Novel 1,5-benzodiazepines as CCK-B ligands. Effect of aryl-carbamic substituents at the C-3 position together with halogen substitution on the benzo-fused ring

Archiv der Pharmazie

Volumn 330, Issue 11, 1997, Pages 353-357

  Tranquillini, M Elvira ^b   Cassarà, Paolo G ^b   Corsi, Mauro ^b   Curotto, Giovanni ^b   Donati, Daniele ^b   Finizia, Gabriella ^b   Pentassuglia, Giorgio ^b   Polinelli, Stefano ^b   Tarzia, Giorgio ^a,b   Ursini, Antonella ^b   Van Amsterdam, Franciscus T M ^b  

^a UNIVERSITY OF URBINO   (Italy)

^b GSK   (Italy)

Author keywords

1,5 Benzodiazepines; Cholecystokinin A (CCK A); Cholecystokinin B (CCK B)

Indexed keywords

BENZODIAZEPINE DERIVATIVE; CHOLECYSTOKININ A RECEPTOR; CHOLECYSTOKININ B RECEPTOR; LIGAND; RECEPTOR SUBUNIT;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BRAIN; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GUINEA PIG; IN VITRO STUDY; INFRARED SPECTROPHOTOMETRY; MASS SPECTROMETRY; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PANCREAS; PRIORITY JOURNAL; RAT; STRUCTURE ACTIVITY RELATION;

EID: 0030667395     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/ardp.19973301107     Document Type: Article

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