Salmeterol-induced desensitization, internalization and phosphorylation of the human β2-adrenoceptor

British Journal of Pharmacology

Volumn 123, Issue 4, 1998, Pages 701-711

  January, Bridgette ^a   Seibold, Anita ^a   Allal, Chafika ^a   Whaley, Brenda S ^a   Knoll, Brian J ^b   Moore, Robert H ^b   Dickey, Burton F ^b   Barber, Roger ^a   Clark, Richard B ^a  

^a UNIVERSITY OF TEXAS   (United States)

^b BAYLOR COLLEGE OF MEDICINE   (United States)

Author keywords

Desensitization; Internalization; Phosphorylation; Salmeterol; 2 adrenoceptor

Indexed keywords

ADENYLATE CYCLASE; ADRENALIN; BETA 2 ADRENERGIC RECEPTOR; BETA ADRENERGIC RECEPTOR STIMULATING AGENT; DRUG DERIVATIVE; SALBUTAMOL; SALMETEROL;

ARTICLE; CELL LINE; DRUG POTENTIATION; ENDOCYTOSIS; ENZYME ACTIVATION; HUMAN; METABOLISM; PHOSPHORYLATION;

ADENYLATE CYCLASE; ADRENERGIC BETA-AGONISTS; ALBUTEROL; CELL LINE; ENDOCYTOSIS; ENZYME ACTIVATION; EPINEPHRINE; HUMANS; PHOSPHORYLATION; RECEPTORS, ADRENERGIC, BETA-2;

EID: 0031990692     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701658     Document Type: Article

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