Synthesis and evaluation of 1,5-benzodiazepines with bridged cycloalkyl substituents at the N-1 position as potent and selective CCK-B ligands

Archiv der Pharmazie

Volumn 331, Issue 1, 1998, Pages 41-44

  Finizia, Gabriella ^a   Donati, Daniele ^a   Pentassuglia, Giorgio ^a   Polinelli, Stefano ^a   Tarzia, Giorgio ^a,b   Tranquillini, Maria Elvira ^a   Ursini, Antonella ^a  

^a GSK   (Italy)

^b UNIVERSITY OF URBINO   (Italy)

Author keywords

1,5 benzodiazepines; CCK A; CCK B

Indexed keywords

ADAMANTANE DERIVATIVE; BENZODIAZEPINE DERIVATIVE; CHOLECYSTOKININ A RECEPTOR; CHOLECYSTOKININ B RECEPTOR; NORBORNANE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GUINEA PIG; IN VITRO STUDY; NONHUMAN; PANCREAS; PRIORITY JOURNAL; RACEMIC MIXTURE; RAT; RECEPTOR AFFINITY;

EID: 0031884364     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1521-4184(199801)331:1<41::AID-ARDP41>3.0.CO;2-S     Document Type: Article

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