Efficient synthesis of substituted oxopiperazines from amino acids

Tetrahedron Letters

Volumn 39, Issue 45, 1998, Pages 8213-8216

  Mohamed, Nazim ^a   Bhatt, Ulhas ^a   Just, George ^a  

^a MCGILL UNIVERSITY   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

OXOPIPERAZINE DERIVATIVE; PIPERAZINE DERIVATIVE; SULFONAMIDE; UNCLASSIFIED DRUG;

ARTICLE; CYCLIZATION; DRUG SYNTHESIS; REACTION ANALYSIS; SOLID PHASE EXTRACTION;

EID: 0032487873     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(98)01878-4     Document Type: Article

References (10)

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2. (b) Goodfellow, V. S.; Laudeman, C. P.; Gerrity, J. L.; Burkard, M.; Strobel, E.; Zuzack, J. S.; McLeod, D. A., Mol. Div. 1996, 2, 97.
3. 2. Bhatt, U.; Mohamed, N.; Just, G.; Roberts, E., Tetrahedron Lett. 1997, 38, 3679.
4. 3. Pohlmann, A.; Schanen, V.; Guillaume, D.; Quirion, J.-C.; Husson, H.-P., J. Org. Chem. 1997, 62, 1016.
5. 4. Gante, J.; Neunhoeffer, H.; Schmidt, A., J. Org. Chem. 1994, 59, 6487.
6. 5. Lindner, E.; Von Au, G.; Eberle, H.-J., Chem. Ber. 1981, 114, 810.
7. 6. Fukuyama, T.; Jow, C. K.; Cheung, M., Tetrahedron Lett. 1995, 36, 6373.
8. 13C NMR spectra as well as correct mass spectra.
9. 8. Barlos, K.; Gatos, D.; Kallitsis, J.; Papaphotiu, G.; Sotiriu, P.; Wenqing, Y.; Schäfer, W., Tetrahedron Lett. 1989, 30, 3943.
10. 9. Structures of all solid phase reaction products were confirmed by LCMS.