu, L.; Otaka, A.; Smith, M. S.; Roller, P. R.; Burke, T. R.; den Hertog, J.; Zhang, Z-Y. Biochem. Biophys. Res. Comm. 1995, 216, 976.
-
(1997)
Tetrahedron Lett.
, vol.38
, pp. 1389
-
-
Liu, W.-Q.1
Roques, B.P.2
Garbay, C.3
-
14
-
-
0028785789
-
-
2 has also been attributed to a direct interaction of the fluorines with active site residues and not to lower pKa values, see: Chen, L.; Wu, L.; Otaka, A.; Smith, M. S.; Roller, P. R.; Burke, T. R.; den Hertog, J.; Zhang, Z-Y. Biochem. Biophys. Res. Comm. 1995, 216, 976.
-
(1995)
Biochem. Biophys. Res. Comm.
, vol.216
, pp. 976
-
-
Chen, L.1
Wu, L.2
Otaka, A.3
Smith, M.S.4
Roller, P.R.5
Burke, T.R.6
Den Hertog, J.7
Zhang, Z.-Y.8
-
15
-
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0010401786
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note
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A2 were subsequently calculated as 7.1 and 7.7 ± 0.3, respectively, using Advanced Chemistry Development, Inc., prediction software.
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-
-
-
16
-
-
0027409064
-
-
8. (a) Waksman, G.; Shoelson, S. E.; Pant, N.; Cowburn, D.; Kuriyan, J. Cell 1993, 72, 779.
-
(1993)
Cell
, vol.72
, pp. 779
-
-
Waksman, G.1
Shoelson, S.E.2
Pant, N.3
Cowburn, D.4
Kuriyan, J.5
-
17
-
-
0027502504
-
-
(b) Eck, M. J.; Shoelson, S. E.; Harrison, S. C. Nature 1993, 362, 87.
-
(1993)
Nature
, vol.362
, pp. 87
-
-
Eck, M.J.1
Shoelson, S.E.2
Harrison, S.C.3
-
18
-
-
0000324835
-
-
9. Kelly, T. R.; Bridger, G. J.; Zhao, C. J. Am. Chem. Soc. 1990, 112, 8024.
-
(1990)
J. Am. Chem. Soc.
, vol.112
, pp. 8024
-
-
Kelly, T.R.1
Bridger, G.J.2
Zhao, C.3
-
19
-
-
0028206694
-
-
10. A similar approach to the synthesis of 4-phosphono(difluoromethyl)-L-phenylalanine and pyridylalanine regioisomers starting from 2-, 3-and 4-bromopyridine and β-iodoalanine have been described, see: (a) Smyth, M. S.; Burke, Jr., T. R. Tetrahedron Lett. 1994, 35, 551
-
(1994)
Tetrahedron Lett.
, vol.35
, pp. 551
-
-
Smyth, M.S.1
Burke T.R., Jr.2
-
20
-
-
0039267611
-
-
(b) Walker, M. A.; Kaplita, K. P.; Chen, T.; King, H. D. Synlett 1997, 169.
-
(1997)
Synlett
, pp. 169
-
-
Walker, M.A.1
Kaplita, K.P.2
Chen, T.3
King, H.D.4
-
22
-
-
0010317879
-
Peptidomimetic inhibitors of the association of platelet derived growth factor-β receptor with phosphatidylinositiol 3-kinase
-
Ann Arbor Michigan, June
-
th National Medicinal Chemistry Symposium, Ann Arbor Michigan, June 18-22.
-
th National Medicinal Chemistry Symposium
, pp. 18-22
-
-
Eaton, S.R.1
Cody, W.L.2
Kent, D.R.3
Paneck, R.L.4
Lu, G.H.5
Dahring, T.K.6
Doherty, A.M.7
-
23
-
-
0029945906
-
-
13. Szardenings, A. K.; Gordeev, M. F.; Patel, D. V. Tetrahedron Lett. 1996, 37, 3635.
-
(1996)
Tetrahedron Lett.
, vol.37
, pp. 3635
-
-
Szardenings, A.K.1
Gordeev, M.F.2
Patel, D.V.3
-
24
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-
0010317705
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note
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++1).
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