Heterologous expression of the cloned guinea pig α2A, α2B, and α2C adrenoceptor subtypes: Radioligand binding and functional coupling to a cAMP-responsive reporter gene

Biochemical Pharmacology

Volumn 51, Issue 3, 1996, Pages 291-300

  Svensson, Samuel P S ^a   Bailey, Thomas J ^a   Porter, Amy C ^a   Richman, Jeremy G ^a   Regan, John W ^a  

^a UNIVERSITY OF ARIZONA   (United States)

Author keywords

Adenylyl cyclase; G protein coupled; Pharmacology; Reporter gene

Indexed keywords

1,3,4,5',6,6',7,12B OCTAHYDRO 1',3' DIMETHYL 2H SPIRO[BENZO[B]FURO[2,3 A]QUINOLIZINE 2,4' PYRIMIDINE] 2' ONE; 6 CHLORO 2,3,4,5 TETRAHYDRO 3 METHYL 9 (3 METHYL 2 BUTENYLOXY) 1H 3 BENZAZEPINE; ADENYLATE CYCLASE; ALPHA 2 ADRENERGIC RECEPTOR; ALPHA 2A ADRENERGIC RECEPTOR; ALPHA 2B ADRENERGIC RECEPTOR; ALPHA 2C ADRENERGIC RECEPTOR; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA ADRENERGIC RECEPTOR STIMULATING AGENT; ATIPAMEZOLE; CHLORAMPHENICOL ACETYLTRANSFERASE; CHLORPROMAZINE; CLONIDINE; COMPLEMENTARY DNA; DEXMEDETOMIDINE; FORSKOLIN; GUANINE NUCLEOTIDE BINDING PROTEIN; MESSENGER RNA; NORADRENALIN; OLIGONUCLEOTIDE; OXYMETAZOLINE; PHENTOLAMINE; PRAZOSIN; RADIOLIGAND; RECEPTOR SUBTYPE; YOHIMBINE;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING COMPETITION; CONTROLLED STUDY; DNA LIBRARY; DRUG RECEPTOR BINDING; ENZYME ACTIVITY; GENE EXPRESSION; GENE SEQUENCE; GENOME; GUINEA PIG; HUMAN; MAMMAL CELL; MOLECULAR CLONING; NONHUMAN; POLYMERASE CHAIN REACTION; PRIORITY JOURNAL; REPORTER GENE;

ADRENERGIC ALPHA-ANTAGONISTS; AMINO ACID SEQUENCE; ANIMALS; BASE SEQUENCE; BENZAZEPINES; BINDING, COMPETITIVE; CLONING, MOLECULAR; CYCLIC AMP RESPONSE ELEMENT-BINDING PROTEIN; GENE EXPRESSION; GENES, REPORTER; GUINEA PIGS; MOLECULAR SEQUENCE DATA; QUINOLIZINES; RADIOLIGAND ASSAY; RECEPTORS, ADRENERGIC, ALPHA; SEQUENCE ALIGNMENT;

EID: 0030040778     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/0006-2952(95)02179-5     Document Type: Article

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